MX2024012493A - Nuevos compuestos de proteina 1 de transicion de fase g1 a s (gspt1) y metodos de uso de los nuevos compuestos - Google Patents

Nuevos compuestos de proteina 1 de transicion de fase g1 a s (gspt1) y metodos de uso de los nuevos compuestos

Info

Publication number
MX2024012493A
MX2024012493A MX2024012493A MX2024012493A MX2024012493A MX 2024012493 A MX2024012493 A MX 2024012493A MX 2024012493 A MX2024012493 A MX 2024012493A MX 2024012493 A MX2024012493 A MX 2024012493A MX 2024012493 A MX2024012493 A MX 2024012493A
Authority
MX
Mexico
Prior art keywords
compounds
novel
methods
gspt1
cancer
Prior art date
Application number
MX2024012493A
Other languages
English (en)
Spanish (es)
Inventor
Joshua Hansen
Mimi L Quan
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of MX2024012493A publication Critical patent/MX2024012493A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • A61K31/4523Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/454Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Oncology (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
MX2024012493A 2022-04-14 2024-10-09 Nuevos compuestos de proteina 1 de transicion de fase g1 a s (gspt1) y metodos de uso de los nuevos compuestos MX2024012493A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US202263331193P 2022-04-14 2022-04-14
PCT/US2023/065699 WO2023201282A1 (en) 2022-04-14 2023-04-13 Novel gspt1 compounds and methods of use of the novel compounds

Publications (1)

Publication Number Publication Date
MX2024012493A true MX2024012493A (es) 2024-11-08

Family

ID=86329395

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2024012493A MX2024012493A (es) 2022-04-14 2024-10-09 Nuevos compuestos de proteina 1 de transicion de fase g1 a s (gspt1) y metodos de uso de los nuevos compuestos

Country Status (12)

Country Link
US (2) US12187699B2 (https=)
EP (1) EP4508044A1 (https=)
JP (1) JP2025513877A (https=)
KR (1) KR20250003774A (https=)
CN (1) CN119013266A (https=)
AR (1) AR129053A1 (https=)
AU (1) AU2023252917A1 (https=)
CA (1) CA3255290A1 (https=)
IL (1) IL316238A (https=)
MX (1) MX2024012493A (https=)
TW (1) TW202406901A (https=)
WO (1) WO2023201282A1 (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2025085416A1 (en) * 2023-10-16 2025-04-24 Bristol-Myers Squibb Company Gspt1 compounds and methods of use of the compounds
WO2026077418A1 (zh) * 2024-10-11 2026-04-16 上海海雁医药科技有限公司 含苯乙氧基亚烷基胺结构的异吲哚啉化合物及其偶联物和用途

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Also Published As

Publication number Publication date
WO2023201282A1 (en) 2023-10-19
TW202406901A (zh) 2024-02-16
CA3255290A1 (en) 2023-10-19
AR129053A1 (es) 2024-07-10
CN119013266A (zh) 2024-11-22
EP4508044A1 (en) 2025-02-19
JP2025513877A (ja) 2025-04-30
AU2023252917A1 (en) 2024-11-28
US20230331693A1 (en) 2023-10-19
US20250092012A1 (en) 2025-03-20
IL316238A (en) 2024-12-01
US12187699B2 (en) 2025-01-07
KR20250003774A (ko) 2025-01-07

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