KR20180083426A - 비스-피리다진 화합물 및 암 치료에서 이의 용도 - Google Patents
비스-피리다진 화합물 및 암 치료에서 이의 용도 Download PDFInfo
- Publication number
- KR20180083426A KR20180083426A KR1020187017944A KR20187017944A KR20180083426A KR 20180083426 A KR20180083426 A KR 20180083426A KR 1020187017944 A KR1020187017944 A KR 1020187017944A KR 20187017944 A KR20187017944 A KR 20187017944A KR 20180083426 A KR20180083426 A KR 20180083426A
- Authority
- KR
- South Korea
- Prior art keywords
- formula
- pyridazin
- pharmaceutically acceptable
- compound
- methoxy
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/50—Pyridazines; Hydrogenated pyridazines
- A61K31/501—Pyridazines; Hydrogenated pyridazines not condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
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| GB1520959.6 | 2015-11-27 | ||
| GBGB1520959.6A GB201520959D0 (en) | 2015-11-27 | 2015-11-27 | Bis-pyridazine compounds and their use in treating cancer |
| PCT/EP2016/078899 WO2017089587A1 (en) | 2015-11-27 | 2016-11-25 | Bis-pyridazine compounds and their use in treating cancer |
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| KR20180083426A true KR20180083426A (ko) | 2018-07-20 |
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| IL (1) | IL259358A (enExample) |
| MX (1) | MX2018006374A (enExample) |
| RU (1) | RU2018122012A (enExample) |
| SG (1) | SG11201803814SA (enExample) |
| TW (1) | TW201731837A (enExample) |
| WO (1) | WO2017089587A1 (enExample) |
Cited By (1)
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| KR20250137464A (ko) | 2024-03-11 | 2025-09-18 | 이석재 | 숏블라스트머신의 연마재탱크 |
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| CN106552296B (zh) | 2015-09-29 | 2020-08-14 | 上海氪励铵勤科技发展有限公司 | 纳米粒子、其制备方法与结石取出装置及应用 |
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| TW201730188A (zh) | 2015-11-30 | 2017-09-01 | 阿斯特捷利康公司 | 1,3,4-噻二唑化合物及其在治療癌症中之用途 |
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| TW201731511A (zh) | 2015-11-30 | 2017-09-16 | 阿斯特捷利康公司 | １，３，４-噻二唑化合物及其在治療癌症中之用途 |
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| KR20250137464A (ko) | 2024-03-11 | 2025-09-18 | 이석재 | 숏블라스트머신의 연마재탱크 |
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| CN108349951B (zh) | 2020-11-13 |
| US10196382B2 (en) | 2019-02-05 |
| CN108349951A (zh) | 2018-07-31 |
| AU2016360970B2 (en) | 2019-11-07 |
| JP2018535226A (ja) | 2018-11-29 |
| SG11201803814SA (en) | 2018-06-28 |
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