KR930007955A - Pyridone alkenyl cephalosporins and preparation method thereof - Google Patents
Pyridone alkenyl cephalosporins and preparation method thereof Download PDFInfo
- Publication number
- KR930007955A KR930007955A KR1019910018792A KR910018792A KR930007955A KR 930007955 A KR930007955 A KR 930007955A KR 1019910018792 A KR1019910018792 A KR 1019910018792A KR 910018792 A KR910018792 A KR 910018792A KR 930007955 A KR930007955 A KR 930007955A
- Authority
- KR
- South Korea
- Prior art keywords
- group
- hydrogen
- general formula
- compound
- pyridone
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D501/14—Compounds having a nitrogen atom directly attached in position 7
- C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
- C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
- C07D501/24—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D501/02—Preparation
- C07D501/04—Preparation from compounds already containing the ring or condensed ring systems, e.g. by dehydrogenation of the ring, by introduction, elimination or modification of substituents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Cephalosporin Compounds (AREA)
Abstract
본 발명은 다음 일반식(Ⅰ)로 표시되는 신규한피리돈계 알케닐세파롤스포린 및 그 제조방법에 관한 것이다.The present invention relates to a novel pyridone-based alkenyl cepharolsporin represented by the following general formula (I) and a method for producing the same.
식 중 R2은 수소, 트리틸, 3급 부톡시카르보닐, 포르밀이고, R2는 수소, 탄소수 1~4의 알킬, 알콕시카보닐메틸, 카르복시메틸, 1-카르복시에틸, 1-카르복시-1-메틸에틸, 탄소수 3~9의 시클로알킬기이고, R3는 수소, 알킬기, Na, K이고, R4및 R5는 수소 또는 대페닐메틸, 파라메톡시벤질임.Wherein R 2 is hydrogen, trityl, tert-butoxycarbonyl, formyl, R 2 is hydrogen, alkyl having 1 to 4 carbon atoms, alkoxycarbonylmethyl, carboxymethyl, 1-carboxyethyl, 1-carboxy- 1-methylethyl, a cycloalkyl group having 3 to 9 carbon atoms, R 3 is hydrogen, an alkyl group, Na, K, R 4 and R 5 are hydrogen or large phenylmethyl, paramethoxybenzyl.
본 발명의 일반식(Ⅰ)로 표시되는 피리돈계 알케닐세팔로스포린은 다음과 같은 반응공정에 따라 제조한다.The pyridone alkenyl cephalosporin represented by the general formula (I) of the present invention is prepared according to the following reaction process.
Description
본 내용은 요부공개 건이므로 전문내용을 수록하지 않았음Since this is an open matter, no full text was included.
Claims (3)
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
KR1019910018792A KR930007813B1 (en) | 1991-10-25 | 1991-10-25 | Process for preparing alkenyl cephalosporin |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
KR1019910018792A KR930007813B1 (en) | 1991-10-25 | 1991-10-25 | Process for preparing alkenyl cephalosporin |
Publications (2)
Publication Number | Publication Date |
---|---|
KR930007955A true KR930007955A (en) | 1993-05-20 |
KR930007813B1 KR930007813B1 (en) | 1993-08-20 |
Family
ID=19321734
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
KR1019910018792A KR930007813B1 (en) | 1991-10-25 | 1991-10-25 | Process for preparing alkenyl cephalosporin |
Country Status (1)
Country | Link |
---|---|
KR (1) | KR930007813B1 (en) |
-
1991
- 1991-10-25 KR KR1019910018792A patent/KR930007813B1/en not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
KR930007813B1 (en) | 1993-08-20 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
KR860003243A (en) | Process for preparing tazolidinedione derivatives | |
KR850001725A (en) | Method for preparing carboxylic ester | |
KR850004492A (en) | Method for preparing an enol ether derivative of oxycam | |
KR850004754A (en) | Method for producing 3-indole carboxamide compounds | |
KR930007955A (en) | Pyridone alkenyl cephalosporins and preparation method thereof | |
AU1866388A (en) | New process for the preparation of cephem compounds and new cephalosporin derivatives | |
KR870003107A (en) | Method for preparing chianthine derivative | |
KR930007954A (en) | Alkenyl cephalosporins and preparation methods thereof | |
EP0485204A3 (en) | Process for the preparation of 3-alkoxymethyl cephalosporin derivatives | |
KR840006667A (en) | Method for preparing cephalosporin derivative | |
ES2070101A1 (en) | Process for the preparation of cephem derivatives | |
KR850005441A (en) | Method for preparing 3-alkoxy-2- (N-pyrrolidino) -N-pyridyl-N-furylmethyl (or furylthienyl) -propylamine | |
KR940021558A (en) | Method for preparing a novel crystalline cephalosporin derivative | |
HUT47929A (en) | Process for producing 4-piperidine-carboxamide derivatives and pharmaceuticals comprising same | |
KR850006406A (en) | Method for preparing 4,7-dihydropyrazole [3,4-b] pyridine derivative | |
KR970061893A (en) | Alkali metal thioalkoxide of 2-hydroxycarbamoyl-7-mercapto-s-triazolo [1,5-a] pyrimidine derivative and method for producing the same | |
KR930000532A (en) | Production method of sugar epitopes | |
KR930023366A (en) | β-carboline derivatives | |
KR920002564A (en) | N-alkyl thiazolidine derivatives | |
KR910000773A (en) | 3-phenylthiosialic acid derivative, sialic acid containing oligosaccharide derivative, and its manufacturing method | |
AU590455B2 (en) | Process for preparing penems | |
KR890002176A (en) | New Cefem Compounds | |
KR880003957A (en) | Method for preparing cephalosporin derivative | |
KR830007509A (en) | Method for preparing amino acid derivative | |
KR940019713A (en) | Method for preparing a novel cephalosporin derivative |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
A201 | Request for examination | ||
G160 | Decision to publish patent application | ||
E701 | Decision to grant or registration of patent right | ||
GRNT | Written decision to grant | ||
FPAY | Annual fee payment |
Payment date: 19970829 Year of fee payment: 6 |
|
LAPS | Lapse due to unpaid annual fee |