MX2023004046A - Proceso para la preparacion de esteres, amidas y nitrilos de acido 5-(1-cianociclopropil)-piridin-2-carboxilico. - Google Patents

Proceso para la preparacion de esteres, amidas y nitrilos de acido 5-(1-cianociclopropil)-piridin-2-carboxilico.

Info

Publication number
MX2023004046A
MX2023004046A MX2023004046A MX2023004046A MX2023004046A MX 2023004046 A MX2023004046 A MX 2023004046A MX 2023004046 A MX2023004046 A MX 2023004046A MX 2023004046 A MX2023004046 A MX 2023004046A MX 2023004046 A MX2023004046 A MX 2023004046A
Authority
MX
Mexico
Prior art keywords
preparation
cyanocyclopropyl
nitriles
pyridine
carboxylic acid
Prior art date
Application number
MX2023004046A
Other languages
English (en)
Inventor
Martin Pouliot
Raphael Dumeunier
Renaud Beaudegnies
Alexander Gaspers
Original Assignee
Syngenta Crop Protection Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syngenta Crop Protection Ag filed Critical Syngenta Crop Protection Ag
Publication of MX2023004046A publication Critical patent/MX2023004046A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/84—Nitriles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/62—Oxygen or sulfur atoms
    • C07D213/70—Sulfur atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/79—Acids; Esters
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/79—Acids; Esters
    • C07D213/803—Processes of preparation
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/81—Amides; Imides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pyridine Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Se proporciona un proceso para la preparación del compuesto de fórmula I: (ver Fórmula) (I) donde R1 y R2 son tal como se definen en la descripción.
MX2023004046A 2020-10-09 2021-10-08 Proceso para la preparacion de esteres, amidas y nitrilos de acido 5-(1-cianociclopropil)-piridin-2-carboxilico. MX2023004046A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP20201119 2020-10-09
PCT/EP2021/077899 WO2022074214A1 (en) 2020-10-09 2021-10-08 Process for the preparation of 5-(1-cyanocyclopropyl)-pyridine-2-carboxylic acid esters amides and nitriles

Publications (1)

Publication Number Publication Date
MX2023004046A true MX2023004046A (es) 2023-04-27

Family

ID=72826783

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2023004046A MX2023004046A (es) 2020-10-09 2021-10-08 Proceso para la preparacion de esteres, amidas y nitrilos de acido 5-(1-cianociclopropil)-piridin-2-carboxilico.

Country Status (10)

Country Link
US (1) US20230382866A1 (es)
EP (1) EP4225736A1 (es)
JP (1) JP2023544212A (es)
KR (1) KR20230084531A (es)
CN (1) CN116390911A (es)
CA (1) CA3195005A1 (es)
IL (1) IL301686A (es)
MX (1) MX2023004046A (es)
TW (1) TW202229238A (es)
WO (1) WO2022074214A1 (es)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2023194496A1 (en) * 2022-04-07 2023-10-12 Syngenta Crop Protection Ag Process for the preparation of diversely substituted cyanocyclopropyl - heteroarenes or arenes

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8536299B2 (en) 2008-12-08 2013-09-17 University Of Dayton Rigid-rod copolymer compositions and the polymeric fibers fabricated from those compositions for enhanced flame resistance
US8912221B2 (en) 2010-12-27 2014-12-16 Hoffmann-La Roche Inc. Biaryl amide derivatives
EP3227284B1 (en) 2014-12-01 2021-04-28 Syngenta Participations AG Pesticidally active amide heterocyclic derivatives with sulphur containing substituents
TWI696612B (zh) 2015-01-29 2020-06-21 日商日本農藥股份有限公司 具有環烷基吡啶基的稠合雜環化合物或其鹽類及含有該化合物的農園藝用殺蟲劑以及其使用方法
CN105218437A (zh) 2015-10-31 2016-01-06 高大元 一种3-氯-5-溴-2-吡啶甲酸的合成方法
JP2018012664A (ja) * 2016-07-21 2018-01-25 日本農薬株式会社 シクロアルキル基を有するピリジン誘導体及び該誘導体を含有する有害生物防除剤及びその使用方法
BR112019012127A2 (pt) * 2016-12-15 2019-11-05 Syngenta Participations Ag derivados heterocíclicos ativos em termos pesticidas com substituintes contendo enxofre
WO2019059244A1 (ja) 2017-09-21 2019-03-28 日本農薬株式会社 シクロプロピルピリジル基を有するベンゾイミダゾール化合物又はその塩類、及びそれらの化合物を含有する農園芸用殺虫剤並びにその使用方法
CN112262140B (zh) * 2018-06-06 2024-05-28 先正达农作物保护股份公司 具有含亚砜亚胺取代基的杀有害生物活性杂环衍生物
MX2021003741A (es) 2018-10-02 2021-05-14 Nippon Soda Co Compuesto de heteroaril-azolo y agente de control de plagas.
IL282553B2 (en) 2018-10-29 2024-06-01 Nippon Soda Co A (hetero)arylimidazole compound and a pest control agent
JP2020079325A (ja) 2020-03-02 2020-05-28 住友化学株式会社 複素環化合物を用いる有害節足動物防除方法

Also Published As

Publication number Publication date
EP4225736A1 (en) 2023-08-16
CA3195005A1 (en) 2022-04-14
CN116390911A (zh) 2023-07-04
TW202229238A (zh) 2022-08-01
KR20230084531A (ko) 2023-06-13
IL301686A (en) 2023-05-01
JP2023544212A (ja) 2023-10-20
US20230382866A1 (en) 2023-11-30
WO2022074214A1 (en) 2022-04-14

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