MX2009010122A - Derivados de purinilo y su uso como moduladores del canal de potasio. - Google Patents
Derivados de purinilo y su uso como moduladores del canal de potasio.Info
- Publication number
- MX2009010122A MX2009010122A MX2009010122A MX2009010122A MX2009010122A MX 2009010122 A MX2009010122 A MX 2009010122A MX 2009010122 A MX2009010122 A MX 2009010122A MX 2009010122 A MX2009010122 A MX 2009010122A MX 2009010122 A MX2009010122 A MX 2009010122A
- Authority
- MX
- Mexico
- Prior art keywords
- potassium channel
- channel modulators
- purinyl derivatives
- derivatives
- purinyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D473/00—Heterocyclic compounds containing purine ring systems
- C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
- C07D473/16—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two nitrogen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/10—Drugs for disorders of the urinary system of the bladder
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D473/00—Heterocyclic compounds containing purine ring systems
- C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
- C07D473/24—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 one nitrogen and one sulfur atom
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Abstract
La presente invención se refiere a nuevos derivados de purinilo y su uso como agentes moduladores del canal de potasio. Sin embargo, la invención se dirige a composiciones farmacéuticas útiles para el tratamiento o alivio de enfermedades o trastornos asociados con la actividad de los canales de potasio.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US90850307P | 2007-03-28 | 2007-03-28 | |
DKPA200700482 | 2007-03-28 | ||
PCT/EP2008/053648 WO2008116909A1 (en) | 2007-03-28 | 2008-03-27 | Purinyl derivatives and their use as potassium channel modulators |
Publications (1)
Publication Number | Publication Date |
---|---|
MX2009010122A true MX2009010122A (es) | 2009-10-19 |
Family
ID=39473604
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MX2009010122A MX2009010122A (es) | 2007-03-28 | 2008-03-27 | Derivados de purinilo y su uso como moduladores del canal de potasio. |
Country Status (8)
Country | Link |
---|---|
US (4) | US8362024B2 (es) |
EP (5) | EP2142546B1 (es) |
AU (1) | AU2008231695B2 (es) |
CA (1) | CA2682019C (es) |
HK (1) | HK1141008A1 (es) |
IL (1) | IL200501A0 (es) |
MX (1) | MX2009010122A (es) |
WO (5) | WO2008116912A2 (es) |
Families Citing this family (29)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AR063141A1 (es) * | 2006-10-04 | 2008-12-30 | Pharmacopeia Inc | Derivados de 2- ( benzimidazolil ) purina 8- sustituida para inmunosupresion |
US20100035934A1 (en) * | 2007-02-02 | 2010-02-11 | Neurosearch A/S | Pyridinyl-pyrazole derivatives and their use as potassium channel modulators |
US20100105705A1 (en) * | 2007-03-28 | 2010-04-29 | Neurosearch A/S | Purinyl derivatives and their use as potassium channel modulators |
EP2142546B1 (en) * | 2007-03-28 | 2017-06-07 | Saniona A/S | Purinyl derivatives and their use as potassium channel modulators |
EP2203436A1 (en) | 2007-09-17 | 2010-07-07 | Neurosearch A/S | Pyrazine derivatives and their use as potassium channel modulators |
KR20110042153A (ko) * | 2008-05-30 | 2011-04-25 | 제넨테크, 인크. | 퓨린 pi3k 억제 화합물 및 사용 방법 |
EP2331527A1 (en) * | 2008-09-02 | 2011-06-15 | NeuroSearch A/S | Pyrazolyl-pyrimidine derivatives and their use as potassium channel modulators |
WO2010034706A1 (en) | 2008-09-26 | 2010-04-01 | Neurosearch A/S | Substituted purinyl-pyrazol derivatives and their use as potassium channel modulators |
US8268838B2 (en) | 2008-09-26 | 2012-09-18 | Neurosearch A/S | Substituted purinyl-pyrazole derivatives and their use as potassium channel modulators |
PE20100362A1 (es) | 2008-10-30 | 2010-05-27 | Irm Llc | Derivados de purina que expanden las celulas madre hematopoyeticas |
WO2010112486A1 (en) | 2009-04-01 | 2010-10-07 | Neurosearch A/S | SUBSTITUTED [1,2,4]TRIAZOLO[1,5-a]PYRIMIDINES AND THEIR USE AS POTASSIUM CHANNEL MODULATORS |
US8685987B2 (en) | 2009-04-01 | 2014-04-01 | Ataxion, Inc. | Substituted [1,2,4]triazolo[1,5-a]pyrimidines and their use as potassium channel modulators |
US20120184517A1 (en) * | 2009-04-30 | 2012-07-19 | Steven Marx | Treatment of diseases with altered smooth muscle contractility |
AR079814A1 (es) | 2009-12-31 | 2012-02-22 | Otsuka Pharma Co Ltd | Compuestos heterociclicos, composiciones farmaceuticas que los contienen y sus usos |
RU2013104038A (ru) | 2010-07-14 | 2014-08-20 | Ф. Хоффманн-Ля Рош Аг | СЕЛЕКТИВНЫЕ В ОТНОШЕНИИ PI3K p110 ДЕЛЬТА ПУРИНОВЫЕ СОЕДИНЕНИЯ И СПОСОБЫ ИХ ПРИМЕНЕНИЯ |
AR084312A1 (es) | 2010-12-16 | 2013-05-08 | Genentech Inc | Compuestos triciclicos inhibidores de la pi3k y composiciones farmaceuticas |
WO2012142029A2 (en) * | 2011-04-10 | 2012-10-18 | Florida A&M University | Serms for the treatment of estrogen receptor-mediated disorders |
CN102351716B (zh) * | 2011-08-17 | 2013-11-06 | 中国石油化工股份有限公司 | 一种降低甲酰苯胺法制备对氨基二苯胺塔设备腐蚀的方法 |
US8889730B2 (en) | 2012-04-10 | 2014-11-18 | Pfizer Inc. | Indole and indazole compounds that activate AMPK |
US9475797B2 (en) | 2012-06-26 | 2016-10-25 | Saniona A/S | Phenyl triazole derivative and its use for modulating the GABAA receptor complex |
US9394285B2 (en) | 2013-03-15 | 2016-07-19 | Pfizer Inc. | Indole and indazole compounds that activate AMPK |
JPWO2015005491A1 (ja) * | 2013-07-12 | 2017-03-02 | 国立大学法人京都大学 | 疾病の発症又は進行の一因となる異常スプライシングを抑制できる物質のスクリーニング方法 |
CA2969587A1 (en) | 2014-12-05 | 2016-06-09 | Centre National De La Recherche Scientifique (Cnrs) | Compounds for treating cystic fibrosis |
NZ738563A (en) | 2015-06-03 | 2019-09-27 | Bristol Myers Squibb Co | 4-hydroxy-3-(heteroaryl)pyridine-2-one apj agonists for use in the treatment of cardiovascular disorders |
EP3341372A1 (en) * | 2015-08-25 | 2018-07-04 | Bristol-Myers Squibb Company | Tgf beta receptor antagonists |
AU2017275657B2 (en) * | 2016-06-02 | 2021-08-19 | Novartis Ag | Potassium channel modulators |
EP3528816A4 (en) * | 2016-10-21 | 2020-04-08 | Nimbus Lakshmi, Inc. | TYK2 INHIBITORS AND USES THEREOF |
LT3571193T (lt) | 2017-01-23 | 2022-02-10 | Cadent Therapeutics, Inc. | Kalio kanalo moduliatoriai |
CN116178374A (zh) * | 2023-01-13 | 2023-05-30 | 河北医科大学 | 小电导钙激活钾离子通道激动剂及其合成和应用 |
Family Cites Families (39)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
PT874846E (pt) | 1995-11-01 | 2003-08-29 | Novartis Ag | Derivados de purina e processos para a sua preparacao |
FR2741881B1 (fr) | 1995-12-01 | 1999-07-30 | Centre Nat Rech Scient | Nouveaux derives de purine possedant notamment des prorietes anti-proliferatives et leurs applications biologiques |
DE19834044A1 (de) * | 1998-07-29 | 2000-02-03 | Bayer Ag | Neue substituierte Pyrazolderivate |
US20020103161A1 (en) * | 1999-12-17 | 2002-08-01 | Manfred Weigele | Novel heterocycles |
JP2003531111A (ja) | 1999-12-17 | 2003-10-21 | アライアッド・ファーマシューティカルズ・インコーポレーテッド | プロトンポンプインヒビター |
IL150060A0 (en) | 1999-12-17 | 2002-12-01 | Ariad Pharma Inc | Novel purines |
AU2441701A (en) | 1999-12-17 | 2001-06-25 | Ariad Pharmaceuticals, Inc. | Purine derivatives |
JP4381804B2 (ja) * | 2001-06-27 | 2009-12-09 | サイクラセル リミテッド | 2,6,9−置換プリン誘導体及び増殖性疾患の治療におけるその使用 |
US20030078232A1 (en) | 2001-08-08 | 2003-04-24 | Elfatih Elzein | Adenosine receptor A3 agonists |
US7262176B2 (en) * | 2001-08-08 | 2007-08-28 | Cv Therapeutics, Inc. | Adenosine A3 receptor agonists |
US20060009642A1 (en) | 2001-10-12 | 2006-01-12 | Irm Llc, A Delaware Limited Liability Company | Methods for the synthesis of substituted purines |
AU2002342051B2 (en) | 2001-10-12 | 2009-06-11 | Irm Llc | Kinase inhibitor scaffolds and methods for their preparation |
US20030229105A1 (en) | 2002-05-21 | 2003-12-11 | Cyclacel Limited | Treatment of autoimmune disorders |
EP1523314A2 (en) * | 2002-07-23 | 2005-04-20 | SmithKline Beecham Corporation | Pyrazolopyrimidines as protein kinase inhibitors |
US20030139427A1 (en) | 2002-08-23 | 2003-07-24 | Osi Pharmaceuticals Inc. | Bicyclic pyrimidinyl derivatives and methods of use thereof |
JP2006503826A (ja) | 2002-09-06 | 2006-02-02 | スミスクライン・ビーチャム・コーポレイション | ピロロ[2,3−d]ピリミジン−4−イルおよびプリン−6−イル尿素化合物 |
MXPA06001758A (es) * | 2003-08-15 | 2006-08-11 | Irm Llc | Anilino purinas sustituidas en la posicion 6 utiles como inhibidores de rtk. |
US20050165029A1 (en) * | 2004-01-13 | 2005-07-28 | Ambit Biosciences Corporation | Pyrrolopyrimidine derivatives and analogs and their use in the treatment and prevention of diseases |
WO2005080377A1 (ja) | 2004-02-20 | 2005-09-01 | Kirin Beer Kabushiki Kaisha | TGFβ阻害活性を有する化合物およびそれを含んでなる医薬組成物 |
GB0407723D0 (en) | 2004-04-05 | 2004-05-12 | Novartis Ag | Organic compounds |
FR2876583B1 (fr) * | 2004-10-15 | 2007-04-13 | Centre Nat Rech Scient Cnrse | Utilisation de derives de purines pour la fabrication de medicaments pour le traitement de la mucoviscidose et de maladies liees a un defaut d'adressage des proteines dans les cellules |
GB0500785D0 (en) * | 2005-01-14 | 2005-02-23 | Novartis Ag | Organic compounds |
JP4966958B2 (ja) | 2005-03-14 | 2012-07-04 | ノイロサーチ アクティーゼルスカブ | カリウムチャネル調節剤及び医療における使用 |
GB0505219D0 (en) | 2005-03-14 | 2005-04-20 | Novartis Ag | Organic compounds |
WO2006100212A1 (en) | 2005-03-22 | 2006-09-28 | Neurosearch A/S | Pyrazolyl-pyrimidines as potassium channel modulating agents and their medical use |
US20090036475A1 (en) * | 2005-03-22 | 2009-02-05 | Neurosearch A/S | Pyrazolyl-Pyrimidines as Potassium Channel Modulating Agents and Their Medical Use |
WO2006125211A1 (en) | 2005-05-19 | 2006-11-23 | Cv Therapeutics, Inc. | A1 adenosine receptor agonists |
EP1966184B1 (en) | 2005-12-20 | 2010-08-25 | NeuroSearch A/S | Pyridinyl-quinazoline derivatives and their medical use |
TW200745847A (en) * | 2005-12-23 | 2007-12-16 | Koninkl Philips Electronics Nv | Apparatus and method for dynamic cache management |
JP2010502674A (ja) | 2006-09-07 | 2010-01-28 | ノイロサーチ アクティーゼルスカブ | カリウムチャンネル調節剤として有用なピリジニル−ピリミジン誘導体 |
WO2008040753A1 (en) | 2006-10-03 | 2008-04-10 | Neurosearch A/S | Indazolyl derivatives useful as potassium channel modulating agents |
EA200900983A1 (ru) * | 2007-01-26 | 2010-02-26 | Айрм Ллк | Соединения и композиции в качестве ингибиторов киназы |
US20100035934A1 (en) | 2007-02-02 | 2010-02-11 | Neurosearch A/S | Pyridinyl-pyrazole derivatives and their use as potassium channel modulators |
US20100105705A1 (en) | 2007-03-28 | 2010-04-29 | Neurosearch A/S | Purinyl derivatives and their use as potassium channel modulators |
EP2142546B1 (en) | 2007-03-28 | 2017-06-07 | Saniona A/S | Purinyl derivatives and their use as potassium channel modulators |
WO2009050199A1 (en) * | 2007-10-17 | 2009-04-23 | Novartis Ag | Purine derivatives as adenosine al receptor ligands |
WO2010034706A1 (en) * | 2008-09-26 | 2010-04-01 | Neurosearch A/S | Substituted purinyl-pyrazol derivatives and their use as potassium channel modulators |
US8268838B2 (en) * | 2008-09-26 | 2012-09-18 | Neurosearch A/S | Substituted purinyl-pyrazole derivatives and their use as potassium channel modulators |
PE20100362A1 (es) * | 2008-10-30 | 2010-05-27 | Irm Llc | Derivados de purina que expanden las celulas madre hematopoyeticas |
-
2008
- 2008-03-27 EP EP08718278.8A patent/EP2142546B1/en active Active
- 2008-03-27 MX MX2009010122A patent/MX2009010122A/es active IP Right Grant
- 2008-03-27 WO PCT/EP2008/053657 patent/WO2008116912A2/en active Application Filing
- 2008-03-27 EP EP08718283A patent/EP2142547A1/en not_active Withdrawn
- 2008-03-27 EP EP08735528A patent/EP2144911A2/en not_active Withdrawn
- 2008-03-27 US US12/593,194 patent/US8362024B2/en active Active
- 2008-03-27 WO PCT/EP2008/053648 patent/WO2008116909A1/en active Application Filing
- 2008-03-27 US US12/593,152 patent/US20100130516A1/en not_active Abandoned
- 2008-03-27 WO PCT/EP2008/053659 patent/WO2008116914A1/en active Application Filing
- 2008-03-27 WO PCT/EP2008/053651 patent/WO2008116911A1/en active Application Filing
- 2008-03-27 WO PCT/EP2008/053649 patent/WO2008116910A1/en active Application Filing
- 2008-03-27 AU AU2008231695A patent/AU2008231695B2/en active Active
- 2008-03-27 US US12/593,218 patent/US20100152210A1/en not_active Abandoned
- 2008-03-27 EP EP08735523A patent/EP2142545A1/en not_active Withdrawn
- 2008-03-27 EP EP08718279A patent/EP2132208A1/en not_active Withdrawn
- 2008-03-27 CA CA2682019A patent/CA2682019C/en active Active
-
2009
- 2009-08-20 IL IL200501A patent/IL200501A0/en unknown
-
2010
- 2010-07-20 HK HK10107002.9A patent/HK1141008A1/xx unknown
-
2012
- 2012-12-19 US US13/720,956 patent/US9340544B2/en active Active
Also Published As
Publication number | Publication date |
---|---|
AU2008231695A1 (en) | 2008-10-02 |
US9340544B2 (en) | 2016-05-17 |
EP2142546B1 (en) | 2017-06-07 |
US20100130516A1 (en) | 2010-05-27 |
EP2144911A2 (en) | 2010-01-20 |
US20100120797A1 (en) | 2010-05-13 |
EP2142545A1 (en) | 2010-01-13 |
US8362024B2 (en) | 2013-01-29 |
EP2142546A1 (en) | 2010-01-13 |
AU2008231695B2 (en) | 2013-03-28 |
HK1141008A1 (en) | 2010-10-29 |
WO2008116914A1 (en) | 2008-10-02 |
WO2008116909A1 (en) | 2008-10-02 |
WO2008116912A3 (en) | 2009-02-05 |
WO2008116911A1 (en) | 2008-10-02 |
EP2142547A1 (en) | 2010-01-13 |
WO2008116910A1 (en) | 2008-10-02 |
CA2682019C (en) | 2016-08-09 |
EP2132208A1 (en) | 2009-12-16 |
CA2682019A1 (en) | 2008-10-02 |
WO2008116912A2 (en) | 2008-10-02 |
US20100152210A1 (en) | 2010-06-17 |
IL200501A0 (en) | 2010-04-29 |
US20130109704A1 (en) | 2013-05-02 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
MX2009010122A (es) | Derivados de purinilo y su uso como moduladores del canal de potasio. | |
UA98482C2 (ru) | Пуринильные производные и их применение в качестве модуляторов каналов калия | |
TN2010000122A1 (en) | Compounds and compositions as modulators of gpr119 activity | |
PL2134704T3 (pl) | Związki i kompozycje pełniące rolę modulatorów aktywności GPR119 | |
MX2020012825A (es) | Compuestos multiciclicos y metodos de uso de los mismos. | |
TW200745109A (en) | Pyrrolo-pyridine kinase modulators | |
EA200901032A1 (ru) | Соединения и композиции в качестве модуляторов активности gpr119 | |
WO2008092942A3 (en) | Pyridinyl-pyrazole derivatives and their use as potassium channel modulators | |
HN2010002774A (es) | DERIVADOS DE 2-(1,5-DIHIDRO-5-OXO-1,2,4-TRIAZOL-4-IL/2-OXOIMIDAZOLIDIN-1-IL)PIRIDIN-4-CARBOXAMIDA ACTIVOS COMO MODULADORES DE ESTEAROIL-CoA | |
AU2007257423A8 (en) | Purine analogs | |
MX2013004329A (es) | 6-amino-nicotinamidas sustituidas como moduladores de kcnq2/3. | |
MX2010004530A (es) | Antagonistas de los canales de calcio tipo t de heterociclo fenil amida. | |
UA94639C2 (ru) | Трициклические соединения и их применение как модуляторов глюкокортикоидного рецептора | |
MX2012004078A (es) | Compuestos y composiciones como moduladores de la actividad de gpr119. | |
ZA201108305B (en) | Novel p2x7r antagonists and their use | |
PL1937669T3 (pl) | Nowe pochodne benzopiranu jako „otwieracze" kanału potasowego | |
TW200734323A (en) | 3-Aminocyclopentanecarboxamides as modulators of chemokine receptors | |
ZA201006782B (en) | Novel p2x7r antagonists and thier use | |
MX2011006006A (es) | Compuestos, composicion farmaceutica y metodos para utilizarse en el tratamiento de trastornos metabolicos. | |
MX2013002118A (es) | 2-oxi-quinolin-3-carboxamidas sustituidas como moduladores de kcnq2/3. | |
WO2008028935A3 (en) | Pyridinyl-pyrimidine derivatives useful as potassium channel modulating agents | |
MX2013002121A (es) | Quinolina-3-carboxamidas sustituidas como moduladores de kcnq2/3. | |
MX2009008286A (es) | Compuestos triciclicos y su uso como moduladores del receptor de glucocorticosteroides. | |
MX2013002119A (es) | Sustituidas-2-oxo- y 2-tioxo-dihidroquinolin-3-carboxamidas como moduladores de kcnq2/3. | |
MX2013002295A (es) | 1-oxo-dihidroisoquinolin-3-carboxamidas sustituidas como moduladores de kcnq2/3. |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
FG | Grant or registration |