MX2009004625A - Derivados de 3-amino-pirazol-4-carboxamida utiles como inhibidores de proteina cinasas. - Google Patents
Derivados de 3-amino-pirazol-4-carboxamida utiles como inhibidores de proteina cinasas.Info
- Publication number
- MX2009004625A MX2009004625A MX2009004625A MX2009004625A MX2009004625A MX 2009004625 A MX2009004625 A MX 2009004625A MX 2009004625 A MX2009004625 A MX 2009004625A MX 2009004625 A MX2009004625 A MX 2009004625A MX 2009004625 A MX2009004625 A MX 2009004625A
- Authority
- MX
- Mexico
- Prior art keywords
- pyrazole
- inhibitors
- amino
- protein kinases
- derivatives useful
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/38—Nitrogen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Abstract
La invención se refiere a compuestos heterocíclicos novedosos de la fórmula (I), en donde todas las variables son como se define en la especificación, en forma libre o en forma de sal, a su preparación, a su uso como medicamentos y a medicamentos que los comprenden. (ver fórmula (I)).
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP06123163 | 2006-10-30 | ||
PCT/EP2007/061636 WO2008052974A1 (en) | 2006-10-30 | 2007-10-29 | 3-amino-pyrazole-4-carboxamide derivatives useful as inhibitors of protein kinases |
Publications (1)
Publication Number | Publication Date |
---|---|
MX2009004625A true MX2009004625A (es) | 2009-05-15 |
Family
ID=37890336
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MX2009004625A MX2009004625A (es) | 2006-10-30 | 2007-10-29 | Derivados de 3-amino-pirazol-4-carboxamida utiles como inhibidores de proteina cinasas. |
Country Status (10)
Country | Link |
---|---|
US (1) | US20100093821A1 (es) |
EP (1) | EP2079702A1 (es) |
JP (1) | JP2010508325A (es) |
KR (1) | KR20090074791A (es) |
CN (1) | CN101522636A (es) |
AU (1) | AU2007316190A1 (es) |
BR (1) | BRPI0717873A2 (es) |
CA (1) | CA2667927A1 (es) |
MX (1) | MX2009004625A (es) |
WO (1) | WO2008052974A1 (es) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2010014453A1 (en) * | 2008-07-31 | 2010-02-04 | Merck & Co., Inc. | Inhibitors of janus kinases |
KR100961410B1 (ko) | 2008-10-14 | 2010-06-09 | (주)네오팜 | 단백질 키나제 억제제로서 헤테로사이클릭 화합물 |
KR101646180B1 (ko) | 2014-09-22 | 2016-08-05 | 한양대학교 에리카산학협력단 | N-(5-아릴아미도-2-메틸페닐)-5-메틸이소옥사졸-4-카복스아미드 유도체, 이의 약학적으로 허용가능한 염, 이의 제조방법 및 이를 유효성분으로 포함하는 fms 키나아제 저해제 |
CN104876879B (zh) * | 2015-04-14 | 2018-05-18 | 中国科学院合肥物质科学研究院 | 一种bcr-abl激酶抑制剂 |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN1816529A (zh) * | 2003-05-01 | 2006-08-09 | 布里斯托尔-迈尔斯.斯奎布公司 | 用作激酶抑制剂的芳基取代的吡唑-酰胺化合物 |
SI2298743T1 (sl) * | 2003-06-26 | 2012-12-31 | Novartis Ag | Inhibitorji p38-kinaze na osnovi 5-ÄŤlenskih heterociklov |
-
2007
- 2007-10-29 US US12/447,315 patent/US20100093821A1/en not_active Abandoned
- 2007-10-29 JP JP2009535068A patent/JP2010508325A/ja active Pending
- 2007-10-29 AU AU2007316190A patent/AU2007316190A1/en not_active Abandoned
- 2007-10-29 CN CNA2007800383257A patent/CN101522636A/zh active Pending
- 2007-10-29 BR BRPI0717873-5A patent/BRPI0717873A2/pt not_active Application Discontinuation
- 2007-10-29 WO PCT/EP2007/061636 patent/WO2008052974A1/en active Application Filing
- 2007-10-29 MX MX2009004625A patent/MX2009004625A/es not_active Application Discontinuation
- 2007-10-29 EP EP07821990A patent/EP2079702A1/en not_active Withdrawn
- 2007-10-29 CA CA002667927A patent/CA2667927A1/en not_active Abandoned
- 2007-10-29 KR KR1020097008810A patent/KR20090074791A/ko not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
WO2008052974A1 (en) | 2008-05-08 |
US20100093821A1 (en) | 2010-04-15 |
CA2667927A1 (en) | 2008-05-08 |
BRPI0717873A2 (pt) | 2013-10-29 |
JP2010508325A (ja) | 2010-03-18 |
KR20090074791A (ko) | 2009-07-07 |
AU2007316190A1 (en) | 2008-05-08 |
CN101522636A (zh) | 2009-09-02 |
EP2079702A1 (en) | 2009-07-22 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FA | Abandonment or withdrawal |