KR20040002871A - 시스-ｆｔｃ의 다형 및 기타 결정형 - Google Patents
시스-ｆｔｃ의 다형 및 기타 결정형 Download PDFInfo
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- KR20040002871A KR20040002871A KR10-2003-7011355A KR20037011355A KR20040002871A KR 20040002871 A KR20040002871 A KR 20040002871A KR 20037011355 A KR20037011355 A KR 20037011355A KR 20040002871 A KR20040002871 A KR 20040002871A
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- Prior art keywords
- ftc
- cis
- hydrate
- amorphous
- compound
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- XMGQYMWWDOXHJM-UHFFFAOYSA-N limonene Chemical compound CC(=C)C1CCC(C)=CC1 XMGQYMWWDOXHJM-UHFFFAOYSA-N 0.000 description 1
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- WTJKGGKOPKCXLL-RRHRGVEJSA-N phosphatidylcholine Chemical compound CCCCCCCCCCCCCCCC(=O)OC[C@H](COP([O-])(=O)OCC[N+](C)(C)C)OC(=O)CCCCCCCC=CCCCCCCCC WTJKGGKOPKCXLL-RRHRGVEJSA-N 0.000 description 1
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- IGFXRKMLLMBKSA-UHFFFAOYSA-N purine Chemical compound N1=C[N]C2=NC=NC2=C1 IGFXRKMLLMBKSA-UHFFFAOYSA-N 0.000 description 1
- 239000002718 pyrimidine nucleoside Substances 0.000 description 1
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- ZLGIYFNHBLSMPS-ATJNOEHPSA-N shellac Chemical compound OCCCCCC(O)C(O)CCCCCCCC(O)=O.C1C23[C@H](C(O)=O)CCC2[C@](C)(CO)[C@@H]1C(C(O)=O)=C[C@@H]3O ZLGIYFNHBLSMPS-ATJNOEHPSA-N 0.000 description 1
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Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D411/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms
- C07D411/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D411/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/20—Antivirals for DNA viruses
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/20—Antivirals for DNA viruses
- A61P31/22—Antivirals for DNA viruses for herpes viruses
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Virology (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Engineering & Computer Science (AREA)
- Molecular Biology (AREA)
- Biotechnology (AREA)
- AIDS & HIV (AREA)
- Tropical Medicine & Parasitology (AREA)
- Gastroenterology & Hepatology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Steroid Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US27256001P | 2001-03-01 | 2001-03-01 | |
| US60/272,560 | 2001-03-01 | ||
| US30960501P | 2001-08-02 | 2001-08-02 | |
| US60/309,605 | 2001-08-02 | ||
| PCT/US2002/006184 WO2002070518A1 (en) | 2001-03-01 | 2002-03-01 | Polymorphic and other crystalline forms of cis-ftc |
Related Child Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR1020087016002A Division KR101015510B1 (ko) | 2001-03-01 | 2002-03-01 | 시스-ｆｔｃ의 다형 및 기타 결정형 |
| KR1020087016003A Division KR100927024B1 (ko) | 2001-03-01 | 2002-03-01 | 시스-ｆｔｃ의 다형 및 기타 결정형 |
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|---|---|
| KR20040002871A true KR20040002871A (ko) | 2004-01-07 |
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| KR1020087016003A Expired - Fee Related KR100927024B1 (ko) | 2001-03-01 | 2002-03-01 | 시스-ｆｔｃ의 다형 및 기타 결정형 |
| KR1020107016624A Expired - Fee Related KR101150250B1 (ko) | 2001-03-01 | 2002-03-01 | 시스-ｆｔｃ의 다형 및 기타 결정형 |
| KR10-2003-7011355A Ceased KR20040002871A (ko) | 2001-03-01 | 2002-03-01 | 시스-ｆｔｃ의 다형 및 기타 결정형 |
Family Applications Before (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR1020087016002A Expired - Fee Related KR101015510B1 (ko) | 2001-03-01 | 2002-03-01 | 시스-ｆｔｃ의 다형 및 기타 결정형 |
| KR1020087016003A Expired - Fee Related KR100927024B1 (ko) | 2001-03-01 | 2002-03-01 | 시스-ｆｔｃ의 다형 및 기타 결정형 |
| KR1020107016624A Expired - Fee Related KR101150250B1 (ko) | 2001-03-01 | 2002-03-01 | 시스-ｆｔｃ의 다형 및 기타 결정형 |
Country Status (14)
| Country | Link |
|---|---|
| US (3) | US6723728B2 (enExample) |
| EP (3) | EP1574512B1 (enExample) |
| JP (4) | JP5105689B2 (enExample) |
| KR (4) | KR101015510B1 (enExample) |
| CN (4) | CN102942563A (enExample) |
| AT (2) | ATE383355T1 (enExample) |
| AU (1) | AU2002335489B2 (enExample) |
| CA (4) | CA2788498C (enExample) |
| CY (2) | CY1107983T1 (enExample) |
| DE (2) | DE60224592T2 (enExample) |
| DK (2) | DK1574512T3 (enExample) |
| ES (3) | ES2537007T3 (enExample) |
| PT (2) | PT1574512E (enExample) |
| WO (1) | WO2002070518A1 (enExample) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE60224592T2 (de) * | 2001-03-01 | 2009-01-29 | Abbott Laboratories, Abbott Park | Polymorphe und andere kristalline Formen von cis-FTC |
| TWI244393B (en) * | 2002-08-06 | 2005-12-01 | Idenix Pharmaceuticals Inc | Crystalline and amorphous forms of beta-L-2'-deoxythymidine |
| NZ540728A (en) | 2003-01-14 | 2008-08-29 | Gilead Sciences Inc | Compositions and methods for combination antiviral therapy |
| US6887855B2 (en) | 2003-03-17 | 2005-05-03 | Pharmion Corporation | Forms of 5-azacytidine |
| US6943249B2 (en) * | 2003-03-17 | 2005-09-13 | Ash Stevens, Inc. | Methods for isolating crystalline Form I of 5-azacytidine |
| US20060014949A1 (en) * | 2004-07-13 | 2006-01-19 | Supergen Inc. | Compositions and formulations of decitabine polymorphs and methods of use thereof |
| TWI375560B (en) | 2005-06-13 | 2012-11-01 | Gilead Sciences Inc | Composition comprising dry granulated emtricitabine and tenofovir df and method for making the same |
| TWI471145B (zh) | 2005-06-13 | 2015-02-01 | Bristol Myers Squibb & Gilead Sciences Llc | 單一式藥學劑量型 |
| WO2009005338A2 (en) * | 2007-07-05 | 2009-01-08 | Ultimorphix Technologies B.V. | Solid forms ult-i, ult-2 and ult-3 of emtricitabine |
| EP2350065A1 (en) | 2008-11-12 | 2011-08-03 | Lupin Ltd. | A novel polymorph of emtricitabine and a process for preparing of the same |
| EP2454244B1 (en) | 2009-07-15 | 2013-06-26 | Lupin Limited | An improved process for preparation of efavirenz |
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| WO1989002733A1 (en) | 1987-09-22 | 1989-04-06 | The Regents Of The University Of California | Liposomal nucleoside analogues for treating aids |
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-
2002
- 2002-03-01 DE DE60224592T patent/DE60224592T2/de not_active Expired - Lifetime
- 2002-03-01 CA CA2788498A patent/CA2788498C/en not_active Expired - Fee Related
- 2002-03-01 CN CN2012101468804A patent/CN102942563A/zh active Pending
- 2002-03-01 ES ES08000264.5T patent/ES2537007T3/es not_active Expired - Lifetime
- 2002-03-01 CN CN201210146877.2A patent/CN102911166B/zh not_active Expired - Fee Related
- 2002-03-01 WO PCT/US2002/006184 patent/WO2002070518A1/en not_active Ceased
- 2002-03-01 CA CA2867970A patent/CA2867970A1/en not_active Abandoned
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