MA55074A - Dérivés de pyrazolopyridine utilisés comme inhibiteurs de pask - Google Patents

Dérivés de pyrazolopyridine utilisés comme inhibiteurs de pask

Info

Publication number
MA55074A
MA55074A MA055074A MA55074A MA55074A MA 55074 A MA55074 A MA 55074A MA 055074 A MA055074 A MA 055074A MA 55074 A MA55074 A MA 55074A MA 55074 A MA55074 A MA 55074A
Authority
MA
Morocco
Prior art keywords
pask
inhibitors
derivatives used
pyrazolopyridine derivatives
pyrazolopyridine
Prior art date
Application number
MA055074A
Other languages
English (en)
Inventor
Stéphane Nicolas Alain Beaumont
Xavier Marie Bock
Martinez Daniel Comas
Agnès Marie Joncour
Frédéric Gilbert Labéguère
Ramos Miriam López
Taoues Temal-Laïb
Original Assignee
Galapagos Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Galapagos Nv filed Critical Galapagos Nv
Publication of MA55074A publication Critical patent/MA55074A/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Endocrinology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
MA055074A 2019-02-25 2020-02-17 Dérivés de pyrazolopyridine utilisés comme inhibiteurs de pask MA55074A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB1902490.0A GB201902490D0 (en) 2019-02-25 2019-02-25 Novel compounds and pharmaceutical compositions thereof for the treatment of diseases

Publications (1)

Publication Number Publication Date
MA55074A true MA55074A (fr) 2022-01-05

Family

ID=65998935

Family Applications (1)

Application Number Title Priority Date Filing Date
MA055074A MA55074A (fr) 2019-02-25 2020-02-17 Dérivés de pyrazolopyridine utilisés comme inhibiteurs de pask

Country Status (18)

Country Link
US (1) US20220144823A1 (fr)
EP (1) EP3931191B1 (fr)
JP (1) JP2022525121A (fr)
KR (1) KR20210134001A (fr)
CN (1) CN113474344A (fr)
AR (1) AR124749A1 (fr)
AU (1) AU2020229041A1 (fr)
BR (1) BR112021016642A2 (fr)
CA (1) CA3130154A1 (fr)
CO (1) CO2021010485A2 (fr)
ES (1) ES2963409T3 (fr)
GB (1) GB201902490D0 (fr)
IL (1) IL285751A (fr)
MA (1) MA55074A (fr)
MX (1) MX2021010093A (fr)
SG (1) SG11202109157TA (fr)
TW (1) TW202045505A (fr)
WO (1) WO2020173739A1 (fr)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2022070288A1 (fr) * 2020-09-30 2022-04-07 旭化成ファーマ株式会社 Composé bicyclique contenant de l'azote

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2002088107A1 (fr) * 2001-04-26 2002-11-07 Eisai Co., Ltd. Compose azote a anneaux condenses possedant un groupe pyrazolyle et servant de substituant, et composition medicale le comprenant
US10392389B2 (en) * 2012-10-25 2019-08-27 Bioenergenix Llc Heterocyclic compounds for the inhibition of PASK

Also Published As

Publication number Publication date
IL285751A (en) 2021-10-31
AR124749A1 (es) 2023-05-03
SG11202109157TA (en) 2021-09-29
EP3931191B1 (fr) 2023-10-04
CA3130154A1 (fr) 2020-09-03
MX2021010093A (es) 2021-09-21
AU2020229041A1 (en) 2021-10-21
CN113474344A (zh) 2021-10-01
BR112021016642A2 (pt) 2021-11-03
GB201902490D0 (en) 2019-04-10
EP3931191A1 (fr) 2022-01-05
TW202045505A (zh) 2020-12-16
US20220144823A1 (en) 2022-05-12
ES2963409T3 (es) 2024-03-27
JP2022525121A (ja) 2022-05-11
CO2021010485A2 (es) 2021-08-19
KR20210134001A (ko) 2021-11-08
WO2020173739A1 (fr) 2020-09-03

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