MX2023013557A - Pauta posologica de sotorasib. - Google Patents
Pauta posologica de sotorasib.Info
- Publication number
- MX2023013557A MX2023013557A MX2023013557A MX2023013557A MX2023013557A MX 2023013557 A MX2023013557 A MX 2023013557A MX 2023013557 A MX2023013557 A MX 2023013557A MX 2023013557 A MX2023013557 A MX 2023013557A MX 2023013557 A MX2023013557 A MX 2023013557A
- Authority
- MX
- Mexico
- Prior art keywords
- sotorasib
- dosing regimen
- cancer
- patient
- kras
- Prior art date
Links
- NXQKSXLFSAEQCZ-SFHVURJKSA-N sotorasib Chemical compound FC1=CC2=C(N(C(N=C2N2[C@H](CN(CC2)C(C=C)=O)C)=O)C=2C(=NC=CC=2C)C(C)C)N=C1C1=C(C=CC=C1O)F NXQKSXLFSAEQCZ-SFHVURJKSA-N 0.000 title abstract 2
- 229940073531 sotorasib Drugs 0.000 title abstract 2
- 206010028980 Neoplasm Diseases 0.000 abstract 2
- 201000011510 cancer Diseases 0.000 abstract 2
- 208000003174 Brain Neoplasms Diseases 0.000 abstract 1
- 206010059282 Metastases to central nervous system Diseases 0.000 abstract 1
- 230000035772 mutation Effects 0.000 abstract 1
- 102200006538 rs121913530 Human genes 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
- Medicines Containing Material From Animals Or Micro-Organisms (AREA)
Abstract
Se proporcionan en la presente métodos para tratar un cáncer que comprende una mutación en KRAS G12C en un paciente con metástasis cerebrales activas, que comprende administrar sotorasib al paciente en la cantidad efectiva para tratar el cáncer.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US202163190061P | 2021-05-18 | 2021-05-18 | |
PCT/US2022/029677 WO2022245857A1 (en) | 2021-05-18 | 2022-05-17 | Sotorasib dosing regimen |
Publications (1)
Publication Number | Publication Date |
---|---|
MX2023013557A true MX2023013557A (es) | 2023-11-29 |
Family
ID=82019614
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MX2023013557A MX2023013557A (es) | 2021-05-18 | 2022-05-17 | Pauta posologica de sotorasib. |
Country Status (7)
Country | Link |
---|---|
EP (1) | EP4340842A1 (es) |
JP (1) | JP2024519060A (es) |
CN (1) | CN117355306A (es) |
AU (1) | AU2022277860A1 (es) |
CA (1) | CA3218575A1 (es) |
MX (1) | MX2023013557A (es) |
WO (1) | WO2022245857A1 (es) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2024072437A1 (en) * | 2022-09-30 | 2024-04-04 | Amgen Inc. | Sotorasib dosing regimen |
-
2022
- 2022-05-17 JP JP2023571589A patent/JP2024519060A/ja active Pending
- 2022-05-17 CA CA3218575A patent/CA3218575A1/en active Pending
- 2022-05-17 EP EP22729925.2A patent/EP4340842A1/en active Pending
- 2022-05-17 AU AU2022277860A patent/AU2022277860A1/en active Pending
- 2022-05-17 CN CN202280035539.3A patent/CN117355306A/zh active Pending
- 2022-05-17 MX MX2023013557A patent/MX2023013557A/es unknown
- 2022-05-17 WO PCT/US2022/029677 patent/WO2022245857A1/en active Application Filing
Also Published As
Publication number | Publication date |
---|---|
CA3218575A1 (en) | 2022-11-24 |
CN117355306A (zh) | 2024-01-05 |
WO2022245857A1 (en) | 2022-11-24 |
EP4340842A1 (en) | 2024-03-27 |
JP2024519060A (ja) | 2024-05-08 |
AU2022277860A1 (en) | 2023-12-07 |
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