MX2024005656A - Inhibidores de proteina tirosina fosfatasa y metodos de uso de estos. - Google Patents

Inhibidores de proteina tirosina fosfatasa y metodos de uso de estos.

Info

Publication number
MX2024005656A
MX2024005656A MX2024005656A MX2024005656A MX2024005656A MX 2024005656 A MX2024005656 A MX 2024005656A MX 2024005656 A MX2024005656 A MX 2024005656A MX 2024005656 A MX2024005656 A MX 2024005656A MX 2024005656 A MX2024005656 A MX 2024005656A
Authority
MX
Mexico
Prior art keywords
methods
protein tyrosine
tyrosine phosphatase
phosphatase inhibitors
agents
Prior art date
Application number
MX2024005656A
Other languages
English (en)
Spanish (es)
Inventor
Andrew Bogdan
Jennifer M Frost
Philip R Kym
Zhaoming Xiong
Christos Economou
Spencer O Scholz
Original Assignee
Calico Life Sciences Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Calico Life Sciences Llc filed Critical Calico Life Sciences Llc
Publication of MX2024005656A publication Critical patent/MX2024005656A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/433—Thidiazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
MX2024005656A 2021-11-11 2022-11-10 Inhibidores de proteina tirosina fosfatasa y metodos de uso de estos. MX2024005656A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US202163278336P 2021-11-11 2021-11-11
PCT/US2022/049581 WO2023086495A1 (en) 2021-11-11 2022-11-10 Protein tyrosine phosphatase inhibitors and methods of use thereof

Publications (1)

Publication Number Publication Date
MX2024005656A true MX2024005656A (es) 2024-08-06

Family

ID=84887566

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2024005656A MX2024005656A (es) 2021-11-11 2022-11-10 Inhibidores de proteina tirosina fosfatasa y metodos de uso de estos.

Country Status (8)

Country Link
US (1) US20250042894A1 (enExample)
EP (1) EP4430039A1 (enExample)
JP (1) JP2024543451A (enExample)
CN (1) CN118556055A (enExample)
AU (1) AU2022386164A1 (enExample)
CA (1) CA3236853A1 (enExample)
MX (1) MX2024005656A (enExample)
WO (1) WO2023086495A1 (enExample)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2024243441A1 (en) 2023-05-24 2024-11-28 Kumquat Biosciences Inc. Heterocyclic compounds and uses thereof

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
UA94921C2 (en) * 2005-12-08 2011-06-25 Новартис Аг 1-orthofluorophenyl substituted 1, 2, 5-thiazolidinedione derivatives as ptp-as inhibitors
TWI888352B (zh) * 2018-06-21 2025-07-01 美商嘉來克生命科學有限責任公司 蛋白質酪胺酸磷酸酯酶抑制劑及其使用方法
KR102983496B1 (ko) * 2019-03-14 2026-06-29 칼리코 라이프 사이언시스 엘엘씨 단백질 티로신 포스파타제 억제제 및 이의 사용 방법
MX2022007441A (es) * 2019-12-18 2022-09-02 Calico Life Sciences Llc Inhibidores de proteína tirosina fosfatasa y sus métodos de uso.

Also Published As

Publication number Publication date
AU2022386164A1 (en) 2024-05-23
CN118556055A (zh) 2024-08-27
JP2024543451A (ja) 2024-11-21
EP4430039A1 (en) 2024-09-18
CA3236853A1 (en) 2023-05-19
US20250042894A1 (en) 2025-02-06
WO2023086495A1 (en) 2023-05-19

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