MX2009013240A - Derivados de carboxamida heterociclicos, su uso farmaceutico y composiciones. - Google Patents

Derivados de carboxamida heterociclicos, su uso farmaceutico y composiciones.

Info

Publication number
MX2009013240A
MX2009013240A MX2009013240A MX2009013240A MX2009013240A MX 2009013240 A MX2009013240 A MX 2009013240A MX 2009013240 A MX2009013240 A MX 2009013240A MX 2009013240 A MX2009013240 A MX 2009013240A MX 2009013240 A MX2009013240 A MX 2009013240A
Authority
MX
Mexico
Prior art keywords
compositions
pharmaceutical use
carboxamide derivatives
hetero bicyclic
bicyclic carboxamide
Prior art date
Application number
MX2009013240A
Other languages
English (en)
Inventor
Mark E Schnute
Peter G Ruminski
Cathleen E Hanau
Jeffery N Carroll
Kirby Sample
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of MX2009013240A publication Critical patent/MX2009013240A/es

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/88—Oxygen atoms
    • C07D239/90—Oxygen atoms with acyclic radicals attached in position 2 or 3
    • A—HUMAN NECESSITIES
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    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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Abstract

La presente invención se refiere a los compuestos de la fórmula I (ver fórmula I) y a sales farmacéuticamente aceptables de los mismos, a procesos para su preparación, a intermedios usados en su preparación y a composiciones que contienen dichos compuestos, y a los usos de dichos compuestos como agentes antiinflamatorios.
MX2009013240A 2007-06-05 2008-05-19 Derivados de carboxamida heterociclicos, su uso farmaceutico y composiciones. MX2009013240A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US94199807P 2007-06-05 2007-06-05
PCT/IB2008/001279 WO2008149191A1 (en) 2007-06-05 2008-05-19 Hetero bicyclic carboxamide derivatives and their pharmaceutical use and compositions

Publications (1)

Publication Number Publication Date
MX2009013240A true MX2009013240A (es) 2010-01-25

Family

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Family Applications (1)

Application Number Title Priority Date Filing Date
MX2009013240A MX2009013240A (es) 2007-06-05 2008-05-19 Derivados de carboxamida heterociclicos, su uso farmaceutico y composiciones.

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US (1) US20110009435A1 (es)
EP (1) EP2170843A1 (es)
JP (1) JP2010529102A (es)
KR (1) KR20100028092A (es)
CN (1) CN101796031A (es)
AU (1) AU2008259542A1 (es)
CA (1) CA2690101A1 (es)
IL (1) IL202383A0 (es)
MX (1) MX2009013240A (es)
WO (1) WO2008149191A1 (es)
ZA (1) ZA201000046B (es)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2011507894A (ja) * 2007-12-19 2011-03-10 グラクソスミスクライン・リミテッド・ライアビリティ・カンパニー プロリルヒドロキシラーゼ阻害剤

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* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6008243A (en) * 1996-10-24 1999-12-28 Agouron Pharmaceuticals, Inc. Metalloproteinase inhibitors, pharmaceutical compositions containing them, and their use
US6933298B2 (en) * 2001-12-08 2005-08-23 Aventis Pharma Deutschland Gmbh Pyridine-2,4-dicarboxylic acid diamides and pyrimidine-4,6-dicarboxylic acid diamides and the use thereof for selectively inhibiting collagenases
US7166609B2 (en) * 2002-11-02 2007-01-23 Sanofi-Aventis Deutschland Gmbh Pyrimidine-4,6-dicarboxylic acid diamides for selectively inhibiting collagenases
US20050004111A1 (en) * 2003-01-03 2005-01-06 Aventis Pharma Deutschland Gmbh Selective MMP-13 inhibitors
EP1740551B9 (en) * 2004-04-30 2013-01-16 Takeda Pharmaceutical Company Limited Heterocyclic amide compound and use thereof as an mmp-13 inhibitor
US20060173183A1 (en) * 2004-12-31 2006-08-03 Alantos Pharmaceuticals, Inc., Multicyclic bis-amide MMP inhibitors
US7915267B2 (en) * 2005-10-28 2011-03-29 Takeda Pharmaceutical Company Limited Heterocyclic amide compound and use thereof

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KR20100028092A (ko) 2010-03-11
AU2008259542A1 (en) 2008-12-11
CA2690101A1 (en) 2008-12-11
CN101796031A (zh) 2010-08-04
IL202383A0 (en) 2010-06-30
US20110009435A1 (en) 2011-01-13
JP2010529102A (ja) 2010-08-26
ZA201000046B (en) 2011-06-29
WO2008149191A1 (en) 2008-12-11
EP2170843A1 (en) 2010-04-07

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