KR850001340B1 - 페니실란산 술폰의 에스테르 제조 방법 - Google Patents

페니실란산 술폰의 에스테르 제조 방법 Download PDF

Info

Publication number
KR850001340B1
KR850001340B1 KR1019810004830A KR810004830A KR850001340B1 KR 850001340 B1 KR850001340 B1 KR 850001340B1 KR 1019810004830 A KR1019810004830 A KR 1019810004830A KR 810004830 A KR810004830 A KR 810004830A KR 850001340 B1 KR850001340 B1 KR 850001340B1
Authority
KR
South Korea
Prior art keywords
sulfone
reaction
group
halogenating agent
chlorine
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
KR1019810004830A
Other languages
English (en)
Korean (ko)
Other versions
KR830007672A (ko
Inventor
러너드 헤이지맨 데이비드
챨스 크로포오드 토마스
Original Assignee
화이자 인코포레이티드
윌리암 데이비스 헌
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 화이자 인코포레이티드, 윌리암 데이비스 헌 filed Critical 화이자 인코포레이티드
Publication of KR830007672A publication Critical patent/KR830007672A/ko
Application granted granted Critical
Publication of KR850001340B1 publication Critical patent/KR850001340B1/ko
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/04—Preparation
    • C07D499/08—Modification of a carboxyl radical directly attached in position 2, e.g. esterification
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
KR1019810004830A 1980-12-11 1981-12-10 페니실란산 술폰의 에스테르 제조 방법 Expired KR850001340B1 (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US215215 1980-12-11
US215,215 1980-12-11
US06/215,215 US4361513A (en) 1980-12-11 1980-12-11 Esters of penicillanic acid sulfone

Publications (2)

Publication Number Publication Date
KR830007672A KR830007672A (ko) 1983-11-04
KR850001340B1 true KR850001340B1 (ko) 1985-09-19

Family

ID=22802118

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019810004830A Expired KR850001340B1 (ko) 1980-12-11 1981-12-10 페니실란산 술폰의 에스테르 제조 방법

Country Status (20)

Country Link
US (1) US4361513A (enExample)
EP (1) EP0054397B1 (enExample)
JP (1) JPS57122089A (enExample)
KR (1) KR850001340B1 (enExample)
AR (1) AR229599A1 (enExample)
AT (1) ATE12233T1 (enExample)
AU (1) AU527159B2 (enExample)
CA (1) CA1177068A (enExample)
DE (1) DE3169462D1 (enExample)
DK (1) DK158228C (enExample)
ES (1) ES8302717A1 (enExample)
FI (1) FI75824C (enExample)
GR (1) GR76963B (enExample)
IE (1) IE52111B1 (enExample)
IL (1) IL64497A0 (enExample)
NO (1) NO160517C (enExample)
PH (1) PH17469A (enExample)
PT (1) PT74111B (enExample)
YU (1) YU43053B (enExample)
ZA (1) ZA818579B (enExample)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4746754A (en) * 1986-05-16 1988-05-24 The Dow Chemical Company Preparation of carbonate diisocyanates and related compounds
US7968279B2 (en) * 2008-08-13 2011-06-28 Beckman Coulter, Inc. Reference control for cell by cell analysis
WO2014140576A1 (en) 2013-03-13 2014-09-18 Andrew Bacon Improvements in the fuel efficiency of road vehicles

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS512477A (en) * 1974-06-25 1976-01-10 Zekoo Kk Ijokeisha shindonokanchisochi
JPS512476A (ja) * 1974-06-25 1976-01-10 Inoue Japax Res Hokokei
JPS6056160B2 (ja) * 1977-06-07 1985-12-09 フアイザ−・インコ−ポレ−テツド β−ラクタマ−ゼ阻害剤としてのペニシラン酸１，１−ジオキシド
US4272439A (en) * 1978-06-02 1981-06-09 Schering Corporation 6-(Substituted-hydroxymethylene penams)
US4241050A (en) * 1978-09-01 1980-12-23 Pfizer Inc. Penam 1,1-dioxides as beta-lactamase inhibitors
US4331677A (en) * 1978-11-24 1982-05-25 Farmitalia Carlo Erba S.P.A. 7-Oxo-4-1-aza-bicyclo-[3,2,0]-heptane derivatives
US4256733A (en) * 1979-09-26 1981-03-17 Pfizer Inc. Acetoxymethyl penam compounds as β-lactamase inhibitors

Also Published As

Publication number Publication date
EP0054397B1 (en) 1985-03-20
ES507867A0 (es) 1983-01-16
AR229599A1 (es) 1983-09-30
PT74111B (en) 1983-12-19
KR830007672A (ko) 1983-11-04
ES8302717A1 (es) 1983-01-16
IE52111B1 (en) 1987-06-24
FI75824C (fi) 1988-08-08
EP0054397A1 (en) 1982-06-23
CA1177068A (en) 1984-10-30
PT74111A (en) 1982-01-01
IL64497A0 (en) 1982-03-31
AU527159B2 (en) 1983-02-17
NO160517B (no) 1989-01-16
ATE12233T1 (de) 1985-04-15
DK158228B (da) 1990-04-16
NO814226L (no) 1982-06-14
ZA818579B (en) 1982-11-24
FI813956L (fi) 1982-06-12
PH17469A (en) 1984-08-29
DK158228C (da) 1990-09-24
GR76963B (enExample) 1984-09-04
YU43053B (en) 1989-02-28
JPS57122089A (en) 1982-07-29
YU288181A (en) 1983-12-31
AU7844681A (en) 1982-06-17
JPS6251959B2 (enExample) 1987-11-02
DK547181A (da) 1982-06-12
NO160517C (no) 1989-04-26
DE3169462D1 (en) 1985-04-25
IE812899L (en) 1982-06-11
FI75824B (fi) 1988-04-29
US4361513A (en) 1982-11-30

Similar Documents

Publication Publication Date Title
KR850001340B1 (ko) 페니실란산 술폰의 에스테르 제조 방법
KR910000238B1 (ko) 티아졸 유도체의 제조방법
CH628900A5 (fr) Procede de preparation de thio-oximes derivees de cephalosporines et de penicillines.
US4020077A (en) Antibiotics
US4075203A (en) Process for preparing a 3-exomethylenecepham sulfoxide from penicillin sulfoxides
US4888429A (en) Process for producing allyl aminothiazole acetate intermediates
US3975385A (en) 7-Trichloroacetamido-3-desacetoxy-cephalosporanic acid esters
US4185053A (en) Process for manufacturing substantially pure dialkyl phosphorochloridothionate
US4474698A (en) Process for preparing esters of penicillanic acid sulfone
HU189125B (en) Process for preparing new penicillanic acid derivatives
US3974150A (en) 7β-Isocyano cephalosporin esters and process of preparation
US3595880A (en) Preparation of (cis-1,2-epoxypropyl) phosphonic acids
JPH0523271B2 (enExample)
EP0397212A1 (en) Process for preparing cephalosporin compounds
SU845790A3 (ru) Способ получени -метокси- -ХлОРМЕТилцЕфЕМОВ
EP0217376B1 (en) Process for preparing optically active alpha-haloalkyl-arylketones
SE444810B (sv) Sulfinyazetidinonforeningar till anvendning for framstellning av 3-metylencefamsulfoxider
EP0122002B1 (en) Process for preparing azetidinone derivatives
KR840000118B1 (ko) 옥사졸리노 아제티디논의 제조방법
KR100477763B1 (ko) 세파트리진 프로필렌글리콜 중간체의 신규한 제조방법
EP0109817A2 (en) Process for preparing oxazolinoazetidinones
CA1221371A (en) Intermediates and process for preparing (s)-3- acylamino-4-substituted-2-azetidinones
KR910001309B1 (ko) 페니실란산 화합물의 제조 방법
KR810000738B1 (ko) 5-알콕시-피콜린산에스테르의 제조법
SU794012A1 (ru) Способ получени бета-1,1- диОКСОТиОлАНТиОлОВ

Legal Events

Date Code Title Description
PA0109 Patent application

St.27 status event code: A-0-1-A10-A12-nap-PA0109

R17-X000 Change to representative recorded

St.27 status event code: A-3-3-R10-R17-oth-X000

PA0201 Request for examination

St.27 status event code: A-1-2-D10-D11-exm-PA0201

PG1501 Laying open of application

St.27 status event code: A-1-1-Q10-Q12-nap-PG1501

PG1605 Publication of application before grant of patent

St.27 status event code: A-2-2-Q10-Q13-nap-PG1605

PE0701 Decision of registration

St.27 status event code: A-1-2-D10-D22-exm-PE0701

PR0701 Registration of establishment

St.27 status event code: A-2-4-F10-F11-exm-PR0701

PR1002 Payment of registration fee

St.27 status event code: A-2-2-U10-U11-oth-PR1002

Fee payment year number: 1

PR1001 Payment of annual fee

St.27 status event code: A-4-4-U10-U11-oth-PR1001

Fee payment year number: 4

PR1001 Payment of annual fee

St.27 status event code: A-4-4-U10-U11-oth-PR1001

Fee payment year number: 5

PR1001 Payment of annual fee

St.27 status event code: A-4-4-U10-U11-oth-PR1001

Fee payment year number: 6

PR1001 Payment of annual fee

St.27 status event code: A-4-4-U10-U11-oth-PR1001

Fee payment year number: 7

PR1001 Payment of annual fee

St.27 status event code: A-4-4-U10-U11-oth-PR1001

Fee payment year number: 8

PR1001 Payment of annual fee

St.27 status event code: A-4-4-U10-U11-oth-PR1001

Fee payment year number: 9

PC1903 Unpaid annual fee

St.27 status event code: A-4-4-U10-U13-oth-PC1903

Not in force date: 19940920

Payment event data comment text: Termination Category : DEFAULT_OF_REGISTRATION_FEE

PC1903 Unpaid annual fee

St.27 status event code: N-4-6-H10-H13-oth-PC1903

Ip right cessation event data comment text: Termination Category : DEFAULT_OF_REGISTRATION_FEE

Not in force date: 19940920

PN2301 Change of applicant

St.27 status event code: A-5-5-R10-R13-asn-PN2301

St.27 status event code: A-5-5-R10-R11-asn-PN2301

R18-X000 Changes to party contact information recorded

St.27 status event code: A-5-5-R10-R18-oth-X000

R18-X000 Changes to party contact information recorded

St.27 status event code: A-5-5-R10-R18-oth-X000