KR890003375A - 암로디핀의 베실레이트 염 - Google Patents
암로디핀의 베실레이트 염 Download PDFInfo
- Publication number
- KR890003375A KR890003375A KR1019870008580A KR870008580A KR890003375A KR 890003375 A KR890003375 A KR 890003375A KR 1019870008580 A KR1019870008580 A KR 1019870008580A KR 870008580 A KR870008580 A KR 870008580A KR 890003375 A KR890003375 A KR 890003375A
- Authority
- KR
- South Korea
- Prior art keywords
- amlodipine
- besylate salt
- excipient
- tablet
- aqueous solution
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/4841—Filling excipients; Inactive ingredients
- A61K9/4858—Organic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K2121/00—Preparations for use in therapy
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- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Cardiology (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Heart & Thoracic Surgery (AREA)
- Biophysics (AREA)
- Molecular Biology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
Abstract
Description
Claims (12)
- 암로디핀의 베실레이트 염
- 제 1 항에 따른 암로디핀의 베실레이트 염을 약제학적으로 허용되는 희석제 또는 담체와 함께 함유하는 약제학적 조성물.
- 제 1 항에 따른 암로디핀의 베실레이트 염이 부형제와 혼합되어 함유된 정제.
- 제 3 항에 있어서, 부형제가 압착보조제, 정제에 광택을 부여하는 첨가제, 붕해제 및 활탁제를 함유하는 정제.
- 제 4 항에 있어서, 부형제가 미세결정성 셀룰로즈, 무수이염기성 인산칼슘, 나트륨 전분글리콜레이트 및 마그네슘 스테아레이트를 함유하는 정제.
- 제 1 항에 따른 암로디핀의 베실레이트 염이 부형제와 혼합되어 함유된 칼셀제.
- 제 6 항에 있어서, 부형제가 불활성 희석제, 건조된 붕해제 및 활탁제를 함유하는 캅셀제.
- 제 6 항에 있어서, 부형제가 미세결정성 셀룰로즈, 건조된 옥수수 전분 및 마그네슘 스테아레이트를 함유하는 캅셀제.
- 암로디핀의 베실레이트 염을 함유하는 비경구 투여용 멸균 수용액.
- 제 9 항에 있어서, 10 내지 40% W/V 의 프로필렌 글리콜을 함유하는 멸균 수용액.
- 제 9 항 또는 10 항에 있어서, 약 1% W/V 의 염화나트륨을 함유하는 멸균 수용액.
- 심장 질환 또는 고혈압 치료에 유용한 암로디핀의 베실레이트 염.※ 참고사항 : 최초출원 내용에 의하여 공개하는 것임.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| KR1019870008580A KR950007228B1 (ko) | 1987-08-05 | 1987-08-05 | 암로디핀의 베실레이트염 |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| KR1019870008580A KR950007228B1 (ko) | 1987-08-05 | 1987-08-05 | 암로디핀의 베실레이트염 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| KR890003375A true KR890003375A (ko) | 1989-04-14 |
| KR950007228B1 KR950007228B1 (ko) | 1995-07-07 |
Family
ID=19263584
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR1019870008580A KR950007228B1 (ko) | 1987-08-05 | 1987-08-05 | 암로디핀의 베실레이트염 |
Country Status (1)
| Country | Link |
|---|---|
| KR (1) | KR950007228B1 (ko) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR100558505B1 (ko) | 2003-01-27 | 2006-03-07 | 한미약품 주식회사 | 안정한 무정형 암로디핀 캠실레이트, 이의 제조방법 및이를 포함하는 경구투여용 조성물 |
| KR100841409B1 (ko) | 2003-12-16 | 2008-06-25 | 에스케이케미칼주식회사 | 암로디핀 겐티세이트 염과 이의 제조방법 |
-
1987
- 1987-08-05 KR KR1019870008580A patent/KR950007228B1/ko not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| KR950007228B1 (ko) | 1995-07-07 |
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