KR890009877A - 1-아실-2-피라졸린유도체의 제조방법 - Google Patents

1-아실-2-피라졸린유도체의 제조방법 Download PDF

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Publication number
KR890009877A
KR890009877A KR1019880016870A KR880016870A KR890009877A KR 890009877 A KR890009877 A KR 890009877A KR 1019880016870 A KR1019880016870 A KR 1019880016870A KR 880016870 A KR880016870 A KR 880016870A KR 890009877 A KR890009877 A KR 890009877A
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South Korea
Prior art keywords
group
acyl
preparing
pyrazoline derivative
formula
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KR1019880016870A
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English (en)
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KR900007197B1 (ko
Inventor
히로유키 야마시타
쿠니오 오쿠무라
하지메 이즈카
노리오 오토
Original Assignee
사와무라 하루오
미쓰이 도오아쯔 카가쿠 가부시기가이샤
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Publication of KR890009877A publication Critical patent/KR890009877A/ko
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Publication of KR900007197B1 publication Critical patent/KR900007197B1/ko

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/06Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/06Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

내용 없음

Description

1 -아실-2-피라졸린유도체의 제조방법
본 내용은 요부공개 건이므로 전문내용을 수록하지 않았음

Claims (1)

  1. 하기 일반식(I)의 아실히드라존 유도체를 가열환화하는 것을 특징으로 하는 하기 일반식(II)의 1-아실-2-피라졸린유도체의 제조방법:
    상기식에서. R1은 수소원자, 피리딜기, 피라지닐기, 알킬기, 아릴기, 또는 알콕시기를 나타내며, R2, R3및 R4는 각각 수소원자, 푸릴기, 피리딜기, 알킬기 또는 아릴기를 나타낸다.
    ※ 참고사항 : 최초출원 내용에 의하여 공개하는 것임.
KR1019880016870A 1987-12-17 1988-12-17 1-아실-2-피라졸린유도체의 제조방법 KR900007197B1 (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP62-317446 1987-12-17
JP31744687 1987-12-17

Publications (2)

Publication Number Publication Date
KR890009877A true KR890009877A (ko) 1989-08-04
KR900007197B1 KR900007197B1 (ko) 1990-10-05

Family

ID=18088310

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019880016870A KR900007197B1 (ko) 1987-12-17 1988-12-17 1-아실-2-피라졸린유도체의 제조방법

Country Status (7)

Country Link
US (1) US4895947A (ko)
EP (1) EP0322691B1 (ko)
KR (1) KR900007197B1 (ko)
CN (1) CN1015177B (ko)
CA (1) CA1319366C (ko)
DE (1) DE3850236T2 (ko)
HU (1) HU201752B (ko)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5089622A (en) * 1988-12-12 1992-02-18 Mitsui Toatsu Chemicals Incorporated (-)-2-pyrazoline compounds and therapeutic agent for cerebrovascular disorders containing the same as effective ingredient
JP4614948B2 (ja) * 2004-03-09 2011-01-19 独立行政法人科学技術振興機構 含窒素5員環化合物の製造方法
TWI730959B (zh) 2015-05-19 2021-06-21 英商葛蘭素史克智慧財產發展有限公司 作為激酶抑制劑之雜環醯胺

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3666772A (en) * 1970-02-26 1972-05-30 Carlisle Chemical Works Preparation of pyrazolines by cyclization of an azine
US3952010A (en) * 1973-09-17 1976-04-20 American Cyanamid Company Catalytic dehydrogenation process for the preparation of 3,5-disubstituted pyrazoles
US4250185A (en) * 1980-03-10 1981-02-10 Stauffer Chemical Company 1-(3,5-Dichlorobenzoyl)-3-phenylpyrazolines and their use as mildewicides
JPH0730031B2 (ja) * 1986-04-02 1995-04-05 日産化学工業株式会社 2―ピラゾリン―5―オン類の製造法
HU202106B (en) * 1987-06-17 1991-02-28 Mitsui Toatsu Chemicals Process for producing pharmaceutical compositions containing pyrazolin derivatives

Also Published As

Publication number Publication date
DE3850236T2 (de) 1994-09-22
HUT49602A (en) 1989-10-30
CN1015177B (zh) 1991-12-25
US4895947A (en) 1990-01-23
EP0322691A1 (en) 1989-07-05
EP0322691B1 (en) 1994-06-15
HU201752B (en) 1990-12-28
CA1319366C (en) 1993-06-22
KR900007197B1 (ko) 1990-10-05
DE3850236D1 (de) 1994-07-21
CN1033994A (zh) 1989-07-19

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