ME02317B - Neuroprotekcija kod demijelinizacijskih bolesti - Google Patents

Neuroprotekcija kod demijelinizacijskih bolesti

Info

Publication number
ME02317B
ME02317B MEP-2015-212A MEP21215A ME02317B ME 02317 B ME02317 B ME 02317B ME P21215 A MEP21215 A ME P21215A ME 02317 B ME02317 B ME 02317B
Authority
ME
Montenegro
Prior art keywords
combination therapy
accordance
dmf
intended
interferon
Prior art date
Application number
MEP-2015-212A
Other languages
English (en)
Inventor
Susan Goelz
Kate Dawson
Ralf Linker
Ralf Gold
Original Assignee
Biogen Ma Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=44368163&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ME02317(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Biogen Ma Inc filed Critical Biogen Ma Inc
Publication of ME02317B publication Critical patent/ME02317B/me

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/21Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • A61K31/22Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin
    • A61K31/225Polycarboxylic acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/194Carboxylic acids, e.g. valproic acid having two or more carboxyl groups, e.g. succinic, maleic or phthalic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/74Synthetic polymeric materials
    • A61K31/785Polymers containing nitrogen
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/02Peptides of undefined number of amino acids; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/16Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/19Cytokines; Lymphokines; Interferons
    • A61K38/21Interferons [IFN]
    • A61K38/215IFN-beta
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2072Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/284Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
    • A61K9/2846Poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4808Preparations in capsules, e.g. of gelatin, of chocolate characterised by the form of the capsule or the structure of the filling; Capsules containing small tablets; Capsules with outer layer for immediate drug release
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Immunology (AREA)
  • Emergency Medicine (AREA)
  • Zoology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Biomedical Technology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Claims (15)

1. Kombinacijska terapija koja se sastoji od (a) dimetil-fumarata (DMF) i/ili monometil-fumarata (MMF) i (b) glatiramer-acetata, naznačena time što je namijenjen upotrebi u liječenju subjekta koji ima multiplu sklerozu (MS).
2. Kombinacijska terapija namijenjena upotrebi u skladu s patentnim zahtjevom 1, naznačena time što na subjektu treba primijeniti 20 mg dnevno glatiramer-acetata.
3. Kombinacijska terapija namijenjena upotrebi u skladu s patentnim zahtjevom 1, naznačena time što na subjektu treba primijeniti manje od 20 mg dnevno glatiramer-acetata.
4. Kombinacijska terapija namijenjena upotrebi u skladu s bilo kojim od prethodnih patentnih zahtjeva, naznačena time što su DMF i/ili MMF i glatiramer-acetat namijenjeni upotrebi u (i) smanjivanju stope recidiva kod subjekta; ili (ii) smanjivanju demijeliniziranje i/ili smrt aksona kod subjekta.
5. Kombinacijska terapija namijenjena upotrebi u skladu s bilo kojim od prethodnih patentnih zahtjeva, naznačena time što su DMF i/ili MMF i glatiramer-acetat formulirani u isti oblik doziranja.
6. Kombinacijska terapija namijenjena upotrebi u skladu s bilo kojim od patentnim zahtjevima 1 do 4, naznačena time što su DMF i/ili MMF i glatiramer-acetat formulirani u odvojene oblike doziranja namijenjene primjeni odvojeno ili zajedno.
7. Kombinacijska terapija koja se sastoji od (a) DMF i/ili MMF i (b) interferona-β, naznačena time što je namijenjena upotrebi u liječenju subjekta koji ima MS.
8. Kombinacijska terapija namijenjena upotrebi u skladu s patentnim zahtjevom 7, naznačena time što se interferon-β bira između interferona-β1a i interferona-β1b.
9. Kombinacijska terapija namijenjena upotrebi u skladu s patentnim zahtjevom 8, naznačena time što je interferon-β interferon-β1a.
10. Kombinacijska terapija namijenjena upotrebi u skladu s patentnim zahtjevom 9, naznačena time što interferon-β1a treba primijeniti u dozi od 5 µg do 80 µg odjednom.
11. Kombinacijska terapija namijenjena upotrebi u skladu s patentnim zahtjevom 10, naznačena time što interferon-β1a treba primijeniti jednom tjedno.
12. Kombinacijska terapija namijenjena upotrebi u skladu s bilo kojim od prethodnih patentnih zahtjeva, naznačena time što se MS bira između recidivirajući remitirajući MS, sekundarni progresivni MS, primarni progresivni MS, progresivni recidivirajući MS, te klinički izolirani sindrom.
13. Kombinacijska terapija namijenjena upotrebi u skladu s bilo kojim od prethodnih patentnih zahtjeva, naznačena time što je spoj koji se bira između DMF, MMF i njihovih kombinacija DMF.
14. Kombinacijska terapija namijenjena upotrebi u skladu s patentnim zahtjevom 13, naznačena time što na subjektu treba odjednom primijeniti 240 mg DMF.
15. Kombinacijska terapija namijenjena upotrebi u skladu s patentnim zahtjevom 14, naznačena time što DMF na subjektu treba primijeniti dva puta dnevno (BID), što je ekvivalent ukupnoj dnevnoj dozi od 480 mg dnevno.
MEP-2015-212A 2010-02-12 2011-02-11 Neuroprotekcija kod demijelinizacijskih bolesti ME02317B (me)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US30432510P 2010-02-12 2010-02-12
US32148610P 2010-04-06 2010-04-06
EP11742896.1A EP2533634B1 (en) 2010-02-12 2011-02-11 Neuroprotection in demyelinating diseases
PCT/US2011/024594 WO2011100589A1 (en) 2010-02-12 2011-02-11 Neuroprotection in demyelinating diseases

Publications (1)

Publication Number Publication Date
ME02317B true ME02317B (me) 2016-06-20

Family

ID=44368163

Family Applications (1)

Application Number Title Priority Date Filing Date
MEP-2015-212A ME02317B (me) 2010-02-12 2011-02-11 Neuroprotekcija kod demijelinizacijskih bolesti

Country Status (13)

Country Link
US (3) US20130287732A1 (me)
EP (2) EP2533634B1 (me)
DK (1) DK2533634T3 (me)
ES (1) ES2555279T3 (me)
HR (1) HRP20151350T1 (me)
HU (1) HUE025878T2 (me)
ME (1) ME02317B (me)
PL (1) PL2533634T3 (me)
PT (1) PT2533634E (me)
RS (1) RS54551B1 (me)
SI (1) SI2533634T1 (me)
SM (1) SMT201600014B (me)
WO (1) WO2011100589A1 (me)

Families Citing this family (30)

* Cited by examiner, † Cited by third party
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SI1663197T1 (sl) 2003-09-09 2008-06-30 Biogen Idec Internat Gmbh Uporaba derivatov fumarne kisline za zdravljenje sräśne insuficience in astme
ES2582942T3 (es) 2004-10-08 2016-09-16 Forward Pharma A/S Composiciones farmacéuticas de liberación controlada que comprenden un éster de ácido fumárico
PL2137537T3 (pl) 2007-02-08 2013-10-31 Biogen Ma Inc Kompozycje i zastosowania do leczenia stwardnienia rozsianego
US20100130607A1 (en) * 2007-02-08 2010-05-27 Ralf Gold Neuroprotection in demyelinating diseases
EP2379063B2 (en) 2009-01-09 2021-02-24 Fwp Ip Aps Pharmaceutical formulation comprising one or more fumaric acid esters in an erosion matrix
EA201391638A1 (ru) 2011-06-08 2014-05-30 Байоджен Айдек Ма Инк. Способ получения высокочистого и кристаллического диметилфумарата
US20130158077A1 (en) 2011-12-19 2013-06-20 Ares Trading S.A. Pharmaceutical compositions
US9504679B2 (en) 2011-12-19 2016-11-29 Bjoern Colin Kahrs Pharmaceutical compositions comprising glitazones and Nrf2 activators
KR102105217B1 (ko) * 2012-02-07 2020-06-01 바이오젠 엠에이 인코포레이티드 다이메틸 푸마레이트를 함유하는 약학 조성물
US20130259856A1 (en) * 2012-03-27 2013-10-03 Teva Pharmaceutical Industries, Ltd. Treatment of multiple sclerosis with combination of laquinimod and dimethyl fumarate
EP2692343A1 (en) 2012-08-03 2014-02-05 Forward Pharma A/S Combination therapy for treatment of multiple sclerosis
US10945984B2 (en) 2012-08-22 2021-03-16 Arbor Pharmaceuticals, Llc Methods of administering monomethyl fumarate and prodrugs thereof having reduced side effects
EP2887933A1 (en) 2012-08-22 2015-07-01 XenoPort, Inc. Oral dosage forms of methyl hydrogen fumarate and prodrugs thereof
UA119032C2 (uk) * 2012-10-02 2019-04-25 Женеро Са Фармацевтична композиція для лікування блокади ремієлінізації при захворюваннях, які пов'язані з експресією білка оболонки herv-w
EP3566701A1 (en) 2012-12-21 2019-11-13 Biogen MA Inc. Deuterium substituted fumarate derivatives
US8669281B1 (en) 2013-03-14 2014-03-11 Alkermes Pharma Ireland Limited Prodrugs of fumarates and their use in treating various diseases
JP6373353B2 (ja) 2013-03-14 2018-08-15 アルカーメス ファーマ アイルランド リミテッド フマル酸エステルのプロドラッグおよび種々の疾患の治療におけるその使用
US10179118B2 (en) 2013-03-24 2019-01-15 Arbor Pharmaceuticals, Llc Pharmaceutical compositions of dimethyl fumarate
US9421182B2 (en) 2013-06-21 2016-08-23 Xenoport, Inc. Cocrystals of dimethyl fumarate
WO2015035184A1 (en) 2013-09-06 2015-03-12 Xenoport, Inc. Crystalline forms of (n,n-diethylcarbamoyl)methyl methyl (2e)but-2-ene-1,4-dioate, methods of synthesis and use
WO2015105757A1 (en) * 2014-01-07 2015-07-16 Biogen Ma Inc. Dimethyl fumarate for treating multiple sclerosis
WO2015127450A1 (en) 2014-02-24 2015-08-27 Alkermes Pharma Ireland Limited Sulfonamide and sulfinamide prodrugs of fumarates and their use in treating various diseases
US9999672B2 (en) 2014-03-24 2018-06-19 Xenoport, Inc. Pharmaceutical compositions of fumaric acid esters
MA40982A (fr) * 2014-11-19 2017-09-26 Biogen Ma Inc Formulation de bille pharmaceutique comprenant du fumarate de diméthyle
MA41785A (fr) 2015-03-20 2018-01-23 Biogen Ma Inc Procédés et compositions pour l'administration intraveineuse de fumarates pour le traitement de maladies neurologiques
US12097292B2 (en) 2016-08-28 2024-09-24 Mapi Pharma Ltd. Process for preparing microparticles containing glatiramer acetate
FI3506921T3 (fi) 2016-08-31 2023-07-21 Mapi Pharma Ltd Glatirameeriasetaattia käsittäviä depot-järjestelmiä
MX2019010174A (es) 2017-03-26 2019-10-15 Mapi Pharma Ltd Sistemas de deposito de glatiramer para el tratamiento de formas progresivas de esclerosis multiple.
US11382889B2 (en) * 2018-04-19 2022-07-12 Institut D'investigació Biomèdica De Bellvitge (Idibell) NRF2 activators for the prevention and/or treatment of axonal degeneration
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DE19853487A1 (de) * 1998-11-19 2000-05-25 Fumapharm Ag Muri Verwendung von Dialkylfumaraten
ES2582942T3 (es) 2004-10-08 2016-09-16 Forward Pharma A/S Composiciones farmacéuticas de liberación controlada que comprenden un éster de ácido fumárico
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US20080089861A1 (en) * 2006-07-10 2008-04-17 Went Gregory T Combination therapy for treatment of demyelinating conditions
US20100130607A1 (en) 2007-02-08 2010-05-27 Ralf Gold Neuroprotection in demyelinating diseases
US20090104142A1 (en) * 2007-10-17 2009-04-23 Txcell Compositions for treating multiple sclerosis

Also Published As

Publication number Publication date
HRP20151350T1 (hr) 2016-01-01
PL2533634T3 (pl) 2016-04-29
EP2533634B1 (en) 2015-10-21
EP2533634A4 (en) 2013-07-10
US20160250172A1 (en) 2016-09-01
SI2533634T1 (sl) 2016-01-29
SMT201600014B (me) 2016-02-25
US20130287732A1 (en) 2013-10-31
PT2533634E (pt) 2015-12-28
RS54551B1 (sr) 2016-06-30
HUE025878T2 (en) 2016-05-30
EP2533634A1 (en) 2012-12-19
WO2011100589A1 (en) 2011-08-18
HK1179116A1 (en) 2013-09-27
DK2533634T3 (en) 2016-01-25
ES2555279T3 (es) 2015-12-30
EP2982371A1 (en) 2016-02-10
US20180021288A1 (en) 2018-01-25

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