MX2019011173A - Compuesto que contiene silicio para la resistencia a la infeccion por el virus de la hepatitis c. - Google Patents

Compuesto que contiene silicio para la resistencia a la infeccion por el virus de la hepatitis c.

Info

Publication number
MX2019011173A
MX2019011173A MX2019011173A MX2019011173A MX2019011173A MX 2019011173 A MX2019011173 A MX 2019011173A MX 2019011173 A MX2019011173 A MX 2019011173A MX 2019011173 A MX2019011173 A MX 2019011173A MX 2019011173 A MX2019011173 A MX 2019011173A
Authority
MX
Mexico
Prior art keywords
hepatitis
virus infection
silicon
resistance
containing compound
Prior art date
Application number
MX2019011173A
Other languages
English (en)
Inventor
Huang Yu
Xu Hongjiang
Zhang Yinsheng
Liu Baomin
Chen Zhengbang
Gai Kuo
LIU Xushi
Wang Xiaojin
Original Assignee
Chia Tai Tianqing Pharmaceutical Group Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chia Tai Tianqing Pharmaceutical Group Co Ltd filed Critical Chia Tai Tianqing Pharmaceutical Group Co Ltd
Publication of MX2019011173A publication Critical patent/MX2019011173A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00Compounds containing elements of Groups 4 or 14 of the Periodic System
    • C07F7/02Silicon compounds
    • C07F7/08Compounds having one or more C—Si linkages
    • C07F7/0803Compounds with Si-C or Si-Si linkages
    • C07F7/081Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te
    • C07F7/0812Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te comprising a heterocyclic ring
    • C07F7/0816Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te comprising a heterocyclic ring said ring comprising Si as a ring atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/695Silicon compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses

Abstract

La presente invención proporciona un compuesto que contiene silicio para la resistencia a la infección por virus de la hepatitis c y, en particular, proporciona un compuesto representado por la fórmula I, o una sal farmacéuticamente aceptable, o un tautómero, o un estereoisómero, o un compuesto deuterado del mismo y una mezcla entre ellos, un proceso para la preparación de este, y una composición farmacéutica que comprende el mismo. La presente solicitud también proporciona un uso del compuesto, o una sal farmacéuticamente aceptable, o un tautómero, o un estereoisómero, o un compuesto deuterado del mismo y una mezcla entre ellos, y una composición farmacéutica que comprende el mismo en el tratamiento de la infección por virus de la hepatitis c.
MX2019011173A 2017-03-22 2018-03-22 Compuesto que contiene silicio para la resistencia a la infeccion por el virus de la hepatitis c. MX2019011173A (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CN201710172925 2017-03-22
CN201710845367 2017-09-19
PCT/CN2018/079965 WO2018171660A1 (zh) 2017-03-22 2018-03-22 用于抗丙型肝炎病毒感染的含硅化合物

Publications (1)

Publication Number Publication Date
MX2019011173A true MX2019011173A (es) 2020-01-09

Family

ID=63585044

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2019011173A MX2019011173A (es) 2017-03-22 2018-03-22 Compuesto que contiene silicio para la resistencia a la infeccion por el virus de la hepatitis c.

Country Status (7)

Country Link
US (1) US10766912B2 (es)
EP (1) EP3604295A4 (es)
JP (1) JP2020512331A (es)
CN (1) CN110382487B (es)
BR (1) BR112019019724A2 (es)
MX (1) MX2019011173A (es)
WO (1) WO2018171660A1 (es)

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8329159B2 (en) 2006-08-11 2012-12-11 Bristol-Myers Squibb Company Hepatitis C virus inhibitors
CN101558059B (zh) 2006-08-11 2014-12-03 百时美施贵宝公司 丙型肝炎病毒抑制剂
CN103819459B (zh) * 2009-06-11 2017-05-17 艾伯维巴哈马有限公司 抗病毒化合物
US8937150B2 (en) * 2009-06-11 2015-01-20 Abbvie Inc. Anti-viral compounds
EA201290882A1 (ru) * 2010-03-09 2013-04-30 Мерк Шарп Энд Домэ Корп. Конденсированные трициклические силильные соединения и способы их применения для лечения вирусных заболеваний
WO2013054275A1 (en) * 2011-10-11 2013-04-18 Council Of Scientific & Industrial Research Sila analogs of oxazolidinone derivatives and synthesis thereof
US8927749B2 (en) * 2013-03-07 2015-01-06 Universal Display Corporation Organic electroluminescent materials and devices
WO2016095814A1 (en) * 2014-12-16 2016-06-23 Sunshine Lake Pharma Co., Ltd. Bridged ring compounds as hepatitis c virus inhibitors and preparation thereof

Also Published As

Publication number Publication date
JP2020512331A (ja) 2020-04-23
US20200017532A1 (en) 2020-01-16
WO2018171660A1 (zh) 2018-09-27
BR112019019724A2 (pt) 2020-04-14
EP3604295A4 (en) 2020-12-16
US10766912B2 (en) 2020-09-08
EP3604295A1 (en) 2020-02-05
CN110382487A (zh) 2019-10-25
CN110382487B (zh) 2021-04-02

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