MX2023003567A - Uso de agonista del receptor de esfingosina-1-fosfato. - Google Patents

Uso de agonista del receptor de esfingosina-1-fosfato.

Info

Publication number
MX2023003567A
MX2023003567A MX2023003567A MX2023003567A MX2023003567A MX 2023003567 A MX2023003567 A MX 2023003567A MX 2023003567 A MX2023003567 A MX 2023003567A MX 2023003567 A MX2023003567 A MX 2023003567A MX 2023003567 A MX2023003567 A MX 2023003567A
Authority
MX
Mexico
Prior art keywords
sphingosine
receptor agonist
phosphate receptor
phosphate
prevention
Prior art date
Application number
MX2023003567A
Other languages
English (en)
Inventor
Tae Hun Kim
Ki Chan Kim
Original Assignee
Lg Chemical Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lg Chemical Ltd filed Critical Lg Chemical Ltd
Publication of MX2023003567A publication Critical patent/MX2023003567A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • A61K31/4523Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/454Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • A61K31/404Indoles, e.g. pindolol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4151,2-Diazoles
    • A61K31/4161,2-Diazoles condensed with carbocyclic ring systems, e.g. indazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/06Antipsoriatics

Landscapes

  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Dermatology (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

La presente invención se relaciona al uso de un compuesto de la fórmula química 1 o una sal farmacéuticamente aceptable del mismo para la prevención o tratamiento de dermatitis atópica.
MX2023003567A 2020-09-28 2021-09-27 Uso de agonista del receptor de esfingosina-1-fosfato. MX2023003567A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
KR20200125583 2020-09-28
PCT/KR2021/013097 WO2022065939A1 (ko) 2020-09-28 2021-09-27 스핑고신-1-인산 수용체 효능제의 용도

Publications (1)

Publication Number Publication Date
MX2023003567A true MX2023003567A (es) 2023-04-04

Family

ID=80846731

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2023003567A MX2023003567A (es) 2020-09-28 2021-09-27 Uso de agonista del receptor de esfingosina-1-fosfato.

Country Status (11)

Country Link
US (1) US20230330077A1 (es)
EP (1) EP4212159A4 (es)
JP (1) JP2023542730A (es)
KR (1) KR20220043046A (es)
CN (1) CN116437921A (es)
AU (1) AU2021349680A1 (es)
BR (1) BR112023005536A2 (es)
CA (1) CA3192701A1 (es)
MX (1) MX2023003567A (es)
TW (2) TW202402285A (es)
WO (1) WO2022065939A1 (es)

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2498609B1 (en) * 2009-11-13 2018-04-18 Celgene International II Sàrl Selective heterocyclic sphingosine 1 phosphate receptor modulators
EP2390252A1 (en) * 2010-05-19 2011-11-30 Almirall, S.A. New pyrazole derivatives
JP6294359B2 (ja) 2013-02-20 2018-03-14 エルジー・ケム・リミテッド スフィンゴシン−1−リン酸受容体アゴニスト、その製造方法及びそれらを活性成分として含有する医薬組成物
AU2016205361C1 (en) * 2015-01-06 2021-04-08 Arena Pharmaceuticals, Inc. Methods of treating conditions related to the S1P1 receptor

Also Published As

Publication number Publication date
BR112023005536A2 (pt) 2023-04-25
KR20220043046A (ko) 2022-04-05
AU2021349680A1 (en) 2023-06-08
TW202402285A (zh) 2024-01-16
EP4212159A1 (en) 2023-07-19
TW202222314A (zh) 2022-06-16
EP4212159A4 (en) 2024-03-06
JP2023542730A (ja) 2023-10-11
CN116437921A (zh) 2023-07-14
US20230330077A1 (en) 2023-10-19
WO2022065939A1 (ko) 2022-03-31
CA3192701A1 (en) 2022-03-31

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