KR880003923A - 2-시아노-2-알콕시미노-아세트 아미드 - Google Patents

2-시아노-2-알콕시미노-아세트 아미드 Download PDF

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KR880003923A
KR880003923A KR870009957A KR870009957A KR880003923A KR 880003923 A KR880003923 A KR 880003923A KR 870009957 A KR870009957 A KR 870009957A KR 870009957 A KR870009957 A KR 870009957A KR 880003923 A KR880003923 A KR 880003923A
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carbon atoms
optionally substituted
straight
cyano
branched
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KR870009957A
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게이어 헤르베르크
젤리히 클라우스
룬켄하이머 빌프리트
브란데스 빌헬름
핸슬러 게르트
Original Assignee
권터 슈마허, 칼-루드비히 슈미트
바이엘 아크티엔게젤샤프트
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Publication of KR880003923A publication Critical patent/KR880003923A/ko

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    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
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    • C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
    • C07D207/32—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C07D207/33—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms with substituted hydrocarbon radicals, directly attached to ring carbon atoms
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    • C07D261/06—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
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    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
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    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
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    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
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    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
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    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

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Abstract

내용 없음

Description

2-시아노-2-알콕시미노-아세트 아미드
본 내용은 요부공개 건이므로 전문내용을 수록하지 않았음

Claims (10)

  1. 일반식(Ⅰ)의 2-시아노-2-알콕시미노-아세트아미드
    상기식에서, R1은 임의로 치환된 하이드록시알킬, 임의로 치환된 하이드록시알콕시알킬, 임의로 치환된 헤테로 아릴알킬 또는 임의로 치환된 헤테로 아릴을 나타내고, R2는 임의로 치환된 알킬, 임의로 치환된 알케닐, 또는 알키닐을 나타낸다.
  2. 제1항에 있어서, R1이 각각의 알킬 부분의 탄소원자수가 1 내지 6인, 직쇄 또는 측쇄의 임의로 페닐-치환된 하이드록시알킬 또는 하이드록시 알콕시알킬을 나타내거나, 각각의 경우 헤테로 아릴 부분의 탄소원자수가 2 내지 10이고 헤테로 원자수가 1내지 3이며, 헤테로 아릴알킬의 경우 직쇄 또는 측쇄 알킬 부분의 탄소원자수가 1내지 6인 임의로 일치환되거나 다치환되고/되거나 벤젠-융합된 헤테로 아릴알킬 또는 헤테로 아릴을 나타내며, 여기에서 치환체는 동일하거나 상이하며, 헤테로아릴 부분 및/또는 벤젠-융합된 환의 적합한 치환체는 각기 하이드록실, 할로겐, 시아노, 가기 탄소원자수가 4이하인, 직쇄 또는 측쇄의 알킬, 알케닐, 알콕시 또는 알킬티오, 아릴 부위의 탄소원자수가 6내지 10이고 직쇄 또는 측쇄 알킬 부분의 탄소원자수가 1내지 3인 아르알킬 탄소원자수가 6내지 10인 아릴, 또는 각각의 경우 직쇄 또는 측쇄알킬 부분의 탄소원자수가 1내지 4인, 알킬카보닐, 알콕시카보닐, 알킬아미노 카보닐 및 디알킬아미노 카보닐이고, R2가 임의로 일치환되거나 다치환된 탄소원자수 1내지 18의 직쇄 또는 측쇄 알킬을 나타내고, 여기에서 치환체는 동일하거나 상이하며 언급될 수 있는 치환체가 시아노, 각각의 알킬 부분의 탄소원자수가 1내지 6인, 직쇄 측쇄 알카노일, 알콕시카보닐 또는 알킬카보닐옥시이고, 탄소원자수가 2내지 9이고 헤테로원자수가 1내지 3이며, 각기 임의로 저급알킬 및/또는 할로겐에 의해 일치환되거나 다치환된 페닐 또는 헤테로 아릴을 나타내거나, 또한, 탄소원자수가 3내지 8이며, 할로게노 알케닐인 경우 할로겐 원자수가 1내지 5인 직쇄 또는 측쇄 알케닐 또는 할로게노알케닐, 또는 탄소원자수가 3내지 8인 직쇄 또는 측쇄 알키닐을 나타내는 일반식(Ⅰ)의 2-시아노-2-알콕시미노-아세트아미드.
  3. 제1항에 있어서, R1이 각각의 알킬 부분의 탄소원자수가 1내지 4인, 직쇄 또는 측쇄의 임의로 페닐-치환된 하이드록시 알킬 또는 하이드록시 알콕시알킬을 나타내거나, 각각의 경우 헤테로 아릴 부분의 탄소원자수가 2내지 10이고 질소 및/또는 산소 및/또는 황 원자수가 1내지 3이며, 직쇄 또는 측쇄 알킬부분의 탄소원자수가 1내지 4이고 각각의 경우 임으로 일치환, 이치환 또는 삼치환 되고/되거나 벤젠-융합된 헤테로 아릴알킬 또는 헤테로 아릴을 나타내며, 여기에서 치환체는 동일하거나 상이하며, 헤테로아릴 부분 및/또는 벤젠-융합된 환의 적합한 치환체는 하이드록실, 불소, 염소, 브롬, 시아노, 메틸, 에틸, n-또는 i-프로필, n-, i-, s-또는 t-부틸,알릴, 부테닐, 메톡시, 에톡시, 메틸티오, 벤질, 페닐, 아세틸, 프로피오닐, 메톡시카보닐, 에톡시카보닐, 메틸아미노카보닐 또는 디메틸아미노 카보닐이고, R2가 탄소원자수가 1내지 12이며, 임의로 일치환, 이치환 또는 삼치환된 직쇄 또는 측쇄 알킬을 나타내고, 여기에서 치환체는 동일하거나 상이하며, 언급될 수 있는 치환체는 시아노, 아세틸, 프로피오닐, 메톡시카보닐, 에톡시카보닐, 메틸카보닐옥시, 에틸카보닐옥시, 또는 불소, 염소, 브롬, 메틸 및/또는 에틸에 의해 임의로 일치환, 이치환 또는 삼치환된 페닐 또는 헤테로아릴이고, 여기에서 치환체는 동일하거나 상이하며, 헤테로 아릴에 적합한 것으로 피리딜, 피리미딜, 트리아지닐, 퀴놀일, 이소퀴놀일, 옥시졸일, 이속 사졸일, 옥사 디아졸일, 벤족사졸알, 타아졸일, 이소티아졸일, 타아디아졸일, 벤즈타아졸일, 이미다졸일, 벤즈 이미다졸일, 비롤일, 푸라닐, 테에닐, 피라졸일 또는 트리아졸일을 나타내거나, 또한 탄소원자수가 3내지 6이고, 경우데 따라 할로겐 원자수가 1내지 3인 각기 직쇄 또는 측쇄 알케닐 또는 할로게노알케닐, 또는 탄소원자수가 3내지 6인 직쇄 또는 측쇄 알케닐을 나타내는 일반식(Ⅰ)의 2-시아노-2-알콕시미노-아세트아미드.
  4. 제1항에 있어서, R1이 각각의 알킬 부분의 탄소원자수가 1내지 4인, 각각 직쇄 또는 측쇄의, 임의로 페닐-치환된 하이드록시알킬 또는 하이드록시알콕시알킬을 나타내거나, 또는 직쇄 또는 측쇄 알킬 부분의 탄소원자수가 1내지 4이고, 각기 임의로 일치환, 이치환 또는 삼치환된 헤테로 아릴 또는 헤테로 아릴알킬을 나타내며, 여기에서 치환체는 동일하거나 상이하며, 헤테로 아릴 라디칼로서 각기 가능한 것은 피리딜, 피리미딜, 트리아지닐, 퀴놀일, 이소퀴놀일, 옥사졸일, 이속사졸일, 옥사디아졸일, 벤즈옥사졸일, 티아졸일, 이소티아졸일, 티아디아졸일, 벤즈티아졸일, 이미다졸일, 벤즈이디마졸일, 피롤일, 푸라닐, 티에닐, 피라졸일 또는 트라이졸일이고, 헤테로 아릴 부분 또는 벤젠-융합된 환의 치환체로서 각기 적합한 것은 하이드록실, 불소, 염소, 브롬, 시아노, 메틸, 에틸, n-또는 i-프로필, n-, i-, s-또는 t-부틸, 아릴, 부테닐, 메톡시, 에톡시, 메틸티오, 벤질, 페닐, 아세틸, 프로피오닐, 메톡시카보닐, 에톡시카보닐, 메틸아미노카보닐 또는 디메틸아미노카보닐이며 R2가 임의로 일치환, 이치환 또는 삼치환된 탄소원자수 1내지 12의 직쇄 또는 측쇄 알킬을 나타내고, 여기에서 치환체가 동일하거나 상이하고, 언급될 수 있는 치환체는 시아노, 아세틸, 프로피오닐, 메톡시카보닐, 에톡시카보닐, 메틸카보닐옥시, 에틸카보닐옥시 또는 불소, 염소, 브롬, 메틸 및/또는 에틸에 의해 임의로 일치환, 이치환 또는 삼치환된 페닐(여기에서 치환체는 동일하거나 상이하다)이거나, 또한 탄소 원자수가 3내지 6이고, 경우에 따라 할로겐 원자수가 1내지 3인 가기; 직쇄 또는 측쇄 알케닐 또는 할로게노 알케닐, 또는 탄소원자수가 3내지 6인, 직쇄 또는 측쇄 알키닐을 나타내는 일반식(Ⅰ)의 2-시아노-2-알콕시미노-아세트아미드.
  5. 일반식(Ⅱ)의 2-시아노-2-옥시미노-아세트 아미드를 경우에 따라 희석제의 존재하, 및 경우에 따라 산-결합제의 존재하에서 일반식(Ⅲ)의 알킬화제와 반응시킴을 특징으로 하여, 일반식(Ⅰ)의 2-시아노-2-알콕시미노-아세트아미드를 제조하는 방법.
    상기식에서, R1은 임의로 치환된 하이드록시알킬, 임의로 치환된 하이드록시알콕시알킬, 임의로 치환된 헤테로 아릴알킬 또는 임의로 치환된 헤테로아릴을 나타내고, R2는 임의로 치환된 알킬, 임의로 치환된 알케닐, 또는 알키닐을 나타내며, M은 수소 또는 알카리 금속 양이온을 나타내고, A는 적합한 이탈 그룹을 나타낸다.
  6. 제1항에 따른 하나 이상의 일반식(Ⅰ)의 화합물을 함유함을 특징으로 하는 살충제.
  7. 제1항에 따른 하나 이상의 일반식(Ⅰ)의 화합물을 해충 및/또는 그의 서식지에 적용시킴을 특징으로 하여, 해충을 퇴치하는 방법.
  8. 해충을 퇴치하기 위한, 제1항에 따른 일반식(Ⅰ)의 화합물의 용도.
  9. 제1항에 따른 일반식(Ⅰ) 화합물을 증량제 및/또는 계면활성제와 혼합시킴을 특징으로 하여, 살충제를 제조하는 방법.
  10. 일반식(Ⅱ)의 2-시아노-2-옥시미노-아세트아미드.
    상기식에서, M은 수소 또는 알카리 금속 양이온을 나타내고 R1은 임의로 치환된 하이드록시알킬, 임의로 치환된 하이드록시알콕시알킬, 임의로 치환된 헤테로 아릴알킬 또는 임의로 치환된 헤테로 아릴을 나타낸다.
    ※ 참고사항 : 최초출원 내용에 의하여 공개하는 것임.
KR870009957A 1986-09-10 1987-09-09 2-시아노-2-알콕시미노-아세트 아미드 KR880003923A (ko)

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ZA731111B (en) * 1972-03-15 1974-03-27 Du Pont 2-cyano-2-hydroxyiminoacetamides and acetates as plant disease control agents
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US3957847A (en) * 1974-03-21 1976-05-18 E. I. Du Pont De Nemours And Company 2-cyano-2-hydroxyiminoacetamides as plant disease control agents
DE3138502A1 (de) * 1981-09-28 1983-04-07 Basf Ag, 6700 Ludwigshafen N-substituierte carbonsaeureamide, verfahren zu ihrer herstellung und diese enthaltende fungizide
DE3208329A1 (de) * 1982-03-09 1983-09-15 Basf Ag, 6700 Ludwigshafen Oximinoessigsaeureamide, ihre herstellung und ihre verwendung zur bekaempfung von fungi und mittel dafuer
GB2173791B (en) * 1985-04-16 1989-07-05 Ici Plc Fungicidal cyano oximes
DE3602243A1 (de) * 1985-06-13 1986-12-18 Bayer Ag, 5090 Leverkusen E-isomere von n(pfeil hoch)(alpha)(pfeil hoch)-(2-cyan-2-alkoximino-acetyl)-aminosaeurederivaten und -peptiden
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