MA31507B1 - Solutions pharmaceutiques orales contenant de la telbivudine - Google Patents

Solutions pharmaceutiques orales contenant de la telbivudine

Info

Publication number
MA31507B1
MA31507B1 MA32485A MA32485A MA31507B1 MA 31507 B1 MA31507 B1 MA 31507B1 MA 32485 A MA32485 A MA 32485A MA 32485 A MA32485 A MA 32485A MA 31507 B1 MA31507 B1 MA 31507B1
Authority
MA
Morocco
Prior art keywords
tilpifudine
oral medication
solutions contain
medication solutions
thymidine
Prior art date
Application number
MA32485A
Other languages
Arabic (ar)
English (en)
Inventor
Nabila Sekkat
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38724394&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MA31507(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of MA31507B1 publication Critical patent/MA31507B1/fr

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/08Solutions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0087Galenical forms not covered by A61K9/02 - A61K9/7023
    • A61K9/0095Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/513Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim having oxo groups directly attached to the heterocyclic ring, e.g. cytosine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/20Antivirals for DNA viruses

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Virology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Molecular Biology (AREA)
  • Biotechnology (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

L'invention porte sur une solution pharmaceutique, appropriée pour une administration orale, qui comporte de la ß-l-thymidine/2'-désoxy-l-thymidine (telbivudine), un système de solvant approprié du point de vue pharmaceutique, un ou plusieurs agents exhausteurs de goût/de masquage du goût, un système de conservateur et un système de tampon approprié pour permettre à la fois la stabilité et la conservation de médicament.
MA32485A 2007-07-12 2010-01-07 Solutions pharmaceutiques orales contenant de la telbivudine MA31507B1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP07112381 2007-07-12
PCT/EP2008/059016 WO2009007426A1 (fr) 2007-07-12 2008-07-10 Solutions pharmaceutiques orales contenant de la telbivudine

Publications (1)

Publication Number Publication Date
MA31507B1 true MA31507B1 (fr) 2010-07-01

Family

ID=38724394

Family Applications (1)

Application Number Title Priority Date Filing Date
MA32485A MA31507B1 (fr) 2007-07-12 2010-01-07 Solutions pharmaceutiques orales contenant de la telbivudine

Country Status (22)

Country Link
US (1) US8445457B2 (fr)
EP (1) EP2178503A1 (fr)
JP (1) JP5314014B2 (fr)
KR (3) KR20100029829A (fr)
CN (1) CN101686938B (fr)
AR (1) AR067630A1 (fr)
AU (1) AU2008274170B2 (fr)
BR (1) BRPI0815562A2 (fr)
CA (1) CA2693609A1 (fr)
CL (1) CL2008002025A1 (fr)
CO (1) CO6270204A2 (fr)
EC (1) ECSP109871A (fr)
IL (1) IL202961A (fr)
MA (1) MA31507B1 (fr)
MY (1) MY147366A (fr)
NZ (1) NZ582443A (fr)
PE (2) PE20130180A1 (fr)
RU (1) RU2493826C2 (fr)
TN (1) TN2010000008A1 (fr)
TW (1) TW200911302A (fr)
WO (1) WO2009007426A1 (fr)
ZA (1) ZA200908993B (fr)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RS55582B1 (sr) 2011-05-13 2017-06-30 Array Biopharma Inc Jedinjenja pirolidinil uree, pirolidinil tiouree i pirolidinil guanidina kao inhibitori trka kinaze
WO2014059363A1 (fr) * 2012-10-11 2014-04-17 Antrim Pharmaceuticals Llc Formulations de solution orale d'aripiprazole
NZ727418A (en) 2014-05-15 2023-03-31 Array Biopharma Inc 1-((3s,4r)-4-(3-fluorophenyl)-1-(2-methoxyethyl)pyrrolidin-3-yl)-3-(4-methyl-3-(2-methylpyrimidin-5-yl)-1-phenyl-1h-pyrazol-5-yl)urea as a trka kinase inhibitor
EP3288562B1 (fr) * 2015-04-26 2022-03-16 MacKay Memorial Hospital Procédé pour améliorer la fonction rénale et/ou cardiaque chez des patients atteints de maladie rénale
CN107550866A (zh) * 2016-06-30 2018-01-09 康普药业股份有限公司 一种替比夫定制剂

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5856364A (en) 1991-03-01 1999-01-05 Warner Lambert Company Therapeutic antiviral-wound healing compositions and methods for preparing and using same
EP1023899A1 (fr) 1997-09-26 2000-08-02 Wakamoto Pharmaceutical Co., Ltd. Preparation aqueuse contenant un agent antiviral a ossature purine ou pyrimidine
DE19817265A1 (de) 1998-04-18 1999-10-21 Bayer Ag Verwendung von Dihydropyrimidinen als Arzneimittel und neue Stoffe
DE19817264A1 (de) 1998-04-18 1999-10-21 Bayer Ag Neue Dihydropyrimidine
AR037131A1 (es) * 2001-10-31 2004-10-20 Schering Corp Formulaciones de jarabe de ribavirina
TWI244393B (en) * 2002-08-06 2005-12-01 Idenix Pharmaceuticals Inc Crystalline and amorphous forms of beta-L-2'-deoxythymidine
WO2006130217A2 (fr) 2005-04-01 2006-12-07 The Regents Of The University Of California Esters de phosphate de phosphonates de nucleosides substitues

Also Published As

Publication number Publication date
PE20130180A1 (es) 2013-03-06
CO6270204A2 (es) 2011-04-20
CN101686938B (zh) 2012-09-05
CL2008002025A1 (es) 2009-05-08
AU2008274170B2 (en) 2011-06-09
AR067630A1 (es) 2009-10-21
KR20100029829A (ko) 2010-03-17
MY147366A (en) 2012-11-30
EP2178503A1 (fr) 2010-04-28
CA2693609A1 (fr) 2009-01-15
CN101686938A (zh) 2010-03-31
ZA200908993B (en) 2010-09-29
PE20090476A1 (es) 2009-05-12
IL202961A (en) 2013-10-31
US8445457B2 (en) 2013-05-21
WO2009007426A1 (fr) 2009-01-15
JP2010533146A (ja) 2010-10-21
US20100197629A1 (en) 2010-08-05
JP5314014B2 (ja) 2013-10-16
TW200911302A (en) 2009-03-16
ECSP109871A (es) 2010-02-26
TN2010000008A1 (en) 2011-09-26
KR20140019040A (ko) 2014-02-13
RU2493826C2 (ru) 2013-09-27
RU2010104395A (ru) 2011-08-20
BRPI0815562A2 (pt) 2015-02-18
AU2008274170A1 (en) 2009-01-15
KR20120078754A (ko) 2012-07-10
NZ582443A (en) 2011-04-29

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