MX2024008821A - Formas solidas cristalinas de inhibidores de la helicasa-primasa y proceso de preparacion de las mismas. - Google Patents

Formas solidas cristalinas de inhibidores de la helicasa-primasa y proceso de preparacion de las mismas.

Info

Publication number
MX2024008821A
MX2024008821A MX2024008821A MX2024008821A MX2024008821A MX 2024008821 A MX2024008821 A MX 2024008821A MX 2024008821 A MX2024008821 A MX 2024008821A MX 2024008821 A MX2024008821 A MX 2024008821A MX 2024008821 A MX2024008821 A MX 2024008821A
Authority
MX
Mexico
Prior art keywords
helicase
crystalline forms
solid crystalline
preparation
primase inhibitors
Prior art date
Application number
MX2024008821A
Other languages
English (en)
Spanish (es)
Inventor
Christian Gege
Gerald Kleymann
Original Assignee
Innovative Molecules Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Innovative Molecules Gmbh filed Critical Innovative Molecules Gmbh
Publication of MX2024008821A publication Critical patent/MX2024008821A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/54Nitrogen and either oxygen or sulfur atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/4261,3-Thiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/20Antivirals for DNA viruses
    • A61P31/22Antivirals for DNA viruses for herpes viruses
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B59/00Introduction of isotopes of elements into organic compounds ; Labelled organic compounds per se
    • C07B59/002Heterocyclic compounds
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13Crystalline forms, e.g. polymorphs

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Virology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Communicable Diseases (AREA)
  • Engineering & Computer Science (AREA)
  • Biotechnology (AREA)
  • Molecular Biology (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
MX2024008821A 2022-01-17 2023-01-16 Formas solidas cristalinas de inhibidores de la helicasa-primasa y proceso de preparacion de las mismas. MX2024008821A (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP22151820 2022-01-17
EP22170332 2022-04-27
PCT/EP2023/050883 WO2023135303A1 (en) 2022-01-17 2023-01-16 Solid crystalline forms of helicase-primase inhibitors and process of preparation thereof

Publications (1)

Publication Number Publication Date
MX2024008821A true MX2024008821A (es) 2024-07-29

Family

ID=84982261

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2024008821A MX2024008821A (es) 2022-01-17 2023-01-16 Formas solidas cristalinas de inhibidores de la helicasa-primasa y proceso de preparacion de las mismas.

Country Status (13)

Country Link
US (1) US20250115565A1 (https=)
EP (1) EP4466255A1 (https=)
JP (1) JP2025502300A (https=)
KR (1) KR20240134979A (https=)
AU (1) AU2023206628A1 (https=)
CA (1) CA3246779A1 (https=)
CL (1) CL2024002124A1 (https=)
IL (1) IL314188A (https=)
MX (1) MX2024008821A (https=)
PY (1) PY2302301A (https=)
TW (1) TW202337444A (https=)
UY (1) UY40111A (https=)
WO (1) WO2023135303A1 (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL319024A (en) * 2022-08-29 2025-04-01 Assembly Biosciences Inc Pharmaceutical preparations for the herpes virus
IL325911A (en) 2023-07-17 2026-03-01 Innovative Molecules Gmbh Micronized crystalline hydrochloride salts of antiviral helicase-primase inhibitor compounds
WO2026078039A1 (en) 2024-10-09 2026-04-16 Innovative Molecules Gmbh Oral administration forms of antiviral helicase-primase inhibitors

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DOP2000000109A (es) 1999-12-23 2002-08-30 Gerald Kleymann Derivados de tiazolilamida
DE10131128A1 (de) 2001-06-28 2003-01-16 Bayer Ag Sekundäre Sulfonamide
GEP20207128B (en) 2016-04-06 2020-07-10 Molecules Gm Innovative Aminothiazole derivatives useful as antiviral agents
MX2020003369A (es) 2017-10-05 2020-07-29 Innovative Molecules Gmbh Enantiomeros de tiazoles sustituidos como compuestos antivirales.
TW202038947A (zh) 2018-11-28 2020-11-01 德商創新分子有限責任公司 在與溶瘤病毒之組合療法中治療癌症的解旋酶引子酶抑制劑
KR20230131177A (ko) 2020-10-29 2023-09-12 이노베이티브 몰리큘스 게엠베하 항바이러스 화합물로서 중수소화된 아미노티아졸 화합물

Also Published As

Publication number Publication date
KR20240134979A (ko) 2024-09-10
WO2023135303A1 (en) 2023-07-20
US20250115565A1 (en) 2025-04-10
PY2302301A (es) 2023-10-31
TW202337444A (zh) 2023-10-01
UY40111A (es) 2023-08-15
CA3246779A1 (en) 2023-07-20
IL314188A (en) 2024-09-01
AU2023206628A1 (en) 2024-08-01
EP4466255A1 (en) 2024-11-27
JP2025502300A (ja) 2025-01-24
CL2024002124A1 (es) 2024-11-22

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