KR850001919B1 - 20'-하이드록시 빈블라스틴 및 유사화합물의 제조방법 - Google Patents

20'-하이드록시 빈블라스틴 및 유사화합물의 제조방법 Download PDF

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Publication number
KR850001919B1
KR850001919B1 KR1019810005164A KR810005164A KR850001919B1 KR 850001919 B1 KR850001919 B1 KR 850001919B1 KR 1019810005164 A KR1019810005164 A KR 1019810005164A KR 810005164 A KR810005164 A KR 810005164A KR 850001919 B1 KR850001919 B1 KR 850001919B1
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KR
South Korea
Prior art keywords
iia
indole
isomer
general formula
desacetyl
Prior art date
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Expired
Application number
KR1019810005164A
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English (en)
Korean (ko)
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KR830007703A (ko
Inventor
코린 밀러 진
리 톰슨 제랄드
Original Assignee
일라이 릴리 앤드 캄파니
아더 알. 웨일
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Application filed by 일라이 릴리 앤드 캄파니, 아더 알. 웨일 filed Critical 일라이 릴리 앤드 캄파니
Publication of KR830007703A publication Critical patent/KR830007703A/ko
Application granted granted Critical
Publication of KR850001919B1 publication Critical patent/KR850001919B1/ko
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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
    • C07D519/04—Dimeric indole alkaloids, e.g. vincaleucoblastine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
KR1019810005164A 1980-12-29 1981-12-28 20'-하이드록시 빈블라스틴 및 유사화합물의 제조방법 Expired KR850001919B1 (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US220471 1980-12-29
US06/220,471 US4320058A (en) 1980-12-29 1980-12-29 20'-Hydroxyvinblastine and related compounds

Publications (2)

Publication Number Publication Date
KR830007703A KR830007703A (ko) 1983-11-04
KR850001919B1 true KR850001919B1 (ko) 1985-12-31

Family

ID=22823662

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019810005164A Expired KR850001919B1 (ko) 1980-12-29 1981-12-28 20'-하이드록시 빈블라스틴 및 유사화합물의 제조방법

Country Status (10)

Country Link
US (1) US4320058A (enExample)
EP (1) EP0055603A1 (enExample)
JP (1) JPS57134491A (enExample)
KR (1) KR850001919B1 (enExample)
CA (1) CA1168231A (enExample)
GB (1) GB2090255B (enExample)
GR (1) GR75400B (enExample)
HU (1) HU185080B (enExample)
IE (1) IE52307B1 (enExample)
IL (1) IL64618A (enExample)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2707988B1 (fr) * 1993-07-21 1995-10-13 Pf Medicament Nouveaux dérivés antimitotiques des alcaloïdes binaires du catharantus rosesus, leur procédé de préparation et les compositions pharmaceutiques les comprenant.
BRPI0809249B1 (pt) 2007-03-21 2019-12-17 Commw Scient Ind Res Org método para planejamento e execução de trajetos livres de obstáculo para a maquinaria de escavação rotatória

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2296418B1 (enExample) 1974-12-30 1978-07-21 Anvar
US4029663A (en) * 1975-07-10 1977-06-14 Eli Lilly And Company Dimeric anhydro-vinca derivatives
US4110330A (en) * 1977-05-27 1978-08-29 Eli Lilly And Company 5'-Acetonylvincristine and related compounds

Also Published As

Publication number Publication date
IE52307B1 (en) 1987-09-02
GB2090255A (en) 1982-07-07
IL64618A (en) 1985-11-29
JPS57134491A (en) 1982-08-19
GB2090255B (en) 1984-11-28
EP0055603A1 (en) 1982-07-07
KR830007703A (ko) 1983-11-04
CA1168231A (en) 1984-05-29
GR75400B (enExample) 1984-07-13
HU185080B (en) 1984-11-28
IL64618A0 (en) 1982-03-31
IE813055L (en) 1982-06-29
US4320058A (en) 1982-03-16

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