MX2018011699A - Composicion farmaceutica sinergica de un antagonista de los receptores de leucotrienos y un agonista inverso de la histamina h1. - Google Patents
Composicion farmaceutica sinergica de un antagonista de los receptores de leucotrienos y un agonista inverso de la histamina h1.Info
- Publication number
- MX2018011699A MX2018011699A MX2018011699A MX2018011699A MX2018011699A MX 2018011699 A MX2018011699 A MX 2018011699A MX 2018011699 A MX2018011699 A MX 2018011699A MX 2018011699 A MX2018011699 A MX 2018011699A MX 2018011699 A MX2018011699 A MX 2018011699A
- Authority
- MX
- Mexico
- Prior art keywords
- pharmaceutical composition
- histamine
- receptor antagonist
- leukotriene receptor
- inverse agonist
- Prior art date
Links
Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
- A61K31/4535—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a heterocyclic ring having sulfur as a ring hetero atom, e.g. pizotifen
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0043—Nose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Pulmonology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Dermatology (AREA)
- Nutrition Science (AREA)
- Physiology (AREA)
- Otolaryngology (AREA)
- Immunology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
La presente invención se refiere a una composición farmacéutica que comprende la combinación sinérgica de un antagonista de los receptores de leucotrienos, como lo es el principio activo: montelukast y sus sales farmacéuticamente aceptables y un antagonista inverso de la histamina H1, como lo es el principio activo: ketotifeno y sus sales farmacéuticamente aceptables, los cuales se encuentran formulados con excipientes y/o vehículos y/o aditivos farmacéuticamente aceptables en una sola unidad de dosificación para ser administrado por vía oral, transdérmica o por dispositivos para inhalación oral, nasal, misma que está indicada para el tratamiento de la enfermedad atópica como: asma, rinitis alérgica y dermatitis atópica.
Priority Applications (6)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
MX2018011699A MX2018011699A (es) | 2018-09-26 | 2018-09-26 | Composicion farmaceutica sinergica de un antagonista de los receptores de leucotrienos y un agonista inverso de la histamina h1. |
US17/280,049 US20220031687A1 (en) | 2018-09-26 | 2019-09-20 | Synergic pharmaceutical combination of a leukotriene-receptor antagonist and an inverse agonist of histamine hi |
PCT/MX2019/000100 WO2020067866A1 (es) | 2018-09-26 | 2019-09-20 | Combinación farmacéutica sinérgica de un antagonista de los receptores de leucotrienos y un agonista inverso de la histamina h1 |
EP19866151.4A EP3858354A4 (en) | 2018-09-26 | 2019-09-20 | SYNERGISTIC PHARMACEUTICAL COMBINATION OF A LEUKOTRIEN RECEPTOR ANTAGONIST AND A HISTAMINE-H1 INVERSE AGONIST |
CA3113220A CA3113220A1 (en) | 2018-09-26 | 2019-09-20 | Synergic pharmaceutical combination of a leukotriene-receptor antagonist and an inverse agonist of histamine h1 |
CONC2021/0004992A CO2021004992A2 (es) | 2018-09-26 | 2021-04-19 | Combinación farmacéutica sinérgica de un antagonista de los receptores de leucotrienos y un agonista inverso de la histamina h1 |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
MX2018011699A MX2018011699A (es) | 2018-09-26 | 2018-09-26 | Composicion farmaceutica sinergica de un antagonista de los receptores de leucotrienos y un agonista inverso de la histamina h1. |
Publications (1)
Publication Number | Publication Date |
---|---|
MX2018011699A true MX2018011699A (es) | 2019-07-24 |
Family
ID=67998847
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MX2018011699A MX2018011699A (es) | 2018-09-26 | 2018-09-26 | Composicion farmaceutica sinergica de un antagonista de los receptores de leucotrienos y un agonista inverso de la histamina h1. |
Country Status (6)
Country | Link |
---|---|
US (1) | US20220031687A1 (es) |
EP (1) | EP3858354A4 (es) |
CA (1) | CA3113220A1 (es) |
CO (1) | CO2021004992A2 (es) |
MX (1) | MX2018011699A (es) |
WO (1) | WO2020067866A1 (es) |
Family Cites Families (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CH531000A (de) | 1970-03-11 | 1972-11-30 | Sandoz Ag | Verfahren zur Herstellung neuer Benzocycloheptathiophene |
US5565473A (en) | 1990-10-12 | 1996-10-15 | Merck Frosst Canada, Inc. | Unsaturated hydroxyalkylquinoline acids as leukotriene antagonists |
US6383471B1 (en) | 1999-04-06 | 2002-05-07 | Lipocine, Inc. | Compositions and methods for improved delivery of ionizable hydrophobic therapeutic agents |
US7815936B2 (en) | 2001-10-30 | 2010-10-19 | Evonik Degussa Gmbh | Use of granular materials based on pyrogenically produced silicon dioxide in pharmaceutical compositions |
US8268352B2 (en) | 2002-08-05 | 2012-09-18 | Torrent Pharmaceuticals Limited | Modified release composition for highly soluble drugs |
US20060263350A1 (en) * | 2003-09-26 | 2006-11-23 | Fairfield Clinical Trials Llc | Combination antihistamine medication |
US8758816B2 (en) | 2004-11-24 | 2014-06-24 | Meda Pharmaceuticals Inc. | Compositions comprising azelastine and methods of use thereof |
US8377994B2 (en) | 2006-05-10 | 2013-02-19 | Evonik Degussa GmeH | Use of roll compacted pyrogenically produced silicon dioxide in pharmaceutical compositions |
TWI455733B (zh) | 2009-03-30 | 2014-10-11 | Toray Industries | 口腔內崩壞性被覆錠劑 |
TR201009398A2 (tr) * | 2010-11-11 | 2012-05-21 | Bi̇lgi̇ç Mahmut | Fiziksel özellikleri geliştirilmiş tablet formülasyonları |
WO2013148366A1 (en) | 2012-03-27 | 2013-10-03 | Duke Unversity | Compositions and methods for the prevention and treatment of mast cell-induced vascular leakage |
-
2018
- 2018-09-26 MX MX2018011699A patent/MX2018011699A/es unknown
-
2019
- 2019-09-20 WO PCT/MX2019/000100 patent/WO2020067866A1/es unknown
- 2019-09-20 EP EP19866151.4A patent/EP3858354A4/en not_active Withdrawn
- 2019-09-20 CA CA3113220A patent/CA3113220A1/en active Pending
- 2019-09-20 US US17/280,049 patent/US20220031687A1/en active Pending
-
2021
- 2021-04-19 CO CONC2021/0004992A patent/CO2021004992A2/es unknown
Also Published As
Publication number | Publication date |
---|---|
EP3858354A4 (en) | 2022-03-16 |
EP3858354A1 (en) | 2021-08-04 |
US20220031687A1 (en) | 2022-02-03 |
WO2020067866A1 (es) | 2020-04-02 |
CA3113220A1 (en) | 2020-04-02 |
CO2021004992A2 (es) | 2021-04-30 |
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