LV15257A - Jauni N-acil-arilsulfonamīda atvasinājumi kā aminoacil-tRNS sintetāzes inhibitori - Google Patents

Jauni N-acil-arilsulfonamīda atvasinājumi kā aminoacil-tRNS sintetāzes inhibitori

Info

Publication number
LV15257A
LV15257A LVP-16-06A LV160006A LV15257A LV 15257 A LV15257 A LV 15257A LV 160006 A LV160006 A LV 160006A LV 15257 A LV15257 A LV 15257A
Authority
LV
Latvia
Prior art keywords
acyl
novel
aminoacyl
arylsulfonamide
derivates
Prior art date
Application number
LVP-16-06A
Other languages
English (en)
Inventor
Aigars Jirgensons
Einārs LOŽA
Paul William Finn
Michael Charlton
Lluis Ribas De Pouplana
Adēlaide SAINT-LĒGER
Original Assignee
Latvijas Organiskās Sintēzes Institūts
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Latvijas Organiskās Sintēzes Institūts filed Critical Latvijas Organiskās Sintēzes Institūts
Priority to LVP-16-06A priority Critical patent/LV15257A/lv
Priority to PCT/LV2016/000001 priority patent/WO2016129983A1/en
Priority to AU2016216782A priority patent/AU2016216782C1/en
Priority to US15/550,839 priority patent/US11072581B2/en
Priority to JP2017561225A priority patent/JP6740256B2/ja
Priority to BR112017016977-0A priority patent/BR112017016977B1/pt
Priority to EP16704945.1A priority patent/EP3259250A1/en
Priority to EA201791530A priority patent/EA036995B1/ru
Priority to KR1020177024740A priority patent/KR102568859B1/ko
Priority to CN201680010072.1A priority patent/CN107257789B/zh
Priority to CA2975682A priority patent/CA2975682A1/en
Priority to MA041542A priority patent/MA41542A/fr
Priority to MX2017010357A priority patent/MX2017010357A/es
Priority to IL253886A priority patent/IL253886B/en
Priority to ZA2017/06108A priority patent/ZA201706108B/en
Publication of LV15257A publication Critical patent/LV15257A/lv

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Izgudrojums attiecas uz medicīnu, galvenokārt bakteriālo infekciju ārstēšanu.Izgudrojums ir jauni N-acil-diarilsulfonamīda atvasinājumi, kas darbojas kā bakteriālo aminoacil-t-RNS sintetāžu inhibitori. Tie ir izmantojami kā medicīniskie preparāti vai kā to sastāvdaļas bakteriālo infekciju ārstēšanai.
LVP-16-06A 2015-02-13 2016-02-10 Jauni N-acil-arilsulfonamīda atvasinājumi kā aminoacil-tRNS sintetāzes inhibitori LV15257A (lv)

Priority Applications (15)

Application Number Priority Date Filing Date Title
LVP-16-06A LV15257A (lv) 2016-02-10 2016-02-10 Jauni N-acil-arilsulfonamīda atvasinājumi kā aminoacil-tRNS sintetāzes inhibitori
PCT/LV2016/000001 WO2016129983A1 (en) 2015-02-13 2016-02-11 Novel n-acyl-arylsulfonamide derivatives as aminoacyl-trna synthetase inhibitors
AU2016216782A AU2016216782C1 (en) 2015-02-13 2016-02-11 Novel N-acyl-arylsulfonamide derivatives as aminoacyl-tRNA synthetase inhibitors
US15/550,839 US11072581B2 (en) 2015-02-13 2016-02-11 N-acyl-arylsulfonamide derivatives as aminoacyl-tRNA synthetase inhibitors
JP2017561225A JP6740256B2 (ja) 2015-02-13 2016-02-11 アミノアシルtRNAシンテターゼ阻害薬としての新規なN−アシル−アリールスルホンアミド誘導体
BR112017016977-0A BR112017016977B1 (pt) 2015-02-13 2016-02-11 Derivados de n-acil-arilsulfonamida como inibidores de aminoacil-trna sintetase
EP16704945.1A EP3259250A1 (en) 2015-02-13 2016-02-11 Novel n-acyl-arylsulfonamide derivatives as aminoacyl-trna synthetase inhibitors
EA201791530A EA036995B1 (ru) 2015-02-13 2016-02-11 НОВЫЕ N-АЦИЛАРИЛСУЛЬФОНАМИДНЫЕ ПРОИЗВОДНЫЕ В КАЧЕСТВЕ ИНГИБИТОРОВ АМИНОАЦИЛ-тРНК СИНТЕТАЗЫ
KR1020177024740A KR102568859B1 (ko) 2015-02-13 2016-02-11 아미노아실-tRNA 합성효소 저해제로서 신규한 N-아실-아릴술폰아미드 유도체
CN201680010072.1A CN107257789B (zh) 2015-02-13 2016-02-11 作为氨酰-trna合成酶抑制剂的新型n-酰基-芳基磺酰胺衍生物
CA2975682A CA2975682A1 (en) 2015-02-13 2016-02-11 N-acyl-arylsulfonamide derivatives as aminoacyl-trna synthetase inhibitors
MA041542A MA41542A (fr) 2015-02-13 2016-02-11 Nouveaux dérivés de n-acyl-arylsulfonamide utilisés en tant qu'inhibiteurs d'aminoacyl-arnt synthétase
MX2017010357A MX2017010357A (es) 2015-02-13 2016-02-11 Derivados novedosos de n-acil-arilsulfonamida como inhibidores de aminoacil acido ribonucleico de transferencia (arnt) sintetasa.
IL253886A IL253886B (en) 2015-02-13 2017-08-07 Novel n-acyl-arylsulfonamide compounds as aminoacyl-tRNA synthetase inhibitors
ZA2017/06108A ZA201706108B (en) 2015-02-13 2017-09-07 Novel n-acyl-arylsulfonamide derivatives as aminoacyl-trna synthetase inhibitors

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
LVP-16-06A LV15257A (lv) 2016-02-10 2016-02-10 Jauni N-acil-arilsulfonamīda atvasinājumi kā aminoacil-tRNS sintetāzes inhibitori

Publications (1)

Publication Number Publication Date
LV15257A true LV15257A (lv) 2017-09-20

Family

ID=61913767

Family Applications (1)

Application Number Title Priority Date Filing Date
LVP-16-06A LV15257A (lv) 2015-02-13 2016-02-10 Jauni N-acil-arilsulfonamīda atvasinājumi kā aminoacil-tRNS sintetāzes inhibitori

Country Status (1)

Country Link
LV (1) LV15257A (lv)

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