KR20100083814A - 옥사디아졸 디아릴 화합물 - Google Patents

옥사디아졸 디아릴 화합물 Download PDF

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Publication number
KR20100083814A
KR20100083814A KR1020107009974A KR20107009974A KR20100083814A KR 20100083814 A KR20100083814 A KR 20100083814A KR 1020107009974 A KR1020107009974 A KR 1020107009974A KR 20107009974 A KR20107009974 A KR 20107009974A KR 20100083814 A KR20100083814 A KR 20100083814A
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South Korea
Prior art keywords
mmol
formula
methyl
disease
acid
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KR1020107009974A
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English (en)
Korean (ko)
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시릴 몬타뉴
안나 콰트로파니
울프강 소어
아그네스 봄브런
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메르크 세로노 에스. 에이.
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Application filed by 메르크 세로노 에스. 에이. filed Critical 메르크 세로노 에스. 에이.
Publication of KR20100083814A publication Critical patent/KR20100083814A/ko

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    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
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    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
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KR1020107009974A 2007-10-04 2008-10-01 옥사디아졸 디아릴 화합물 KR20100083814A (ko)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
EP07117925 2007-10-04
EP07117925.3 2007-10-04
US99813607P 2007-10-09 2007-10-09
US60/998,136 2007-10-09

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KR20100083814A true KR20100083814A (ko) 2010-07-22

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US (2) US8404676B2 (US07846941-20101207-C00217.png)
EP (1) EP2193126B1 (US07846941-20101207-C00217.png)
JP (3) JP5727223B2 (US07846941-20101207-C00217.png)
KR (1) KR20100083814A (US07846941-20101207-C00217.png)
CN (2) CN104478821B (US07846941-20101207-C00217.png)
AR (1) AR068730A1 (US07846941-20101207-C00217.png)
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