KR20100028656A - 치료 조성물 및 그의 용도 - Google Patents
치료 조성물 및 그의 용도 Download PDFInfo
- Publication number
- KR20100028656A KR20100028656A KR1020107001984A KR20107001984A KR20100028656A KR 20100028656 A KR20100028656 A KR 20100028656A KR 1020107001984 A KR1020107001984 A KR 1020107001984A KR 20107001984 A KR20107001984 A KR 20107001984A KR 20100028656 A KR20100028656 A KR 20100028656A
- Authority
- KR
- South Korea
- Prior art keywords
- pharmaceutically acceptable
- acceptable salt
- compound
- lopinavir
- oxo
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Ceased
Links
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- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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| EA022099B1 (ru) | 2006-09-12 | 2015-11-30 | Джилид Сайэнс, Инк. | Способы и интермедиаты для получения ингибиторов интегразы |
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| AR068403A1 (es) * | 2007-09-11 | 2009-11-18 | Gilead Sciences Inc | Proceso e intermediarios para la preparacion de inhibidores de integrasa |
| HRP20151357T1 (hr) | 2008-05-02 | 2016-01-29 | Gilead Sciences, Inc. | Upotreba äśestica äśvrstog nosaäśa kako bi se poboljšala procesabilnost farmaceutskog agensa |
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| EA030003B1 (ru) | 2012-12-21 | 2018-06-29 | Джилид Сайэнс, Инк. | Полициклическое карбамоилпиридоновое соединение и его фармацевтическое применение для лечения вич-инфекции |
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| TWI677489B (zh) | 2014-06-20 | 2019-11-21 | 美商基利科學股份有限公司 | 多環型胺甲醯基吡啶酮化合物之合成 |
| TW201613936A (en) | 2014-06-20 | 2016-04-16 | Gilead Sciences Inc | Crystalline forms of(2R,5S,13aR)-8-hydroxy-7,9-dioxo-n-(2,4,6-trifluorobenzyl)-2,3,4,5,7,9,13,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepine-10-carboxamide |
| TWI695003B (zh) | 2014-12-23 | 2020-06-01 | 美商基利科學股份有限公司 | 多環胺甲醯基吡啶酮化合物及其醫藥用途 |
| DK3236972T3 (en) | 2014-12-26 | 2021-10-04 | Univ Emory | Antivirale N4-hydroxycytidin-derivativer |
| JP6402259B2 (ja) | 2015-04-02 | 2018-10-10 | ギリアード サイエンシーズ， インコーポレイテッド | 多環式カルバモイルピリドン化合物およびそれらの薬学的使用 |
| JP6804790B1 (ja) | 2017-12-07 | 2020-12-23 | エモリー ユニバーシティー | Ｎ４−ヒドロキシシチジンおよび誘導体ならびにそれらに関連する抗ウイルス用途 |
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| US5484926A (en) * | 1993-10-07 | 1996-01-16 | Agouron Pharmaceuticals, Inc. | HIV protease inhibitors |
| US5914332A (en) * | 1995-12-13 | 1999-06-22 | Abbott Laboratories | Retroviral protease inhibiting compounds |
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2008
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- 2008-06-26 KR KR1020107001984A patent/KR20100028656A/ko not_active Ceased
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- 2008-06-26 CN CN200880022821A patent/CN101743004A/zh active Pending
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- 2008-06-26 CN CN2013101948825A patent/CN103356622A/zh active Pending
- 2008-06-26 AP AP2009005083A patent/AP2490A/xx active
- 2008-06-26 EP EP20080781024 patent/EP2167089A1/en not_active Withdrawn
- 2008-06-26 US US12/666,995 patent/US20110009411A1/en not_active Abandoned
- 2008-06-26 US US12/147,220 patent/US20090093482A1/en not_active Abandoned
- 2008-06-26 SG SG2012046926A patent/SG182228A1/en unknown
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2014
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|---|---|
| EA200971096A1 (ru) | 2010-08-30 |
| CA2691736A1 (en) | 2009-01-08 |
| AR067184A1 (es) | 2009-09-30 |
| US20090093482A1 (en) | 2009-04-09 |
| JP2013199494A (ja) | 2013-10-03 |
| JP5547067B2 (ja) | 2014-07-09 |
| JP5769762B2 (ja) | 2015-08-26 |
| JP2010532373A (ja) | 2010-10-07 |
| CO6251236A2 (es) | 2011-02-21 |
| AP2490A (en) | 2012-10-04 |
| US20140343062A1 (en) | 2014-11-20 |
| AU2008270634A1 (en) | 2009-01-08 |
| US20110009411A1 (en) | 2011-01-13 |
| MX2009013828A (es) | 2010-03-10 |
| IL202745A0 (en) | 2010-06-30 |
| CN101743004A (zh) | 2010-06-16 |
| AU2008270634B2 (en) | 2014-01-16 |
| NZ582089A (en) | 2013-01-25 |
| BRPI0813955A2 (pt) | 2017-05-09 |
| JP2015143277A (ja) | 2015-08-06 |
| ECSP109889A (es) | 2010-03-31 |
| US20170136000A1 (en) | 2017-05-18 |
| AP2009005083A0 (en) | 2009-12-31 |
| UA103881C2 (ru) | 2013-12-10 |
| CN103356622A (zh) | 2013-10-23 |
| SG182228A1 (en) | 2012-07-30 |
| TW200916103A (en) | 2009-04-16 |
| WO2009006203A1 (en) | 2009-01-08 |
| ZA201000468B (en) | 2011-06-29 |
| EP2167089A1 (en) | 2010-03-31 |
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