MD2939F1 - Saliciliden tiosemicarbazido-[6-(4-aminobenzensulfamido)-3-metoxipiridazin]-nichel - Google Patents
Saliciliden tiosemicarbazido-[6-(4-aminobenzensulfamido)-3-metoxipiridazin]-nichel Download PDFInfo
- Publication number
- MD2939F1 MD2939F1 MDA20050013A MD20050013A MD2939F1 MD 2939 F1 MD2939 F1 MD 2939F1 MD A20050013 A MDA20050013 A MD A20050013A MD 20050013 A MD20050013 A MD 20050013A MD 2939 F1 MD2939 F1 MD 2939F1
- Authority
- MD
- Moldova
- Prior art keywords
- gram
- nickel
- activity against
- medicine
- methoxypyridazine
- Prior art date
Links
- PXHVJJICTQNCMI-UHFFFAOYSA-N nickel Substances [Ni] PXHVJJICTQNCMI-UHFFFAOYSA-N 0.000 title abstract 4
- 229910052759 nickel Inorganic materials 0.000 title abstract 3
- 239000003814 drug Substances 0.000 abstract 3
- 230000000844 anti-bacterial effect Effects 0.000 abstract 2
- 230000000845 anti-microbial effect Effects 0.000 abstract 2
- 230000003385 bacteriostatic effect Effects 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- 244000005700 microbiome Species 0.000 abstract 2
- 241000295644 Staphylococcaceae Species 0.000 abstract 1
- 239000004599 antimicrobial Substances 0.000 abstract 1
- 230000015572 biosynthetic process Effects 0.000 abstract 1
- 238000002360 preparation method Methods 0.000 abstract 1
- 238000001228 spectrum Methods 0.000 abstract 1
- 238000003786 synthesis reaction Methods 0.000 abstract 1
- 229910052723 transition metal Inorganic materials 0.000 abstract 1
- 150000003624 transition metals Chemical class 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Inventia se refera la chimie si medicina, si anume la un compus coordinativ de nichel biologic activ din clasa salicilidentiosemicarbazidatilor metalelor de tranzitie si poate gasi aplicare in medicina si in medicina veterinara in calitate de preparat antimicrobian.Esenta inventiei consta in sinteza salicilidentiosemicarbazido-[6-(4-aminobenzen-sulfamido)-3-metoxipiridazin]-nichelului cu formula:Compusul obtinut manifesta activitate bacteriostatica si bactericida inalta fata de un spectru larg de microorganisme gram-pozitive si gram-negative, totodata activitatea antimicrobiana fata de stafilococi si streptococi este de 2,6...41,6 ori mai inalta decat la analog si de 2,4...240 ori depaseste activitatea lui bacteriostatica si bactericida fata de microorganismele gram-negative.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| MDA20050013A MD2939G2 (ro) | 2005-01-11 | 2005-01-11 | Salicilidentiosemicarbazido-[6-(4-aminobenzensulfamido)-3-metoxipiridazin]-nichel |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| MDA20050013A MD2939G2 (ro) | 2005-01-11 | 2005-01-11 | Salicilidentiosemicarbazido-[6-(4-aminobenzensulfamido)-3-metoxipiridazin]-nichel |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| MD2939F1 true MD2939F1 (ro) | 2005-12-31 |
| MD2939G2 MD2939G2 (ro) | 2006-06-30 |
Family
ID=35508823
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MDA20050013A MD2939G2 (ro) | 2005-01-11 | 2005-01-11 | Salicilidentiosemicarbazido-[6-(4-aminobenzensulfamido)-3-metoxipiridazin]-nichel |
Country Status (1)
| Country | Link |
|---|---|
| MD (1) | MD2939G2 (ro) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MD4462C1 (ro) * | 2016-02-29 | 2017-08-31 | Государственный Университет Молд0 | Cloro-{N-(3,4-dimetilfenil)-2-[1-(2-hidroxifenil)etiliden]-hidrazincarbotioamido(1-)}nichel, care manifestă activitate antimicrobiană faţă de bacteriile din speciile Klebsiella pneumoniae şi Pseudomonas aeruginosa |
-
2005
- 2005-01-11 MD MDA20050013A patent/MD2939G2/ro not_active IP Right Cessation
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MD4462C1 (ro) * | 2016-02-29 | 2017-08-31 | Государственный Университет Молд0 | Cloro-{N-(3,4-dimetilfenil)-2-[1-(2-hidroxifenil)etiliden]-hidrazincarbotioamido(1-)}nichel, care manifestă activitate antimicrobiană faţă de bacteriile din speciile Klebsiella pneumoniae şi Pseudomonas aeruginosa |
Also Published As
| Publication number | Publication date |
|---|---|
| MD2939G2 (ro) | 2006-06-30 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FG4A | Patent for invention issued | ||
| KA4A | Patent for invention lapsed due to non-payment of fees (with right of restoration) | ||
| MM4A | Patent for invention definitely lapsed due to non-payment of fees |