KR20070086332A - 울혈성 심부전 치료용 ｐｐａｒ 효능제의 용도 - Google Patents
울혈성 심부전 치료용 ｐｐａｒ 효능제의 용도 Download PDFInfo
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- KR20070086332A KR20070086332A KR1020077013671A KR20077013671A KR20070086332A KR 20070086332 A KR20070086332 A KR 20070086332A KR 1020077013671 A KR1020077013671 A KR 1020077013671A KR 20077013671 A KR20077013671 A KR 20077013671A KR 20070086332 A KR20070086332 A KR 20070086332A
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- 230000000302 ischemic effect Effects 0.000 description 1
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- 229940099563 lactobionic acid Drugs 0.000 description 1
- 229940039717 lanolin Drugs 0.000 description 1
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- VZCYOOQTPOCHFL-UPHRSURJSA-N maleic acid Chemical compound OC(=O)\C=C/C(O)=O VZCYOOQTPOCHFL-UPHRSURJSA-N 0.000 description 1
- 239000011976 maleic acid Substances 0.000 description 1
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- 210000000107 myocyte Anatomy 0.000 description 1
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- CWCMIVBLVUHDHK-ZSNHEYEWSA-N phleomycin D1 Chemical compound N([C@H](C(=O)N[C@H](C)[C@@H](O)[C@H](C)C(=O)N[C@@H]([C@H](O)C)C(=O)NCCC=1SC[C@@H](N=1)C=1SC=C(N=1)C(=O)NCCCCNC(N)=N)[C@@H](O[C@H]1[C@H]([C@@H](O)[C@H](O)[C@H](CO)O1)O[C@@H]1[C@H]([C@@H](OC(N)=O)[C@H](O)[C@@H](CO)O1)O)C=1N=CNC=1)C(=O)C1=NC([C@H](CC(N)=O)NC[C@H](N)C(N)=O)=NC(N)=C1C CWCMIVBLVUHDHK-ZSNHEYEWSA-N 0.000 description 1
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Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/08—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D263/10—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
- C07D263/14—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms with radicals substituted by oxygen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/42—Oxazoles
- A61K31/421—1,3-Oxazoles, e.g. pemoline, trimethadione
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Organic Chemistry (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Cardiology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Heart & Thoracic Surgery (AREA)
- Epidemiology (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Hospice & Palliative Care (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP04029946A EP1671633A1 (en) | 2004-12-17 | 2004-12-17 | Use of PPAR agonists for the treatment of congestive heart failure |
| EP04029946.3 | 2004-12-17 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| KR20070086332A true KR20070086332A (ko) | 2007-08-27 |
Family
ID=34927823
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR1020077013671A Withdrawn KR20070086332A (ko) | 2004-12-17 | 2005-12-06 | 울혈성 심부전 치료용 ｐｐａｒ 효능제의 용도 |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US7601863B2 (enExample) |
| EP (2) | EP1671633A1 (enExample) |
| JP (1) | JP2008524129A (enExample) |
| KR (1) | KR20070086332A (enExample) |
| CN (1) | CN101072557A (enExample) |
| AR (1) | AR051723A1 (enExample) |
| AT (1) | ATE498400T1 (enExample) |
| AU (1) | AU2005315920A1 (enExample) |
| BR (1) | BRPI0519661A2 (enExample) |
| CA (1) | CA2590391A1 (enExample) |
| DE (1) | DE602005026443D1 (enExample) |
| IL (1) | IL183810A0 (enExample) |
| MX (1) | MX2007006678A (enExample) |
| MY (1) | MY141010A (enExample) |
| TW (1) | TW200635584A (enExample) |
| WO (1) | WO2006063715A1 (enExample) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7399777B2 (en) | 2001-08-31 | 2008-07-15 | Sanofi-Aventis Deutschland Gmbh | Diarylcycloalkyl derivatives, processes for their preparation and their use as pharmceuticals |
| PL3523283T3 (pl) | 2016-10-05 | 2021-12-13 | Mitobridge, Inc. | Postacie krystaliczne i postacie soli związków stanowiących agonistów ppar |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN101070316A (zh) * | 1999-04-28 | 2007-11-14 | 萨诺费－阿文蒂斯德国有限公司 | 作为ppar受体配体的二芳基酸衍生物 |
| IL160556A0 (en) * | 2001-08-31 | 2004-07-25 | Aventis Pharma Gmbh | Diaryl cycloalkyl derivatives, method for producing the same and the use thereof as ppar activators |
| WO2004082621A2 (en) * | 2003-03-15 | 2004-09-30 | Bethesda Pharmaceuticals, Inc. | Novel ppar agonists, pharmaceutical compositions and uses thereof |
| US6989462B2 (en) * | 2003-03-25 | 2006-01-24 | Sanofi-Aventis Deutschland Gmbh | Synthesis of 2-chloromethyl-6-methylbenzoic ester |
| US6987118B2 (en) * | 2003-05-21 | 2006-01-17 | Pfizer Inc. | Tetrahydroisoquinoline derivatives as PPAR-alpha activators |
-
2004
- 2004-12-17 EP EP04029946A patent/EP1671633A1/en not_active Withdrawn
-
2005
- 2005-12-06 CN CNA2005800416904A patent/CN101072557A/zh active Pending
- 2005-12-06 CA CA002590391A patent/CA2590391A1/en not_active Abandoned
- 2005-12-06 WO PCT/EP2005/013046 patent/WO2006063715A1/en not_active Ceased
- 2005-12-06 AT AT05824351T patent/ATE498400T1/de not_active IP Right Cessation
- 2005-12-06 MX MX2007006678A patent/MX2007006678A/es not_active Application Discontinuation
- 2005-12-06 EP EP05824351A patent/EP1827425B1/en not_active Expired - Lifetime
- 2005-12-06 BR BRPI0519661-2A patent/BRPI0519661A2/pt not_active IP Right Cessation
- 2005-12-06 AU AU2005315920A patent/AU2005315920A1/en not_active Abandoned
- 2005-12-06 DE DE602005026443T patent/DE602005026443D1/de not_active Expired - Lifetime
- 2005-12-06 KR KR1020077013671A patent/KR20070086332A/ko not_active Withdrawn
- 2005-12-06 JP JP2007545894A patent/JP2008524129A/ja not_active Withdrawn
- 2005-12-15 AR ARP050105284A patent/AR051723A1/es not_active Application Discontinuation
- 2005-12-15 TW TW094144376A patent/TW200635584A/zh unknown
- 2005-12-16 MY MYPI20055943A patent/MY141010A/en unknown
-
2007
- 2007-06-10 IL IL183810A patent/IL183810A0/en unknown
- 2007-06-14 US US11/762,799 patent/US7601863B2/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| US7601863B2 (en) | 2009-10-13 |
| WO2006063715A1 (en) | 2006-06-22 |
| DE602005026443D1 (de) | 2011-03-31 |
| EP1827425B1 (en) | 2011-02-16 |
| EP1827425A1 (en) | 2007-09-05 |
| AR051723A1 (es) | 2007-01-31 |
| TW200635584A (en) | 2006-10-16 |
| MX2007006678A (es) | 2007-08-14 |
| CN101072557A (zh) | 2007-11-14 |
| MY141010A (en) | 2010-02-25 |
| EP1671633A1 (en) | 2006-06-21 |
| US20080039512A1 (en) | 2008-02-14 |
| BRPI0519661A2 (pt) | 2009-03-03 |
| IL183810A0 (en) | 2007-10-31 |
| AU2005315920A1 (en) | 2006-06-22 |
| JP2008524129A (ja) | 2008-07-10 |
| CA2590391A1 (en) | 2006-06-22 |
| ATE498400T1 (de) | 2011-03-15 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PA0105 | International application |
Patent event date: 20070615 Patent event code: PA01051R01D Comment text: International Patent Application |
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| PG1501 | Laying open of application | ||
| PC1203 | Withdrawal of no request for examination | ||
| WITN | Application deemed withdrawn, e.g. because no request for examination was filed or no examination fee was paid |