MX2014002105A - Ligandos de receptor de estrogeno y metodos de uso de los mismos. - Google Patents

Ligandos de receptor de estrogeno y metodos de uso de los mismos.

Info

Publication number
MX2014002105A
MX2014002105A MX2014002105A MX2014002105A MX2014002105A MX 2014002105 A MX2014002105 A MX 2014002105A MX 2014002105 A MX2014002105 A MX 2014002105A MX 2014002105 A MX2014002105 A MX 2014002105A MX 2014002105 A MX2014002105 A MX 2014002105A
Authority
MX
Mexico
Prior art keywords
compound
another embodiment
prostate cancer
levels
castration
Prior art date
Application number
MX2014002105A
Other languages
English (en)
Spanish (es)
Inventor
Mitchell S Steiner
James Dalton
Christopher C Coss
Original Assignee
Gtx Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US13/215,679 external-priority patent/US9427418B2/en
Application filed by Gtx Inc filed Critical Gtx Inc
Priority claimed from PCT/US2012/052141 external-priority patent/WO2013043304A1/en
Publication of MX2014002105A publication Critical patent/MX2014002105A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/137Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • A61K31/165Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • A61K31/167Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the nitrogen of a carboxamide group directly attached to the aromatic ring, e.g. lidocaine, paracetamol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • A61K31/4453Non condensed piperidines, e.g. piperocaine only substituted in position 1, e.g. propipocaine, diperodon
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca

Landscapes

  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Emergency Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Steroid Compounds (AREA)
MX2014002105A 2011-08-23 2012-08-23 Ligandos de receptor de estrogeno y metodos de uso de los mismos. MX2014002105A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US13/215,679 US9427418B2 (en) 2009-02-23 2011-08-23 Estrogen receptor ligands and methods of use thereof
PCT/US2012/052141 WO2013043304A1 (en) 2009-02-23 2012-08-23 Estrogen receptor ligands and methods of use thereof

Publications (1)

Publication Number Publication Date
MX2014002105A true MX2014002105A (es) 2014-09-25

Family

ID=48444651

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2014002105A MX2014002105A (es) 2011-08-23 2012-08-23 Ligandos de receptor de estrogeno y metodos de uso de los mismos.

Country Status (10)

Country Link
EP (1) EP2747562A4 (enExample)
JP (1) JP2014524479A (enExample)
KR (1) KR20140064906A (enExample)
CN (1) CN103957706A (enExample)
AU (1) AU2012312902B2 (enExample)
CA (1) CA2845890A1 (enExample)
IL (1) IL231070A0 (enExample)
IN (1) IN2014DN01959A (enExample)
MX (1) MX2014002105A (enExample)
RU (1) RU2014111060A (enExample)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN111164093A (zh) * 2017-09-27 2020-05-15 塔尔格免疫治疗有限公司 去势抵抗性前列腺癌
JP2022523094A (ja) * 2019-01-30 2022-04-21 アラゴン ファーマシューティカルズ,インコーポレイテッド 転移性去勢感受性前立腺癌の治療のための抗アンドロゲン剤
CN113853216A (zh) * 2019-02-01 2021-12-28 肿瘤学研究所基金会(Ior) 治疗去势抵抗性前列腺癌的方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8546451B2 (en) * 2005-11-28 2013-10-01 Gtx, Inc. Estrogen receptor ligands and methods of use thereof
EA023472B1 (ru) * 2005-11-28 2016-06-30 Джи Ти Икс, ИНК. Агенты, связывающиеся с ядерными рецепторами
US8158828B2 (en) * 2005-11-28 2012-04-17 Gtx, Inc. Nuclear receptor binding agents
WO2010096801A1 (en) * 2009-02-23 2010-08-26 Gtx, Inc. Estrogen receptor ligands and methods of use thereof

Also Published As

Publication number Publication date
AU2012312902B2 (en) 2016-03-17
JP2014524479A (ja) 2014-09-22
KR20140064906A (ko) 2014-05-28
CN103957706A (zh) 2014-07-30
CA2845890A1 (en) 2013-03-28
RU2014111060A (ru) 2015-09-27
IN2014DN01959A (enExample) 2015-05-15
EP2747562A4 (en) 2015-05-06
IL231070A0 (en) 2014-03-31
EP2747562A1 (en) 2014-07-02
AU2012312902A1 (en) 2013-05-23

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