JPWO2024111560A5 - - Google Patents

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Publication number
JPWO2024111560A5
JPWO2024111560A5 JP2024560149A JP2024560149A JPWO2024111560A5 JP WO2024111560 A5 JPWO2024111560 A5 JP WO2024111560A5 JP 2024560149 A JP2024560149 A JP 2024560149A JP 2024560149 A JP2024560149 A JP 2024560149A JP WO2024111560 A5 JPWO2024111560 A5 JP WO2024111560A5
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JP
Japan
Prior art keywords
carbonyl
indazol
azetidin
ethan
trifluoromethyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2024560149A
Other languages
English (en)
Japanese (ja)
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JPWO2024111560A1 (https=
JP7823226B2 (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/JP2023/041679 external-priority patent/WO2024111560A1/ja
Publication of JPWO2024111560A1 publication Critical patent/JPWO2024111560A1/ja
Publication of JPWO2024111560A5 publication Critical patent/JPWO2024111560A5/ja
Application granted granted Critical
Publication of JP7823226B2 publication Critical patent/JP7823226B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2024560149A 2022-11-21 2023-11-20 Ddr1キナーゼ阻害剤としての化合物および医薬 Active JP7823226B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2022185827 2022-11-21
JP2022185827 2022-11-21
PCT/JP2023/041679 WO2024111560A1 (ja) 2022-11-21 2023-11-20 Ddr1キナーゼ阻害剤としての化合物および医薬

Publications (3)

Publication Number Publication Date
JPWO2024111560A1 JPWO2024111560A1 (https=) 2024-05-30
JPWO2024111560A5 true JPWO2024111560A5 (https=) 2025-12-09
JP7823226B2 JP7823226B2 (ja) 2026-03-03

Family

ID=91195603

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024560149A Active JP7823226B2 (ja) 2022-11-21 2023-11-20 Ddr1キナーゼ阻害剤としての化合物および医薬

Country Status (12)

Country Link
EP (1) EP4624465A1 (https=)
JP (1) JP7823226B2 (https=)
KR (1) KR20250109234A (https=)
CN (1) CN120569374A (https=)
AU (1) AU2023386923A1 (https=)
CL (1) CL2025001435A1 (https=)
CO (1) CO2025006877A2 (https=)
IL (1) IL320735A (https=)
MX (1) MX2025005556A (https=)
PE (1) PE20251709A1 (https=)
TW (1) TW202430151A (https=)
WO (1) WO2024111560A1 (https=)

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2017A (en) 1841-03-26 The graphic co
IL165863A0 (en) * 2002-06-24 2006-01-15 Schering Corp Indole derivatives useful as histamine H3 antagonists
DE10337184A1 (de) * 2003-08-13 2005-03-10 Gruenenthal Gmbh Substituierte 3-Pyrrolidin-Indol-Derivate
EP1965862A2 (en) * 2005-12-21 2008-09-10 Schering Corporation Combination of an h3 antagonist/inverse agonist and an appetite suppressant
SMT201800070T1 (it) 2012-12-19 2018-03-08 Celgene Quanticel Res Inc Inibiorti di istone demetilasi
US9199945B2 (en) 2013-06-21 2015-12-01 MyoKardia, Inc. Cycloalkyl-substituted pyrimidinedione compounds
US9598419B1 (en) 2014-06-24 2017-03-21 Universite De Montreal Imidazotriazine and imidazodiazine compounds
CN108276388B (zh) * 2017-03-10 2020-01-14 成都医学院 1h-吲哚类衍生物及其用途
KR102297587B1 (ko) * 2018-08-07 2021-09-06 재단법인 대구경북첨단의료산업진흥재단 치환된 n-헤테로아릴 유도체, 이의 제조방법 및 이를 유효성분으로 포함하는 암의 예방 또는 치료용 약학적 조성물
KR102886315B1 (ko) 2018-12-21 2025-11-14 닛산 가가쿠 가부시키가이샤 고분자 및 금속미립자를 포함하는 무전해도금하지제
WO2020210642A1 (en) * 2019-04-10 2020-10-15 Camp4 Therapeutics Corporation Methods and compositions for treating urea cycle disorders
US12403137B2 (en) 2019-10-28 2025-09-02 Tango Therapeutics, Inc. Compounds and methods of use
WO2022051569A1 (en) * 2020-09-04 2022-03-10 Ikena Oncology, Inc. Substituted 3-piperidinyl-pyrrolo[2,3-b]pyridines and related compounds and their use in treating medical conditions
WO2022140290A1 (en) * 2020-12-21 2022-06-30 Cytokinetics, Inc. Pyrazole derivatives useful as nampt modulators

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