MX2008014890A - Nuevos derivados de 1,4-diaza-biciclo[3.2.2]nonil pirimidinilo y su uso medico. - Google Patents
Nuevos derivados de 1,4-diaza-biciclo[3.2.2]nonil pirimidinilo y su uso medico.Info
- Publication number
- MX2008014890A MX2008014890A MX2008014890A MX2008014890A MX2008014890A MX 2008014890 A MX2008014890 A MX 2008014890A MX 2008014890 A MX2008014890 A MX 2008014890A MX 2008014890 A MX2008014890 A MX 2008014890A MX 2008014890 A MX2008014890 A MX 2008014890A
- Authority
- MX
- Mexico
- Prior art keywords
- disorders
- diaza
- bicyclo
- pain
- disease
- Prior art date
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| US80902306P | 2006-05-30 | 2006-05-30 | |
| DKPA200600730 | 2006-05-30 | ||
| PCT/EP2007/055171 WO2007138040A1 (en) | 2006-05-30 | 2007-05-29 | Novel 1,4-diaza-bicyclo[3.2.2]nonyl pyrimidinyl derivative and its medical use |
Publications (1)
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| MX2008014890A true MX2008014890A (es) | 2008-12-05 |
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| MX2008014889A MX2008014889A (es) | 2006-05-30 | 2007-05-29 | Nuevos derivados de 1,4-diaza-biciclo[3.2.2.]nonil pirimidinilo y su uso medico. |
| MX2008014885A MX2008014885A (es) | 2006-05-30 | 2007-05-29 | Nuevos derivados de 1,4-diaza-biciclo[3.2.2]nonil pirimidinilo y su uso medico. |
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| MX2008014885A MX2008014885A (es) | 2006-05-30 | 2007-05-29 | Nuevos derivados de 1,4-diaza-biciclo[3.2.2]nonil pirimidinilo y su uso medico. |
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| WO (3) | WO2007138040A1 (OSRAM) |
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| KR20060125885A (ko) * | 2004-02-04 | 2006-12-06 | 뉴로서치 에이/에스 | 콜린 수용체 조절제로서의 디아자바이사이클릭 아릴 유도체 |
| AU2007267178A1 (en) | 2006-05-30 | 2007-12-06 | Neurosearch A/S | Novel 1,4-diaza-bicyclo[3.2.2]nonyl pyrimidinyl derivatives and their medical use |
| JP2010536726A (ja) | 2007-08-17 | 2010-12-02 | ノイロサーチ アクティーゼルスカブ | ニコチン性アセチルコリン受容体リガンドとして有用な新規１，４−ジアザ−ビシクロ〔３．２．２〕ノニルヘテロアリール誘導体 |
| DE102007053771A1 (de) * | 2007-11-12 | 2009-05-14 | Merck Patent Gmbh | Organische Elektrolumineszenzvorrichtungen |
| EP2209783B8 (en) * | 2007-11-14 | 2016-06-01 | Saniona A/S | Novel 1,4-diaza-bicyclo[3.2.2]nonyl pyrimidine derivatives and their medical use |
| JP2011503144A (ja) * | 2007-11-14 | 2011-01-27 | ノイロサーチ アクティーゼルスカブ | 新規の１，４−ジアザ−ビシクロ［３．２．２］ノニルピリミジン誘導体及びその医療への使用 |
| JP2011503146A (ja) * | 2007-11-14 | 2011-01-27 | ノイロサーチ アクティーゼルスカブ | 新規な１，４−ジアザ−ビシクロ［３．２．２］ノニルピリミジン誘導体及びこれらの医療上の使用 |
| WO2010026176A1 (en) * | 2008-09-05 | 2010-03-11 | Neurosearch A/S | 1,4 -diaza- bicyclo [3.2.2]n0nyl pyrimidine derivatives as nicotinic and monoamine receptor modulators |
| WO2010026177A1 (en) * | 2008-09-05 | 2010-03-11 | Neurosearch A/S | 1,4-diaza-bicyclo [3.2.2] nonyl pyridine derivatives as nicotinic and monoamine receptor modulators |
| WO2010040806A1 (en) * | 2008-10-10 | 2010-04-15 | Neurosearch A/S | Novel diphenyl purine derivatives useful as modulators of nicotinic acetylcholine receptors |
| US20110257161A1 (en) * | 2008-12-04 | 2011-10-20 | Neurosearch A/S | Novel diaza-bicyclononyl-phenyl derivatives and their medical use |
| WO2010084120A1 (en) * | 2009-01-21 | 2010-07-29 | Neurosearch A/S | N-oxides of 1,4-diaza-bicyclo[3.2.2]nonyl pyrimidinyl derivatives useful as nicotinic acetylcholine receptor ligands |
| WO2010084121A1 (en) * | 2009-01-21 | 2010-07-29 | Neurosearch A/S | Novel diaza-bicyclononyl-pyrimidinyl derivatives and their medical use |
| TWI558398B (zh) | 2009-09-22 | 2016-11-21 | 諾華公司 | 菸鹼乙醯膽鹼受體α７活化劑之用途 |
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| FR2786770B1 (fr) * | 1998-12-04 | 2001-01-19 | Synthelabo | Derives de 1,4-diazabicyclo[3.2.2.]nonane, leur preparation et leur application en therapeutique |
| EP1368323B1 (en) * | 2001-02-14 | 2010-06-30 | Warner-Lambert Company LLC | Pyrimidine matrix metalloproteinase inhibitors |
| WO2002100399A1 (en) * | 2001-06-12 | 2002-12-19 | Elan Pharmaceuticals, Inc. | Macrocycles useful in the treatment of alzheimer's disease |
| SE0202430D0 (sv) | 2002-08-14 | 2002-08-14 | Astrazeneca Ab | New Compounds |
| AU2003255993A1 (en) * | 2002-09-10 | 2004-04-30 | Pfizer Products Inc. | Diazabicyclic compounds useful in the treatment of cns and other disorders |
| DE60326894D1 (de) | 2002-09-30 | 2009-05-07 | Neurosearch As | 1,4-Diazabicycloalkanderivate, deren Herstellung und Verwendung |
| ATE345342T1 (de) | 2002-11-11 | 2006-12-15 | Neurosearch As | 1,4-dizabicyclo(3,2,2)nonane derivative, verfahren zur ihre herstellung und therapeutical verwendung |
| US7223753B2 (en) * | 2002-11-11 | 2007-05-29 | Neurosearch A/S | Diazabicyclic biaryl derivatives |
| KR20060125885A (ko) * | 2004-02-04 | 2006-12-06 | 뉴로서치 에이/에스 | 콜린 수용체 조절제로서의 디아자바이사이클릭 아릴 유도체 |
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| WO2009024515A1 (en) | 2007-08-17 | 2009-02-26 | Neurosearch A/S | 1,4-diaza-bicycl0(3.2.2)n0nyl pyrimidinyl derivatives useful as nicotinic acetylcholine- receptor ligands |
| JP2011503144A (ja) * | 2007-11-14 | 2011-01-27 | ノイロサーチ アクティーゼルスカブ | 新規の１，４−ジアザ−ビシクロ［３．２．２］ノニルピリミジン誘導体及びその医療への使用 |
| JP2011503146A (ja) * | 2007-11-14 | 2011-01-27 | ノイロサーチ アクティーゼルスカブ | 新規な１，４−ジアザ−ビシクロ［３．２．２］ノニルピリミジン誘導体及びこれらの医療上の使用 |
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2007
- 2007-05-29 AU AU2007267178A patent/AU2007267178A1/en not_active Abandoned
- 2007-05-29 AU AU2007267177A patent/AU2007267177A1/en not_active Abandoned
- 2007-05-29 EP EP07729593A patent/EP2049538A1/en not_active Withdrawn
- 2007-05-29 MX MX2008014890A patent/MX2008014890A/es not_active Application Discontinuation
- 2007-05-29 CA CA002653460A patent/CA2653460A1/en not_active Abandoned
- 2007-05-29 EP EP07729594A patent/EP2029595B1/en not_active Not-in-force
- 2007-05-29 JP JP2009512571A patent/JP2009538869A/ja not_active Abandoned
- 2007-05-29 CA CA002653681A patent/CA2653681A1/en not_active Abandoned
- 2007-05-29 WO PCT/EP2007/055171 patent/WO2007138040A1/en not_active Ceased
- 2007-05-29 CA CA002653371A patent/CA2653371A1/en not_active Abandoned
- 2007-05-29 US US12/299,114 patent/US7915272B2/en not_active Expired - Fee Related
- 2007-05-29 MX MX2008014889A patent/MX2008014889A/es not_active Application Discontinuation
- 2007-05-29 EP EP07729592A patent/EP2041134A1/en not_active Withdrawn
- 2007-05-29 WO PCT/EP2007/055172 patent/WO2007138041A1/en not_active Ceased
- 2007-05-29 WO PCT/EP2007/055170 patent/WO2007138039A1/en not_active Ceased
- 2007-05-29 JP JP2009512572A patent/JP2009538870A/ja not_active Abandoned
- 2007-05-29 JP JP2009512570A patent/JP2009538868A/ja not_active Abandoned
- 2007-05-29 AU AU2007267176A patent/AU2007267176A1/en not_active Abandoned
- 2007-05-29 MX MX2008014885A patent/MX2008014885A/es not_active Application Discontinuation
- 2007-05-29 US US12/299,108 patent/US20090197872A1/en not_active Abandoned
- 2007-05-29 US US12/299,106 patent/US8148365B2/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| US20090197872A1 (en) | 2009-08-06 |
| AU2007267178A1 (en) | 2007-12-06 |
| JP2009538868A (ja) | 2009-11-12 |
| EP2029595A1 (en) | 2009-03-04 |
| JP2009538869A (ja) | 2009-11-12 |
| WO2007138041A8 (en) | 2008-11-20 |
| WO2007138039A1 (en) | 2007-12-06 |
| CA2653460A1 (en) | 2007-12-06 |
| JP2009538870A (ja) | 2009-11-12 |
| AU2007267176A1 (en) | 2007-12-06 |
| EP2029595B1 (en) | 2011-09-21 |
| MX2008014889A (es) | 2008-12-05 |
| CA2653371A1 (en) | 2007-12-06 |
| AU2007267177A1 (en) | 2007-12-06 |
| WO2007138040A8 (en) | 2008-11-20 |
| WO2007138041A1 (en) | 2007-12-06 |
| US20090270403A1 (en) | 2009-10-29 |
| EP2041134A1 (en) | 2009-04-01 |
| MX2008014885A (es) | 2008-12-05 |
| US8148365B2 (en) | 2012-04-03 |
| EP2049538A1 (en) | 2009-04-22 |
| US7915272B2 (en) | 2011-03-29 |
| WO2007138040A1 (en) | 2007-12-06 |
| US20090181984A1 (en) | 2009-07-16 |
| CA2653681A1 (en) | 2007-12-06 |
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| Date | Code | Title | Description |
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| FA | Abandonment or withdrawal |