MX2020010502A - Agentes farmacológicos para el tratamiento de enfermedades oculares. - Google Patents

Agentes farmacológicos para el tratamiento de enfermedades oculares.

Info

Publication number
MX2020010502A
MX2020010502A MX2020010502A MX2020010502A MX2020010502A MX 2020010502 A MX2020010502 A MX 2020010502A MX 2020010502 A MX2020010502 A MX 2020010502A MX 2020010502 A MX2020010502 A MX 2020010502A MX 2020010502 A MX2020010502 A MX 2020010502A
Authority
MX
Mexico
Prior art keywords
pharmacological agents
ocular diseases
treating ocular
subject
methods
Prior art date
Application number
MX2020010502A
Other languages
English (en)
Spanish (es)
Inventor
Surya Kanta De
G Sridhar Prasad
Marshall Clarke Peterman
Bernard Collins
Original Assignee
Calasia Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Calasia Pharmaceuticals Inc filed Critical Calasia Pharmaceuticals Inc
Publication of MX2020010502A publication Critical patent/MX2020010502A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/12Ketones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/66Phosphorus compounds
    • A61K31/661Phosphorus acids or esters thereof not having P—C bonds, e.g. fosfosal, dichlorvos, malathion or mevinphos
    • A61K31/6615Compounds having two or more esterified phosphorus acid groups, e.g. inositol triphosphate, phytic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/4738Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4741Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems condensed with ring systems having oxygen as a ring hetero atom, e.g. tubocuraran derivatives, noscapine, bicuculline
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16Anti-Parkinson drugs
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • A61P27/10Ophthalmic agents for accommodation disorders, e.g. myopia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • A61P27/12Ophthalmic agents for cataracts
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Ophthalmology & Optometry (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Psychology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
MX2020010502A 2018-04-05 2019-04-05 Agentes farmacológicos para el tratamiento de enfermedades oculares. MX2020010502A (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862653249P 2018-04-05 2018-04-05
US201862694729P 2018-07-06 2018-07-06
PCT/US2019/026112 WO2019195761A2 (en) 2018-04-05 2019-04-05 Pharmacological agents for treating ocular diseases

Publications (1)

Publication Number Publication Date
MX2020010502A true MX2020010502A (es) 2021-03-25

Family

ID=68101528

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2020010502A MX2020010502A (es) 2018-04-05 2019-04-05 Agentes farmacológicos para el tratamiento de enfermedades oculares.

Country Status (6)

Country Link
US (1) US11872236B2 (https=)
JP (1) JP7532259B2 (https=)
CN (1) CN112601513B (https=)
BR (1) BR112020020351A2 (https=)
MX (1) MX2020010502A (https=)
WO (1) WO2019195761A2 (https=)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN120097859A (zh) * 2019-02-19 2025-06-06 加利福尼亚大学董事会 Nurr1受体调节剂
EP3976017A4 (en) * 2019-05-31 2023-06-14 Plex Pharmaceuticals, Inc. PHARMACOLOGICAL SUBSTANCES FOR THE TREATMENT OF PROTEIN AGGREGATION DISEASES OF THE EYE
WO2021086834A1 (en) * 2019-10-28 2021-05-06 Kebotix, Inc. Electronic control of transmittance of visible and near-infrared radiation
WO2022098847A1 (en) * 2020-11-04 2022-05-12 Corino Therapeutics, Inc. Tolcapone analogs and methods of use
CN116963727A (zh) * 2020-11-13 2023-10-27 普莱克斯医药公司 用于治疗眼部病症的药剂
JP2023549533A (ja) * 2020-11-13 2023-11-27 プレックス ファーマスーティカルズ,インク 眼の状態を処置するための薬理剤
US20250019352A1 (en) * 2021-06-29 2025-01-16 Plex Pharmaceuticals, Inc. Pharmacological agents for treating ophthalmic diseases
GB202204798D0 (en) 2022-04-01 2022-05-18 Bial Portela & Ca Sa Prodrugs of opicapone
WO2024123100A1 (ko) * 2022-12-09 2024-06-13 경희대학교 산학협력단 신규 아밀로이드-베타 응집체 분해제와 이를 이용한 뇌 표적화 약물 전달 시스템

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5236952A (en) * 1986-03-11 1993-08-17 Hoffmann-La Roche Inc. Catechol derivatives
DK175069B1 (da) 1986-03-11 2004-05-24 Hoffmann La Roche Pyrocatecholderivater
JPH1036257A (ja) * 1996-05-22 1998-02-10 Kikkoman Corp メイラード反応阻害剤
ID19540A (id) 1997-01-22 1998-07-23 Hoffmann La Roche Metode pembuatan turunan-turunan benzofenon
JP2000256259A (ja) * 1999-03-11 2000-09-19 Nippon Zoki Pharmaceut Co Ltd メイラード反応阻害剤
US8299079B2 (en) 2009-05-22 2012-10-30 Kaufman Herbert E Preparations and methods for ameliorating or reducing presbyopia
WO2011047412A1 (en) * 2009-10-22 2011-04-28 The Heart Research Institute Ltd Tyrosine and l-dopa for reducing l-dopa incorporation into proteins
WO2011140333A1 (en) * 2010-05-07 2011-11-10 The Board Of Trustees Of The Leland Stanford Junior University Identification of stabilizers of multimeric proteins
WO2014147464A2 (en) 2013-03-20 2014-09-25 Ra Chem Pharma Limited Novel process for the preparation of tolcapone
WO2015095257A2 (en) * 2013-12-18 2015-06-25 Emory University Managing visual dysfunction or loss of vision for diabetic subjects
RU2724190C2 (ru) 2014-02-08 2020-06-23 Дженентек, Инк. Способы лечения болезни альцгеймера
KR20170048426A (ko) * 2014-08-22 2017-05-08 광저우 캉루이 바이오로지컬 파마슈티컬 테크놀로지 씨오., 엘티디. 시각 장애를 치료하기 위한 조성물 및 방법
WO2017039525A1 (en) 2015-09-04 2017-03-09 Lobsor Pharmaceuticals Aktiebolag Method of treating a dopamine related disorder in a subject by administering levodopa, in combination with a dopamine decarboxylase inhibitor and a catechol-o-methyltransferase inhibitor
CN116963727A (zh) 2020-11-13 2023-10-27 普莱克斯医药公司 用于治疗眼部病症的药剂
JP2023549533A (ja) 2020-11-13 2023-11-27 プレックス ファーマスーティカルズ,インク 眼の状態を処置するための薬理剤

Also Published As

Publication number Publication date
EP3773438A2 (en) 2021-02-17
WO2019195761A2 (en) 2019-10-10
WO2019195761A3 (en) 2020-07-23
CN112601513A (zh) 2021-04-02
JP7532259B2 (ja) 2024-08-13
BR112020020351A2 (pt) 2021-01-12
CN112601513B (zh) 2023-12-22
US20210154213A1 (en) 2021-05-27
US11872236B2 (en) 2024-01-16
JP2021532059A (ja) 2021-11-25

Similar Documents

Publication Publication Date Title
MX2020010502A (es) Agentes farmacológicos para el tratamiento de enfermedades oculares.
EP4491229A3 (en) Coding rna administered into the suprachoroidal space in the treatment of ophtalmic diseases
MX2010003774A (es) Formulaciones oftalmicas acuosas.
TW200633709A (en) Aminopyrazine analogs for treating glaucoma and other rho kinase-mediated diseases and conditions
BR112016025997A8 (pt) compostos para tratamento de doenças e lesões oftalmológicas, uma composição farmacêutica e uma formulação oftálmica
JP2015025011A5 (https=)
WO2011053801A3 (en) Methods and cosmetic preparations for the sustained delivery of therapeutic agents to the eye
MX2015012653A (es) Formulaciones oculares para suministro de farmaco al segmento porterior del ojo.
MX2020006309A (es) Fórmulaciones de parasiticida de isoxazolina y métodos para el tratamiento de la blefaritis.
EP4324454A3 (en) Cross-linking agents and associated methods
MX2024010655A (es) Uso de profarmacos de riluzol para tratar enfermedad de alzheimer.
AU2017261303A1 (en) Ophthalmic compositions
EA200800336A1 (ru) Лечение состояний, связанных с присутствием макромолекулярных агрегатов, в частности глазных расстройств
MX2021016055A (es) Formulaciones y métodos de parasiticidas de isoxazolina para el tratamiento de la blefaritis.
MX2021014682A (es) Agentes farmacológicos para tratar enfermedades de agregación de proteínas de los ojos.
HRP20190561T1 (hr) Postupci liječenja bolesti oka povezanih s upalom i vaskularnom proliferacijom
CA3167959A1 (en) Prodrug for the treatment of disease and injury of oxidative stress
MX2015016750A (es) Composicion inmunogenica para uso en terapia.
BRPI0407693A (pt) uso de esteróides para preparação de formulações utilizáveis no tratamento de pessoas sofrendo de distúrbios oculares, bem como formulação assim obtidos
MX2023002350A (es) Composiciones y metodos para mejorar enfermedades y trastornos neurologicos.
PH12020550722A1 (en) Ophthalmic topical composition comprising dobesilic acid for treating diseases of the posterior segment of the eye
MY195178A (en) Composition for Treating Joint Disease and Kit Containing Same
MX2021009777A (es) Formulaciones inyectables de fenol y metodos de su uso.
MX2023010918A (es) Metodos y composiciones para el tratamiento de enfermedades oculares.
MX2021015796A (es) Composiciones y metodos para tratar enfermedades oculares.