LV15257A - Jauni N-acil-arilsulfonamīda atvasinājumi kā aminoacil-tRNS sintetāzes inhibitori - Google Patents
Jauni N-acil-arilsulfonamīda atvasinājumi kā aminoacil-tRNS sintetāzes inhibitoriInfo
- Publication number
- LV15257A LV15257A LVP-16-06A LV160006A LV15257A LV 15257 A LV15257 A LV 15257A LV 160006 A LV160006 A LV 160006A LV 15257 A LV15257 A LV 15257A
- Authority
- LV
- Latvia
- Prior art keywords
- acyl
- novel
- aminoacyl
- arylsulfonamide
- derivates
- Prior art date
Links
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
Izgudrojums attiecas uz medicīnu, galvenokārt bakteriālo infekciju ārstēšanu.Izgudrojums ir jauni N-acil-diarilsulfonamīda atvasinājumi, kas darbojas kā bakteriālo aminoacil-t-RNS sintetāžu inhibitori. Tie ir izmantojami kā medicīniskie preparāti vai kā to sastāvdaļas bakteriālo infekciju ārstēšanai.
Priority Applications (15)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
LVP-16-06A LV15257A (lv) | 2016-02-10 | 2016-02-10 | Jauni N-acil-arilsulfonamīda atvasinājumi kā aminoacil-tRNS sintetāzes inhibitori |
AU2016216782A AU2016216782C1 (en) | 2015-02-13 | 2016-02-11 | Novel N-acyl-arylsulfonamide derivatives as aminoacyl-tRNA synthetase inhibitors |
US15/550,839 US11072581B2 (en) | 2015-02-13 | 2016-02-11 | N-acyl-arylsulfonamide derivatives as aminoacyl-tRNA synthetase inhibitors |
MX2017010357A MX2017010357A (es) | 2015-02-13 | 2016-02-11 | Derivados novedosos de n-acil-arilsulfonamida como inhibidores de aminoacil acido ribonucleico de transferencia (arnt) sintetasa. |
CA2975682A CA2975682A1 (en) | 2015-02-13 | 2016-02-11 | N-acyl-arylsulfonamide derivatives as aminoacyl-trna synthetase inhibitors |
JP2017561225A JP6740256B2 (ja) | 2015-02-13 | 2016-02-11 | アミノアシルtRNAシンテターゼ阻害薬としての新規なN−アシル−アリールスルホンアミド誘導体 |
PCT/LV2016/000001 WO2016129983A1 (en) | 2015-02-13 | 2016-02-11 | Novel n-acyl-arylsulfonamide derivatives as aminoacyl-trna synthetase inhibitors |
CN201680010072.1A CN107257789B (zh) | 2015-02-13 | 2016-02-11 | 作为氨酰-trna合成酶抑制剂的新型n-酰基-芳基磺酰胺衍生物 |
KR1020177024740A KR102568859B1 (ko) | 2015-02-13 | 2016-02-11 | 아미노아실-tRNA 합성효소 저해제로서 신규한 N-아실-아릴술폰아미드 유도체 |
BR112017016977-0A BR112017016977B1 (pt) | 2015-02-13 | 2016-02-11 | Derivados de n-acil-arilsulfonamida como inibidores de aminoacil-trna sintetase |
EP16704945.1A EP3259250A1 (en) | 2015-02-13 | 2016-02-11 | Novel n-acyl-arylsulfonamide derivatives as aminoacyl-trna synthetase inhibitors |
EA201791530A EA036995B1 (ru) | 2015-02-13 | 2016-02-11 | НОВЫЕ N-АЦИЛАРИЛСУЛЬФОНАМИДНЫЕ ПРОИЗВОДНЫЕ В КАЧЕСТВЕ ИНГИБИТОРОВ АМИНОАЦИЛ-тРНК СИНТЕТАЗЫ |
MA041542A MA41542A (fr) | 2015-02-13 | 2016-02-11 | Nouveaux dérivés de n-acyl-arylsulfonamide utilisés en tant qu'inhibiteurs d'aminoacyl-arnt synthétase |
IL253886A IL253886B (en) | 2015-02-13 | 2017-08-07 | Novel n-acyl-arylsulfonamide compounds as aminoacyl-tRNA synthetase inhibitors |
ZA2017/06108A ZA201706108B (en) | 2015-02-13 | 2017-09-07 | Novel n-acyl-arylsulfonamide derivatives as aminoacyl-trna synthetase inhibitors |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
LVP-16-06A LV15257A (lv) | 2016-02-10 | 2016-02-10 | Jauni N-acil-arilsulfonamīda atvasinājumi kā aminoacil-tRNS sintetāzes inhibitori |
Publications (1)
Publication Number | Publication Date |
---|---|
LV15257A true LV15257A (lv) | 2017-09-20 |
Family
ID=61913767
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
LVP-16-06A LV15257A (lv) | 2015-02-13 | 2016-02-10 | Jauni N-acil-arilsulfonamīda atvasinājumi kā aminoacil-tRNS sintetāzes inhibitori |
Country Status (1)
Country | Link |
---|---|
LV (1) | LV15257A (lv) |
-
2016
- 2016-02-10 LV LVP-16-06A patent/LV15257A/lv unknown
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