MX2022001647A - Terapia de combinacion con vildagliptina y metformina. - Google Patents

Terapia de combinacion con vildagliptina y metformina.

Info

Publication number
MX2022001647A
MX2022001647A MX2022001647A MX2022001647A MX2022001647A MX 2022001647 A MX2022001647 A MX 2022001647A MX 2022001647 A MX2022001647 A MX 2022001647A MX 2022001647 A MX2022001647 A MX 2022001647A MX 2022001647 A MX2022001647 A MX 2022001647A
Authority
MX
Mexico
Prior art keywords
metformin
pharmaceutically acceptable
acceptable salt
vildagliptin
combination therapy
Prior art date
Application number
MX2022001647A
Other languages
English (en)
Inventor
Paivi M Paldanius
Wolfgang Kothny
James E Foley
David R Matthews
Michael Stumvoll
Prato Stefano Del
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of MX2022001647A publication Critical patent/MX2022001647A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/155Amidines (), e.g. guanidine (H2N—C(=NH)—NH2), isourea (N=C(OH)—NH2), isothiourea (—N=C(SH)—NH2)
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Diabetes (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Engineering & Computer Science (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

La invención se refiere a un inhibidor de DPP-IV (preferentemente vildagliptina o una sal farmacéuticamente aceptable de la misma) y metformina o una sal farmacéuticamente aceptable de la misma, para su uso en el tratamiento de la diabetes tipo 2. La invención también se refiere al uso de un inhibidor de DPP-IV (preferentemente vildagliptina o una sal farmacéuticamente aceptable de la misma) y metformina o una sal farmacéuticamente aceptable de la misma, en la fabricación de un medicamento para tratar la diabetes tipo 2. La invención también se refiere a un método para tratar la diabetes tipo 2 usando un inhibidor de DPP-IV (preferentemente vildagliptina o una sal farmacéuticamente aceptable de la misma) y metformina o una sal farmacéuticamente aceptable de la misma.
MX2022001647A 2019-09-17 2020-09-17 Terapia de combinacion con vildagliptina y metformina. MX2022001647A (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201962901645P 2019-09-17 2019-09-17
US202063004230P 2020-04-02 2020-04-02
PCT/EP2020/075993 WO2021053076A1 (en) 2019-09-17 2020-09-17 Combination therapy with vildagliptin and metformin

Publications (1)

Publication Number Publication Date
MX2022001647A true MX2022001647A (es) 2022-03-11

Family

ID=72561784

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2022001647A MX2022001647A (es) 2019-09-17 2020-09-17 Terapia de combinacion con vildagliptina y metformina.

Country Status (8)

Country Link
US (2) US11103469B2 (es)
EP (2) EP4335438A1 (es)
JP (1) JP2022548214A (es)
KR (1) KR20220063157A (es)
BR (1) BR112022003183A2 (es)
MA (1) MA55763A (es)
MX (1) MX2022001647A (es)
WO (1) WO2021053076A1 (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP4335438A1 (en) * 2019-09-17 2024-03-13 Novartis AG Combination therapy with vildagliptin and metformin
KR20230163635A (ko) 2022-05-24 2023-12-01 주식회사 엘지에너지솔루션 심플 배터리팩 및 이의 제조방법

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE122010000020I1 (de) 1996-04-25 2010-07-08 Prosidion Ltd Verfahren zur Senkung des Blutglukosespiegels in Säugern
BRPI0107715B8 (pt) 2000-01-21 2021-05-25 Novartis Ag produto farmacêutico compreendendo um inibidor de dipeptidilpeptidase-iv e metformina, bem como usos do dito produto farmacêutico e do inibidor de dipeptidilpeptidase-iv
KR20130105741A (ko) 2003-11-17 2013-09-25 노파르티스 아게 디펩티딜 펩티다제 ⅳ 억제제의 용도
US7935723B2 (en) 2004-06-04 2011-05-03 Novartis Pharma Ag Use of organic compounds
KR20070068407A (ko) 2004-10-25 2007-06-29 노파르티스 아게 Dpp―iv 억제제, ppar 항당뇨병제 및메트포르민의 조합물
GB0526291D0 (en) 2005-12-23 2006-02-01 Prosidion Ltd Therapeutic method
PE20110235A1 (es) * 2006-05-04 2011-04-14 Boehringer Ingelheim Int Combinaciones farmaceuticas que comprenden linagliptina y metmorfina
EP4335438A1 (en) * 2019-09-17 2024-03-13 Novartis AG Combination therapy with vildagliptin and metformin

Also Published As

Publication number Publication date
EP3958857A1 (en) 2022-03-02
WO2021053076A1 (en) 2021-03-25
US20220184006A1 (en) 2022-06-16
EP4335438A1 (en) 2024-03-13
US11103469B2 (en) 2021-08-31
US20210077430A1 (en) 2021-03-18
MA55763A (fr) 2022-04-20
BR112022003183A2 (pt) 2022-05-17
JP2022548214A (ja) 2022-11-17
US12090125B2 (en) 2024-09-17
KR20220063157A (ko) 2022-05-17

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