KR820001341B1 - 새로운 옥사디아졸로 피리미딘 유도체의 제법 - Google Patents

새로운 옥사디아졸로 피리미딘 유도체의 제법 Download PDF

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Publication number
KR820001341B1
KR820001341B1 KR7902426A KR790002426A KR820001341B1 KR 820001341 B1 KR820001341 B1 KR 820001341B1 KR 7902426 A KR7902426 A KR 7902426A KR 790002426 A KR790002426 A KR 790002426A KR 820001341 B1 KR820001341 B1 KR 820001341B1
Authority
KR
South Korea
Prior art keywords
dihydro
formula
oxide
pyridyl
pyrimidine
Prior art date
Application number
KR7902426A
Other languages
English (en)
Korean (ko)
Inventor
뮬러 제인-클라우드
라뮤즈 헨리
Original Assignee
쿠르트 네젤보쉬
에프 · 호프만-라 롯슈 앤드 캄파니
한스 스튀클린
에프·호프만-라 롯슈 앤드 캄파니
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 쿠르트 네젤보쉬, 에프 · 호프만-라 롯슈 앤드 캄파니, 한스 스튀클린, 에프·호프만-라 롯슈 앤드 캄파니 filed Critical 쿠르트 네젤보쉬
Application granted granted Critical
Publication of KR820001341B1 publication Critical patent/KR820001341B1/ko

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48Two nitrogen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/08Vasodilators for multiple indications
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Chemistry (AREA)
  • Cardiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Compositions Of Macromolecular Compounds (AREA)
KR7902426A 1978-07-21 1979-07-20 새로운 옥사디아졸로 피리미딘 유도체의 제법 KR820001341B1 (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH7910/78 1978-07-21
CH791078 1978-07-21

Publications (1)

Publication Number Publication Date
KR820001341B1 true KR820001341B1 (ko) 1982-07-28

Family

ID=4332239

Family Applications (1)

Application Number Title Priority Date Filing Date
KR7902426A KR820001341B1 (ko) 1978-07-21 1979-07-20 새로운 옥사디아졸로 피리미딘 유도체의 제법

Country Status (14)

Country Link
US (2) US4220772A (US07655688-20100202-C00086.png)
EP (1) EP0008652B1 (US07655688-20100202-C00086.png)
JP (1) JPS5517386A (US07655688-20100202-C00086.png)
KR (1) KR820001341B1 (US07655688-20100202-C00086.png)
AT (1) ATE1584T1 (US07655688-20100202-C00086.png)
CA (1) CA1103245A (US07655688-20100202-C00086.png)
DE (1) DE2963729D1 (US07655688-20100202-C00086.png)
DK (1) DK305879A (US07655688-20100202-C00086.png)
ES (1) ES482675A1 (US07655688-20100202-C00086.png)
FI (1) FI792206A (US07655688-20100202-C00086.png)
GR (1) GR72471B (US07655688-20100202-C00086.png)
HU (1) HU179029B (US07655688-20100202-C00086.png)
NO (1) NO792412L (US07655688-20100202-C00086.png)
PT (1) PT69950A (US07655688-20100202-C00086.png)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK148826C (da) * 1980-12-19 1986-03-24 Hoffmann La Roche Analogifremgangsmaade til fremstilling af oxadiazolopyrimidinderivater eller salte deraf med baser og pyrimidinderivat til anvendelse som mellemprodukt ved denne fremgangsmaade
US5514672A (en) * 1981-02-17 1996-05-07 Bazzano; Gail S. Use of retinoids and compositions containing same for hair growth
US5183817A (en) * 1981-02-17 1993-02-02 Bazzano Gail S Combinations of retinoids and minoxidil-type compounds for hair growth
CA1179344A (en) * 1981-07-15 1984-12-11 Jean-Claude Muller Process for the preparation of 6-¬3,6-dihydro-1(2h)- pyridyl| pyrimidine-3-oxides
CH649291A5 (de) * 1982-03-16 1985-05-15 Hoffmann La Roche Dicarbamate.
EP0187854A4 (en) * 1984-07-13 1987-01-22 Gail S Bazzano SUBSTITUTED PYRIMIDINE OXIDES USEFUL FOR PROMOTING HAIR GROWTH.
JPS62182310U (US07655688-20100202-C00086.png) * 1986-05-12 1987-11-19
JPH0540802Y2 (US07655688-20100202-C00086.png) * 1987-02-26 1993-10-15
JPH0540803Y2 (US07655688-20100202-C00086.png) * 1987-03-26 1993-10-15
JPH0349705U (US07655688-20100202-C00086.png) * 1989-09-22 1991-05-15
US5122075A (en) * 1991-05-17 1992-06-16 Amp Incorporated Electrical connector with improved retention feature

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3317534A (en) * 1963-10-30 1967-05-02 Chugai Pharmaceutical Co Ltd Benzamidopyrimidines
US3705159A (en) * 1970-03-05 1972-12-05 Sandoz Ltd Herbicidal 2,4-di(substituted) amino-6-chloro pyrimidines
US3910928A (en) * 1974-04-26 1975-10-07 Upjohn Co 3-(Cyanimino)-propionitriles
CH638216A5 (de) * 1977-02-04 1983-09-15 Hoffmann La Roche Oxadiazolopyrimidin-deriate.
CH638215A5 (de) * 1977-02-04 1983-09-15 Hoffmann La Roche Oxadiazolopyrimidin-derivate.
JPS6024794A (ja) * 1983-07-19 1985-02-07 Matsushita Electric Ind Co Ltd 撮像素子

Also Published As

Publication number Publication date
US4256886A (en) 1981-03-17
JPS6330908B2 (US07655688-20100202-C00086.png) 1988-06-21
US4220772A (en) 1980-09-02
FI792206A (fi) 1980-01-22
PT69950A (en) 1979-08-01
ES482675A1 (es) 1980-09-01
ATE1584T1 (de) 1982-10-15
NO792412L (no) 1980-01-22
HU179029B (en) 1982-08-28
GR72471B (US07655688-20100202-C00086.png) 1983-11-11
DK305879A (da) 1980-01-22
CA1103245A (en) 1981-06-16
EP0008652A1 (de) 1980-03-19
JPS5517386A (en) 1980-02-06
EP0008652B1 (de) 1982-09-22
DE2963729D1 (en) 1982-11-04

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