MC509A1 - Nouveaux benzylsulfamides substitués et leur préparation - Google Patents
Nouveaux benzylsulfamides substitués et leur préparationInfo
- Publication number
- MC509A1 MC509A1 MC538A MC538A MC509A1 MC 509 A1 MC509 A1 MC 509A1 MC 538 A MC538 A MC 538A MC 538 A MC538 A MC 538A MC 509 A1 MC509 A1 MC 509A1
- Authority
- MC
- Monaco
- Prior art keywords
- sulfamide
- methyl
- amine
- prepared
- trichlorobenzyl
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/16—Amides, e.g. hydroxamic acids
- A61K31/18—Sulfonamides
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C307/00—Amides of sulfuric acids, i.e. compounds having singly-bound oxygen atoms of sulfate groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
- C07C307/02—Monoamides of sulfuric acids or esters thereof, e.g. sulfamic acids
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pyridine Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US33935464A | 1964-01-22 | 1964-01-22 | |
| US375288A US3320314A (en) | 1964-01-22 | 1964-06-15 | Chlorobenzyl sulfamides |
| US383507A US3351584A (en) | 1964-01-22 | 1964-07-17 | Nu-propargyl sulfamides |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MC509A1 true MC509A1 (fr) | 1965-08-27 |
Family
ID=27407336
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MC538A MC509A1 (fr) | 1964-01-22 | 1965-01-20 | Nouveaux benzylsulfamides substitués et leur préparation |
| MC537A MC508A1 (fr) | 1964-01-22 | 1965-01-20 | Nouveaux n-propargyl benzylsulfamides et leur préparation |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MC537A MC508A1 (fr) | 1964-01-22 | 1965-01-20 | Nouveaux n-propargyl benzylsulfamides et leur préparation |
Country Status (10)
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CH452504A (de) * | 1962-11-20 | 1968-03-15 | Ciba Geigy | Neues Sulfamid |
| US3475541A (en) * | 1967-06-13 | 1969-10-28 | Unimed Inc | Treatment of epilepsy with polyglycerols and polyglycerol esters |
| DE3234037A1 (de) * | 1982-09-14 | 1984-03-29 | Bayer Ag, 5090 Leverkusen | Jodpropargylsulfamide |
| IT1181871B (it) * | 1985-04-01 | 1987-09-30 | Consiglio Nazionale Ricerche | Inibitori selettivi delle benzilamminossidasi rispetto ad altre amminossidasi |
| MY147767A (en) | 2004-06-16 | 2013-01-31 | Janssen Pharmaceutica Nv | Novel sulfamate and sulfamide derivatives useful for the treatment of epilepsy and related disorders |
| EP1881959A1 (en) * | 2005-05-20 | 2008-01-30 | Janssen Pharmaceutica N.V. | Process for preparation of sulfamide derivatives |
| US8937096B2 (en) | 2005-12-19 | 2015-01-20 | Janssen Pharmaceutica Nv | Use of benzo-fused heterocyle sulfamide derivatives for the treatment of mania and bipolar disorder |
| US8691867B2 (en) | 2005-12-19 | 2014-04-08 | Janssen Pharmaceutica Nv | Use of benzo-fused heterocycle sulfamide derivatives for the treatment of substance abuse and addiction |
| US8716231B2 (en) | 2005-12-19 | 2014-05-06 | Janssen Pharmaceutica Nv | Use of benzo-fused heterocycle sulfamide derivatives for the treatment of pain |
| US8497298B2 (en) | 2005-12-19 | 2013-07-30 | Janssen Pharmaceutica Nv | Use of benzo-fused heterocycle sulfamide derivatives for lowering lipids and lowering blood glucose levels |
| AR058389A1 (es) | 2005-12-19 | 2008-01-30 | Janssen Pharmaceutica Nv | Uso de derivados heterociclicos benzo-fusionados de sulfamida para el tratamiento de la obesidad |
| EP2026790A2 (en) | 2006-05-19 | 2009-02-25 | Janssen Pharmaceutica, N.V. | Co-therapy for the treatment of epilepsy and related disorders |
| BRPI0915890A2 (pt) | 2008-06-23 | 2015-11-03 | Janssen Pharmaceutica Nv | forma cristalina de (2s)-(-)-n-(6-cloro-2,3-di-hidro-benzo[1,4]dioxin-2-ilmetil)-sulfamida |
| US8815939B2 (en) | 2008-07-22 | 2014-08-26 | Janssen Pharmaceutica Nv | Substituted sulfamide derivatives |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE947554C (de) * | 1953-09-18 | 1956-08-16 | Farbenwerke Hoechst Ag Vormals | Verfahren zur Herstellung von Derivaten des Sulfamids |
| GB789273A (en) * | 1955-04-07 | 1958-01-15 | Bayer Ag | Trichloro-methyl-mercaptan derivatives and production |
| BE636655A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) * | 1962-09-14 |
-
1964
- 1964-06-15 US US375288A patent/US3320314A/en not_active Expired - Lifetime
- 1964-07-17 US US383507A patent/US3351584A/en not_active Expired - Lifetime
-
1965
- 1965-01-11 CH CH34365A patent/CH456572A/de unknown
- 1965-01-11 CH CH34265A patent/CH456574A/de unknown
- 1965-01-12 GB GB1366/65A patent/GB1087934A/en not_active Expired
- 1965-01-15 NL NL6500481A patent/NL6500481A/xx unknown
- 1965-01-15 NL NL6500542A patent/NL6500542A/xx unknown
- 1965-01-19 GB GB2318/65A patent/GB1087602A/en not_active Expired
- 1965-01-19 DE DES95068A patent/DE1240846B/de active Pending
- 1965-01-19 DE DE19651518298 patent/DE1518298A1/de active Pending
- 1965-01-20 MC MC538A patent/MC509A1/fr unknown
- 1965-01-20 BE BE658587A patent/BE658587A/xx unknown
- 1965-01-20 MC MC537A patent/MC508A1/fr unknown
- 1965-01-20 BE BE658586A patent/BE658586A/xx unknown
- 1965-01-21 LU LU47821D patent/LU47821A1/xx unknown
- 1965-01-22 BR BR166384/65A patent/BR6566384D0/pt unknown
- 1965-01-22 LU LU47834D patent/LU47834A1/xx unknown
- 1965-01-22 OA OA51300A patent/OA01502A/xx unknown
- 1965-01-22 OA OA51299A patent/OA01501A/xx unknown
- 1965-01-22 BR BR166383/65A patent/BR6566383D0/pt unknown
Also Published As
| Publication number | Publication date |
|---|---|
| OA01501A (fr) | 1969-07-21 |
| CH456574A (de) | 1968-07-31 |
| US3351584A (en) | 1967-11-07 |
| CH456572A (de) | 1968-07-31 |
| LU47821A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1965-07-21 |
| DE1240846B (de) | 1967-05-24 |
| BE658586A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1965-07-20 |
| LU47834A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1965-07-22 |
| NL6500542A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1965-07-23 |
| OA01502A (fr) | 1969-07-21 |
| GB1087602A (en) | 1967-10-18 |
| BR6566384D0 (pt) | 1973-08-02 |
| MC508A1 (fr) | 1965-08-27 |
| DE1518298A1 (de) | 1969-07-24 |
| BE658587A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1965-07-20 |
| US3320314A (en) | 1967-05-16 |
| NL6500481A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1965-07-23 |
| GB1087934A (en) | 1967-10-18 |
| BR6566383D0 (pt) | 1973-08-02 |
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