MA56043A - Dérivés hétérocycliques fusionnés - Google Patents

Dérivés hétérocycliques fusionnés

Info

Publication number
MA56043A
MA56043A MA056043A MA56043A MA56043A MA 56043 A MA56043 A MA 56043A MA 056043 A MA056043 A MA 056043A MA 56043 A MA56043 A MA 56043A MA 56043 A MA56043 A MA 56043A
Authority
MA
Morocco
Prior art keywords
fused heterocyclic
heterocyclic derivatives
derivatives
fused
heterocyclic
Prior art date
Application number
MA056043A
Other languages
English (en)
Inventor
Jan Martin Berke
Zhanling Cheng
Gang Deng
Lindsey Graham Deratt
Sandrine Céline Grosse
Lili Hu
Yimin Jiang
Tim Hugo Maria Jonckers
Bart Rudolf Romanie Kesteleyn
Scott D Kuduk
Morgan Charles R Lecomte
Lamenca Carolina Martinez
Serge Maria Aloysius Pieters
Pierre Jean-Marie Bernard Raboisson
Koen Vandyck
Wim Gaston Verschueren
Yanping Xu
Original Assignee
Janssen Sciences Ireland Unlimited Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Sciences Ireland Unlimited Co filed Critical Janssen Sciences Ireland Unlimited Co
Publication of MA56043A publication Critical patent/MA56043A/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/12Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D498/14Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/551Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/20Antivirals for DNA viruses

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Virology (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biotechnology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Molecular Biology (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
MA056043A 2019-05-28 2020-05-27 Dérivés hétérocycliques fusionnés MA56043A (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201962853533P 2019-05-28 2019-05-28
EP19176933 2019-05-28
CN2020085720 2020-04-20

Publications (1)

Publication Number Publication Date
MA56043A true MA56043A (fr) 2022-04-06

Family

ID=71741889

Family Applications (1)

Application Number Title Priority Date Filing Date
MA056043A MA56043A (fr) 2019-05-28 2020-05-27 Dérivés hétérocycliques fusionnés

Country Status (17)

Country Link
EP (1) EP3976617A1 (fr)
JP (1) JP2022535734A (fr)
KR (1) KR20220012913A (fr)
CN (1) CN113906028A (fr)
AU (1) AU2020285718A1 (fr)
BR (1) BR112021022889A8 (fr)
CA (1) CA3138168A1 (fr)
CL (1) CL2021003155A1 (fr)
CO (1) CO2021016433A2 (fr)
CR (1) CR20210666A (fr)
IL (1) IL288322A (fr)
JO (1) JOP20210313A1 (fr)
MA (1) MA56043A (fr)
MX (1) MX2021014575A (fr)
PE (1) PE20220767A1 (fr)
SG (1) SG11202113167QA (fr)
WO (1) WO2020243135A1 (fr)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2022116999A1 (fr) * 2020-12-02 2022-06-09 Janssen Sciences Ireland Unlimited Company Dérivés hétérocycliques fusionnés et leur utilisation dans le traitement d'une infection par le vhb
CN116744927A (zh) * 2020-12-02 2023-09-12 杨森科学爱尔兰无限公司 稠合杂环衍生物及其在治疗hbv感染中的用途
WO2022116998A1 (fr) * 2020-12-02 2022-06-09 Janssen Sciences Ireland Unlimited Company Dérivés hétérocycliques fusionnés utilisés en tant qu'inhibiteurs du vhb
AR126048A1 (es) * 2021-06-02 2023-09-06 Janssen Sciences Ireland Unlimited Co Derivados heterocíclicos condensados
UY39794A (es) 2021-06-02 2022-11-30 Janssen Sciences Ireland Unlimited Co Derivados heterocíclicos condensados

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2993174A1 (fr) * 2014-09-08 2016-03-09 Helmholtz Zentrum München Deutsches Forschungszentrum für Gesundheit und Umwelt GmbH Dérivés de pyrazolopyridine et leur utilisation en thérapie
WO2016109684A2 (fr) * 2014-12-30 2016-07-07 Novira Therapeutics, Inc. Dérivés et méthodes de traitement d'infections provoquées par le virus de l'hépatite b
CN109641896B (zh) * 2016-06-29 2021-09-21 诺维拉治疗公司 二氮杂酮衍生物及其在治疗乙型肝炎感染中的用途
CN109843892B (zh) * 2016-06-29 2022-01-25 诺维拉治疗公司 噁二氮杂卓酮衍生物及其在治疗乙型肝炎感染中的用途

Also Published As

Publication number Publication date
JOP20210313A1 (ar) 2023-01-30
JP2022535734A (ja) 2022-08-10
CA3138168A1 (fr) 2020-12-03
KR20220012913A (ko) 2022-02-04
IL288322A (en) 2022-01-01
EP3976617A1 (fr) 2022-04-06
PE20220767A1 (es) 2022-05-16
BR112021022889A2 (pt) 2022-01-04
CN113906028A (zh) 2022-01-07
CR20210666A (es) 2022-03-11
AU2020285718A1 (en) 2022-02-03
BR112021022889A8 (pt) 2024-03-05
MX2021014575A (es) 2022-05-24
CL2021003155A1 (es) 2022-07-22
WO2020243135A1 (fr) 2020-12-03
CO2021016433A2 (es) 2021-12-10
SG11202113167QA (en) 2021-12-30

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