KR20040018359A - 지방족 폴리아민으로 ｘ 증후군을 치료하는 방법 - Google Patents
지방족 폴리아민으로 ｘ 증후군을 치료하는 방법 Download PDFInfo
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- KR20040018359A KR20040018359A KR10-2003-7013679A KR20037013679A KR20040018359A KR 20040018359 A KR20040018359 A KR 20040018359A KR 20037013679 A KR20037013679 A KR 20037013679A KR 20040018359 A KR20040018359 A KR 20040018359A
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- QJGQUHMNIGDVPM-UHFFFAOYSA-N nitrogen group Chemical group [N] QJGQUHMNIGDVPM-UHFFFAOYSA-N 0.000 description 1
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- FYPMFJGVHOHGLL-UHFFFAOYSA-N probucol Chemical compound C=1C(C(C)(C)C)=C(O)C(C(C)(C)C)=CC=1SC(C)(C)SC1=CC(C(C)(C)C)=C(O)C(C(C)(C)C)=C1 FYPMFJGVHOHGLL-UHFFFAOYSA-N 0.000 description 1
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- 230000000069 prophylactic effect Effects 0.000 description 1
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- 239000004405 propyl p-hydroxybenzoate Substances 0.000 description 1
- DNIAPMSPPWPWGF-UHFFFAOYSA-N propylene glycol Substances CC(O)CO DNIAPMSPPWPWGF-UHFFFAOYSA-N 0.000 description 1
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- 102000004169 proteins and genes Human genes 0.000 description 1
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- 238000007142 ring opening reaction Methods 0.000 description 1
- CVHZOJJKTDOEJC-UHFFFAOYSA-N saccharin Chemical compound C1=CC=C2C(=O)NS(=O)(=O)C2=C1 CVHZOJJKTDOEJC-UHFFFAOYSA-N 0.000 description 1
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Classifications
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
- A61K31/352—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline
- A61K31/353—3,4-Dihydrobenzopyrans, e.g. chroman, catechin
- A61K31/355—Tocopherols, e.g. vitamin E
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- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/365—Lactones
- A61K31/375—Ascorbic acid, i.e. vitamin C; Salts thereof
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4415—Pyridoxine, i.e. Vitamin B6
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- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7135—Compounds containing heavy metals
- A61K31/714—Cobalamins, e.g. cyanocobalamin, i.e. vitamin B12
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- A61K31/74—Synthetic polymeric materials
- A61K31/765—Polymers containing oxygen
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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- A61K31/785—Polymers containing nitrogen
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P13/12—Drugs for disorders of the urinary system of the kidneys
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- A—HUMAN NECESSITIES
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- A61P3/12—Drugs for disorders of the metabolism for electrolyte homeostasis
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- A—HUMAN NECESSITIES
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- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/08—Plasma substitutes; Perfusion solutions; Dialytics or haemodialytics; Drugs for electrolytic or acid-base disorders, e.g. hypovolemic shock
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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- Urology & Nephrology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
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| US28444501P | 2001-04-18 | 2001-04-18 | |
| US60/284,445 | 2001-04-18 | ||
| US35591702P | 2002-02-11 | 2002-02-11 | |
| US60/355,917 | 2002-02-11 | ||
| PCT/US2002/011495 WO2002085382A1 (en) | 2001-04-18 | 2002-04-10 | Methods of treating syndrome x with aliphatic polyamines |
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| KR20040018359A true KR20040018359A (ko) | 2004-03-03 |
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| EP (2) | EP2172204A1 (enExample) |
| JP (1) | JP2004526778A (enExample) |
| KR (1) | KR20040018359A (enExample) |
| CN (1) | CN1509180A (enExample) |
| AU (1) | AU2002257147B9 (enExample) |
| BR (1) | BR0209124A (enExample) |
| CA (1) | CA2444028A1 (enExample) |
| MX (1) | MXPA03009562A (enExample) |
| WO (1) | WO2002085382A1 (enExample) |
| ZA (1) | ZA200308066B (enExample) |
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| US6733780B1 (en) | 1999-10-19 | 2004-05-11 | Genzyme Corporation | Direct compression polymer tablet core |
| KR20040018359A (ko) * | 2001-04-18 | 2004-03-03 | 젠자임 코포레이션 | 지방족 폴리아민으로 ｘ 증후군을 치료하는 방법 |
| US7220406B2 (en) * | 2002-10-22 | 2007-05-22 | Genzyme Corporation | Method for promoting bone formation |
| US7335795B2 (en) * | 2004-03-22 | 2008-02-26 | Ilypsa, Inc. | Crosslinked amine polymers |
| US7608674B2 (en) * | 2003-11-03 | 2009-10-27 | Ilypsa, Inc. | Pharmaceutical compositions comprising cross-linked small molecule amine polymers |
| US7459502B2 (en) * | 2003-11-03 | 2008-12-02 | Ilypsa, Inc. | Pharmaceutical compositions comprising crosslinked polyamine polymers |
| US7767768B2 (en) * | 2003-11-03 | 2010-08-03 | Ilypsa, Inc. | Crosslinked amine polymers |
| US7449605B2 (en) * | 2003-11-03 | 2008-11-11 | Ilypsa, Inc. | Crosslinked amine polymers |
| US7385012B2 (en) * | 2003-11-03 | 2008-06-10 | Ilypsa, Inc. | Polyamine polymers |
| US7985418B2 (en) | 2004-11-01 | 2011-07-26 | Genzyme Corporation | Aliphatic amine polymer salts for tableting |
| EP1951266A2 (en) * | 2005-09-02 | 2008-08-06 | Genzyme Corporation | Method for removing phosphate and polymer used therefore |
| CN101272762B (zh) | 2005-09-15 | 2013-02-06 | 基酶有限公司 | 胺聚合物的小袋制剂 |
| EP2016114A2 (en) * | 2006-05-05 | 2009-01-21 | Genzyme Corporation | Amine condensation polymers as phosphate sequestrants |
| BRPI0715053A2 (pt) * | 2006-07-18 | 2013-03-19 | Genzyme Corp | composiÇço farmacÊutica, mÉtodo para tratar doenÇas, e, polÍmero |
| JP2010504975A (ja) | 2006-09-29 | 2010-02-18 | ゲンズイメ コーポレーション | アミドデンドリマー組成物 |
| US8163799B2 (en) * | 2006-12-14 | 2012-04-24 | Genzyme Corporation | Amido-amine polymer compositions |
| WO2008103368A1 (en) * | 2007-02-23 | 2008-08-28 | Genzyme Corporation | Amine polymer compositions |
| EP2131820A1 (en) * | 2007-03-08 | 2009-12-16 | Genzyme Corporation | Sulfone polymer compositions |
| EP2152277A1 (en) * | 2007-04-27 | 2010-02-17 | Genzyme Corporation | Amido-amine dendrimer compositions |
| WO2009078958A1 (en) * | 2007-12-14 | 2009-06-25 | Genzyme Corporation | Coated pharmaceutical compositions |
| US20110142952A1 (en) * | 2008-06-20 | 2011-06-16 | Harris David J | Pharmaceutical Compositions |
| EP2361171A4 (en) * | 2008-09-15 | 2014-11-05 | Shasun Chemicals And Drugs Ltd | PROCESS FOR PREPARING NETWORKED POLYMERS IN A NON-AQUEOUS SOLUTION |
| US9181364B2 (en) | 2010-02-24 | 2015-11-10 | Relypsa, Inc. | Crosslinked polyvinylamine, polyallylamine, and polyethyleneimine for use as bile acid sequestrants |
| US9475891B2 (en) * | 2013-09-19 | 2016-10-25 | Navinta, Llc | Process for the preparation of colesevelam hydrochloride |
| JP6792640B2 (ja) | 2016-12-28 | 2020-11-25 | 富士フイルム株式会社 | 窒素原子含有ポリマー又はその塩の乳化液、その製造方法、及び粒子の製造方法 |
| CN111225674A (zh) | 2017-10-16 | 2020-06-02 | 富士胶片株式会社 | 高磷血症治疗剂 |
| JP6708764B1 (ja) * | 2019-01-28 | 2020-06-10 | 久保田 徹 | 機能水 |
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| US6569905B1 (en) * | 1998-12-23 | 2003-05-27 | G.D. Searle, Llc | Combinations of cholesteryl ester transfer protein inhibitors and bile acid sequestering agents for cardiovascular indications |
| EA004877B1 (ru) * | 1998-12-23 | 2004-08-26 | Джи.Ди.Сирл Ллс | Сочетания ингибиторов транспорта желчных кислот в подвздошной кишке и агентов, секвестрирующих желчные кислоты, для сердечно-сосудистых показаний |
| US6190649B1 (en) | 1999-04-23 | 2001-02-20 | Geltex Pharmaceuticals, Inc. | Polyether-based bile acid sequestrants |
| EP1180114B1 (en) | 1999-04-27 | 2011-09-21 | The Trustees of The University of Pennsylvania | Use of resisitin specific antibodies in the treatment of diabetes |
| EP1212065A4 (en) | 1999-07-08 | 2004-02-11 | Tularik Inc | COMPILATIONS AND METHODS FOR INCREASING THE HDL CHOLESTEROL LEVEL |
| WO2001025291A1 (en) | 1999-10-07 | 2001-04-12 | University Of Maryland | Sugar binding polymers and the use thereof |
| US6627636B2 (en) * | 2000-06-15 | 2003-09-30 | Bristol-Myers Squibb Company | HMG-CoA reductase inhibitors and method |
| KR20040018359A (ko) * | 2001-04-18 | 2004-03-03 | 젠자임 코포레이션 | 지방족 폴리아민으로 ｘ 증후군을 치료하는 방법 |
| US20020198202A1 (en) | 2001-06-07 | 2002-12-26 | Wyeth | Combination of a PTPase inhibitor and an antilipemic agent |
-
2002
- 2002-04-10 KR KR10-2003-7013679A patent/KR20040018359A/ko not_active Withdrawn
- 2002-04-10 EP EP09015042A patent/EP2172204A1/en not_active Withdrawn
- 2002-04-10 EP EP02726735A patent/EP1379259A1/en not_active Ceased
- 2002-04-10 AU AU2002257147A patent/AU2002257147B9/en not_active Ceased
- 2002-04-10 CA CA002444028A patent/CA2444028A1/en not_active Abandoned
- 2002-04-10 WO PCT/US2002/011495 patent/WO2002085382A1/en not_active Ceased
- 2002-04-10 JP JP2002582955A patent/JP2004526778A/ja not_active Withdrawn
- 2002-04-10 MX MXPA03009562A patent/MXPA03009562A/es unknown
- 2002-04-10 CN CNA028100042A patent/CN1509180A/zh active Pending
- 2002-04-10 BR BR0209124-0A patent/BR0209124A/pt not_active Application Discontinuation
- 2002-04-17 US US10/125,701 patent/US7261880B2/en not_active Expired - Lifetime
-
2003
- 2003-10-16 ZA ZA2003/08066A patent/ZA200308066B/en unknown
-
2007
- 2007-06-28 US US11/823,853 patent/US20080085872A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| CN1509180A (zh) | 2004-06-30 |
| AU2002257147B9 (en) | 2005-08-18 |
| AU2002257147B2 (en) | 2005-07-14 |
| ZA200308066B (en) | 2005-03-30 |
| WO2002085382A1 (en) | 2002-10-31 |
| BR0209124A (pt) | 2005-02-09 |
| US20030049226A1 (en) | 2003-03-13 |
| US20080085872A1 (en) | 2008-04-10 |
| JP2004526778A (ja) | 2004-09-02 |
| CA2444028A1 (en) | 2002-10-31 |
| US7261880B2 (en) | 2007-08-28 |
| EP2172204A1 (en) | 2010-04-07 |
| MXPA03009562A (es) | 2004-02-12 |
| EP1379259A1 (en) | 2004-01-14 |
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Legal Events
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| PA0105 | International application |
Patent event date: 20031018 Patent event code: PA01051R01D Comment text: International Patent Application |
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| PG1501 | Laying open of application | ||
| PC1203 | Withdrawal of no request for examination | ||
| WITN | Application deemed withdrawn, e.g. because no request for examination was filed or no examination fee was paid |