MC666A1 - Amidino-urées et leur préparation - Google Patents

Amidino-urées et leur préparation

Info

Publication number
MC666A1
MC666A1 MC705A MC705A MC666A1 MC 666 A1 MC666 A1 MC 666A1 MC 705 A MC705 A MC 705A MC 705 A MC705 A MC 705A MC 666 A1 MC666 A1 MC 666A1
Authority
MC
Monaco
Prior art keywords
group
formula
halogen
chloro
nitrile
Prior art date
Application number
MC705A
Other languages
English (en)
French (fr)
Original Assignee
Wellcome Found
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wellcome Found filed Critical Wellcome Found
Publication of MC666A1 publication Critical patent/MC666A1/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C279/00Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups
    • C07C279/20Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups containing any of the groups, X being a hetero atom, Y being any atom, e.g. acylguanidines
    • C07C279/24Y being a hetero atom
    • C07C279/26X and Y being nitrogen atoms, i.e. biguanides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Structures Of Non-Positive Displacement Pumps (AREA)
MC705A 1966-07-07 1967-07-06 Amidino-urées et leur préparation MC666A1 (fr)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GB19028/67A GB1194835A (en) 1966-07-07 1966-07-07 Novel 1-Amidino-3-Phenyl-Urea Derivatives, the preparation thereof and Compositions containing the same
GB3047966 1966-07-07
GB5654666 1966-12-16
GB539167 1967-02-03

Publications (1)

Publication Number Publication Date
MC666A1 true MC666A1 (fr) 1968-04-01

Family

ID=27447446

Family Applications (1)

Application Number Title Priority Date Filing Date
MC705A MC666A1 (fr) 1966-07-07 1967-07-06 Amidino-urées et leur préparation

Country Status (15)

Country Link
US (2) US3539616A (forum.php)
BE (1) BE700895A (forum.php)
CA (1) CA947316A (forum.php)
CH (5) CH501599A (forum.php)
DE (2) DE1668843A1 (forum.php)
DK (1) DK125705B (forum.php)
FR (2) FR1548340A (forum.php)
GB (1) GB1194835A (forum.php)
IL (1) IL28189A (forum.php)
LU (1) LU54053A1 (forum.php)
MC (1) MC666A1 (forum.php)
NL (1) NL6709484A (forum.php)
NO (1) NO126225B (forum.php)
OA (1) OA02467A (forum.php)
SE (1) SE330010B (forum.php)

Families Citing this family (29)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3761597A (en) * 1967-06-30 1973-09-25 L Walls 1-amidino-3-(substituted-phenyl) urea antimalarial composition and method of use
IL37047A0 (en) * 1970-06-30 1971-08-25 Wellcome Found Substituted amidines,their preparation and pharmaceutical compositions containing them
US4025652A (en) * 1975-03-31 1977-05-24 William H. Rorer, Inc. Amidinoureas
US4220658A (en) * 1972-09-22 1980-09-02 William H. Rorer, Inc. Treatment of hypertension with amidinoureas
US4488993A (en) * 1972-09-22 1984-12-18 William H. Rorer, Inc. Amidinoureas
US4326074A (en) * 1972-09-22 1982-04-20 William H. Rorer, Inc. Amidinoureas
FR2223361B1 (forum.php) * 1973-03-27 1977-04-29 Philagro Sa
JPS5646157B2 (forum.php) * 1973-06-05 1981-10-31
GB1480643A (en) * 1973-07-16 1977-07-20 Rorer Inc William H Amidino-phenyl-ureas processes for their preparation and compositions incorporating them
US4060635A (en) * 1975-03-31 1977-11-29 William H. Rorer, Inc. Amidinoureas for treating diarrhea
US4283555A (en) * 1973-07-16 1981-08-11 William H. Rorer, Inc. Amidinoureas
US4216229A (en) * 1973-07-16 1980-08-05 William H. Rorer, Inc. Method for treating gastrointestinal hyperacidity or ulceration with amidinoureas
US4150154A (en) * 1975-03-03 1979-04-17 William H. Rorer, Inc. Amidinoureas
US4216230A (en) * 1973-07-16 1980-08-05 William H. Rorer, Inc. Method for alleviating hypertension with amidinoureas
ZA743750B (en) * 1973-07-16 1975-06-25 Rorer Inc William H Amindinoureas
US4203920A (en) * 1975-03-31 1980-05-20 William H. Rorer, Inc. Amidinoureas
US4204000A (en) * 1975-03-31 1980-05-20 William H. Rorer, Inc. Anti-ulcer amidinoureas
US4242337A (en) * 1976-03-30 1980-12-30 William H. Rorer, Inc. Method for treatment of diarrheal disease conditions or symptons in mammals
US4058557A (en) * 1976-03-30 1977-11-15 William H. Rorer, Inc. Amidinoureas
US4242339A (en) * 1976-03-30 1980-12-30 William H. Rorer, Inc. Method for treatment of gastrointestinal spasmodic disease conditions or symptoms in mammals
US4353842A (en) * 1978-09-14 1982-10-12 William H. Rorer, Inc. Amidinoureas
US4440949A (en) * 1979-01-08 1984-04-03 William H. Rorer, Inc. Amidinoureas
US4340609A (en) * 1980-01-02 1982-07-20 William H. Rorer, Inc. Amidinourea derivative veterinary compositions for suppression of parasitemia
NL8120313A (nl) * 1981-08-24 1983-07-01 Rorer Int Overseas Heterocyclische amidino-gesubstitueerde ureums en de farmaceutische toepassingen daarvan.
WO1986004935A1 (en) * 1985-02-15 1986-08-28 Rorer International (Overseas) Inc. Amidinourea process and pharmaceutical composition
DE4412079A1 (de) * 1993-08-18 1995-02-23 Bayer Ag N-Cyanoaryl-Stickstoffheterocyclen
US5681794A (en) * 1993-08-18 1997-10-28 Bayer Aktiengesellschaft N-cyanoaryl-nitrogen heterocycles
ES2110667T3 (es) * 1993-08-18 1998-02-16 Bayer Ag N-cianoaril-heterociclos nitrogenados.
DE4335438A1 (de) * 1993-10-18 1995-04-20 Bayer Ag 4-Cyanophenyliminoheterocyclen

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3119867A (en) * 1962-01-26 1964-01-28 Clairol Inc Amino, nitro-phenyl-biguanides and amino, nitro-phenyl; guanyl-ureas

Also Published As

Publication number Publication date
DK125705B (da) 1973-03-26
CH500952A (de) 1970-12-31
NO126225B (forum.php) 1973-01-08
DE1668843A1 (de) 1972-02-24
CH501598A (de) 1971-01-15
IL28189A (en) 1971-04-28
US3784582A (en) 1974-01-08
NL6709484A (forum.php) 1968-01-08
FR7055M (forum.php) 1969-06-23
SE330010B (forum.php) 1970-11-02
US3539616A (en) 1970-11-10
CH554318A (de) 1974-09-30
CH501597A (de) 1971-01-15
OA02467A (fr) 1970-05-05
CA947316A (en) 1974-05-14
GB1194835A (en) 1970-06-10
CH501599A (de) 1971-01-15
FR1548340A (forum.php) 1968-12-06
DE1793745A1 (de) 1973-05-30
BE700895A (forum.php) 1968-01-04
LU54053A1 (forum.php) 1968-03-12

Similar Documents

Publication Publication Date Title
MC666A1 (fr) Amidino-urées et leur préparation
EP0172096B1 (fr) Dérivés d'acylaminométhyl-3 imidazo[1,2-a]pyridines, leur préparation et leur application en thérapeutique
CH643546A5 (fr) Procede pour la preparation de derives d'hydantoine.
FR2561647A1 (fr) Derives de 1-(hydroxymethyl)-1,6,7,11b-tetrahydro-2h,4h-(1,3)-oxazino- ou -thiazino(4,3,a)isoquinoleine, procede pour leur preparation et compositions pharmaceutiques les contenant
EP0110781A1 (fr) (Amino-2 éthyl)-6 benzoxazolinones substituées, leur préparation et une composition pharmaceutique les contenant
AU2001280004A1 (en) Substituted phthalides as anti-convulsive drugs
EP1242389B1 (fr) Nouveaux derives amino substitues ramifies du 3-amino-1-phenyl-1h[1,2,4]triazole, procedes pour leur preparation et compositions pharmaceutiques les contenant
FR2676057A1 (fr) Derives de 1,2-dithiole-3-thione, procede de preparation de ces derives, ainsi que l'utilisation de ces derives comme intermediaires de synthese ou comme medicaments.
MC528A1 (fr) Nouvelles benzenesulfonyl-urées et leur préparation
EP0246126A1 (fr) Benzimidazoles et imidazopyridines sulfonamides, leur préparation et leur application en tant que médicaments
FR2491064A1 (fr) Quinolones, leurs procedes de preparation et composition therapeutique les contenant
EP1486503B1 (fr) Dérivés de benzothiazine et benzothiadiazine, leur procédé de préparation et les compositions pharmaceutiques qui les contiennent
EP0280603A1 (fr) Enantiomères de configuration absolue S de dérivés amide de l'amino-3 quinuclidine, leur procédé de préparation et leur application en thérapeutique
FR2492821A1 (fr) Derives de la pyrimidine, leur procede de preparation et les compositions pharmaceutiques les contenant
CA2010529A1 (fr) Derives de la 1-arylsulfonyl 2-piperidinone, leur procede et les intermediaires de preparation, leur application comme medicaments et les compositions les renfermant
MC593A1 (fr) Nouveaux benzène sulfonyl-semicarbazides et leur préparation
EP0105881B1 (fr) Nouvelles cyanoguanidines, leur procede d'obtention et les compositions pharmaceutiques en renfermant
FR2560193A1 (fr) Derives d'aminodiaryl sulfoxyde, procede pour leur preparation et compositions pharmaceutiques et pesticides les contenant
MC546A1 (fr) Nouvelles benzène-sufonyl-urées et leur préparation
FR2653999A1 (fr) Nouveaux derives de la morpholine, leur procede de preparation et les compositions pharmaceutiques les renfermant.
EP0433163A2 (fr) Nouveau procédé de préparation d'imidazobenzodiazépines et de leurs sels
CA1068270A (fr) Diamino-2,4-bromo-5 chloro-6 pyrimidines utilisables comme medicaments et procede pour leur preparation
FR2807754A1 (fr) Nouveaux derives de cyclobuta-indole carboxamide, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
EP0220104A2 (fr) Dérivés d'amino-5 pentanenitrile, leurs procédés de préparation et les compositions pharmaceutiques qui les contiennent
MC682A1 (fr) Benzène-sulfonyl-urées et leur préparation