JPWO2024075813A1 - - Google Patents

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Publication number
JPWO2024075813A1
JPWO2024075813A1 JP2024521089A JP2024521089A JPWO2024075813A1 JP WO2024075813 A1 JPWO2024075813 A1 JP WO2024075813A1 JP 2024521089 A JP2024521089 A JP 2024521089A JP 2024521089 A JP2024521089 A JP 2024521089A JP WO2024075813 A1 JPWO2024075813 A1 JP WO2024075813A1
Authority
JP
Japan
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2024521089A
Other languages
Japanese (ja)
Other versions
JPWO2024075813A5 (https=
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of JPWO2024075813A1 publication Critical patent/JPWO2024075813A1/ja
Publication of JPWO2024075813A5 publication Critical patent/JPWO2024075813A5/ja
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/02—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
    • C07D241/06—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having one or two double bonds between ring members or between ring members and non-ring members
    • C07D241/08—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having one or two double bonds between ring members or between ring members and non-ring members with oxygen atoms directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/10—Tetrapeptides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04—Linear peptides containing only normal peptide links
    • C07K7/06—Linear peptides containing only normal peptide links having 5 to 11 amino acids

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Analytical Chemistry (AREA)
  • Peptides Or Proteins (AREA)
JP2024521089A 2022-10-07 2023-10-05 Pending JPWO2024075813A1 (https=)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2022162425 2022-10-07
PCT/JP2023/036352 WO2024075813A1 (ja) 2022-10-07 2023-10-05 ジケトピペラジン化合物を用いるポリペプチド合成

Publications (2)

Publication Number Publication Date
JPWO2024075813A1 true JPWO2024075813A1 (https=) 2024-04-11
JPWO2024075813A5 JPWO2024075813A5 (https=) 2024-10-03

Family

ID=90608434

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024521089A Pending JPWO2024075813A1 (https=) 2022-10-07 2023-10-05

Country Status (2)

Country Link
JP (1) JPWO2024075813A1 (https=)
WO (1) WO2024075813A1 (https=)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN119591553A (zh) * 2024-11-19 2025-03-11 上海昊海生物科技股份有限公司 一种二氨基二酮哌嗪类化合物的用途

Citations (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1991014378A1 (en) * 1990-03-15 1991-10-03 The Nutrasweet Company Process for manufacturing aspartame from a diketopiperazine and novel intermediates and derivatives therefor
US5144073A (en) * 1988-08-31 1992-09-01 Hubbs John C Process for preparation of dipeptides
WO2017204144A1 (ja) * 2016-05-23 2017-11-30 学校法人中部大学 水酸基を配向基とするエステルからアミドへの変換触媒
WO2018199146A1 (ja) * 2017-04-25 2018-11-01 学校法人中部大学 オキシム・ヒドロキシアミンを基質とするエステルからアミドへの変換触媒
WO2018199147A1 (ja) * 2017-04-25 2018-11-01 学校法人中部大学 アミド化合物の製造方法
WO2019208731A1 (ja) * 2018-04-25 2019-10-31 学校法人中部大学 アミド化合物の製造方法
WO2021085635A1 (ja) * 2019-10-30 2021-05-06 学校法人中部大学 アミド反応用反応剤及びそれを用いたアミド化合物の製造方法
WO2021149814A1 (ja) * 2020-01-22 2021-07-29 学校法人中部大学 アミド化合物の製造用触媒及び製造方法
JP7181662B1 (ja) * 2021-06-17 2022-12-01 学校法人中部大学 ペプチド化合物の製造方法

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7456184B2 (en) * 2003-05-01 2008-11-25 Palatin Technologies Inc. Melanocortin receptor-specific compounds
CA2506843A1 (en) * 2002-11-22 2004-06-10 Novo-Nordisk A/S 2,5-diketopiperazines for the treatment of obesity
US20110144336A1 (en) * 2008-08-13 2011-06-16 Basf Se Method for Preparation of Piperazindione Derivatives
JP2012504576A (ja) * 2008-10-02 2012-02-23 ビーエーエスエフ ソシエタス・ヨーロピア 除草活性を有するピペラジン化合物
WO2017025031A1 (zh) * 2015-08-10 2017-02-16 于跃 一种抗病毒活性双氮氧杂环螺二酮哌嗪生物碱衍生物及其制备方法
JP7810643B2 (ja) * 2019-11-05 2026-02-03 上▲海▼翰森生物医▲薬▼科技有限公司 ベンゾチオフェン誘導体レギュレーター、その調製法及び使用

Patent Citations (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5144073A (en) * 1988-08-31 1992-09-01 Hubbs John C Process for preparation of dipeptides
WO1991014378A1 (en) * 1990-03-15 1991-10-03 The Nutrasweet Company Process for manufacturing aspartame from a diketopiperazine and novel intermediates and derivatives therefor
WO2017204144A1 (ja) * 2016-05-23 2017-11-30 学校法人中部大学 水酸基を配向基とするエステルからアミドへの変換触媒
WO2018199146A1 (ja) * 2017-04-25 2018-11-01 学校法人中部大学 オキシム・ヒドロキシアミンを基質とするエステルからアミドへの変換触媒
WO2018199147A1 (ja) * 2017-04-25 2018-11-01 学校法人中部大学 アミド化合物の製造方法
WO2019208731A1 (ja) * 2018-04-25 2019-10-31 学校法人中部大学 アミド化合物の製造方法
WO2021085635A1 (ja) * 2019-10-30 2021-05-06 学校法人中部大学 アミド反応用反応剤及びそれを用いたアミド化合物の製造方法
WO2021149814A1 (ja) * 2020-01-22 2021-07-29 学校法人中部大学 アミド化合物の製造用触媒及び製造方法
JP7181662B1 (ja) * 2021-06-17 2022-12-01 学校法人中部大学 ペプチド化合物の製造方法

Non-Patent Citations (8)

* Cited by examiner, † Cited by third party
Title
ANGEW. CHEM. INT. ED. 2006, V.45, PP.1248-1252, vol. 45, JPN6025004909, 2006, pages 1248 - 1252, ISSN: 0005526524 *
BULL. CHEM. SOC. JPN., vol. 58, JPN6024036769, 1985, pages 1413 - 1420, ISSN: 0005417487 *
CHEM. SCI., vol. 13, JPN6025004910, 2022, pages 6309 - 6315, ISSN: 0005526525 *
ORG. BIOMOL. CHEM., vol. 3, JPN6024036768, 2005, pages 1435 - 1447, ISSN: 0005417486 *
SCIENCE, vol. 256, JPN6025004908, 1992, pages 221 - 225, ISSN: 0005526523 *
SYNLETT, JPN6024036767, 1997, pages 483 - 484, ISSN: 0005417485 *
TETRAHEDRON: ASYMMETRY, vol. 12, JPN6024036765, 2001, pages 3387 - 3398, ISSN: 0005417483 *
TETRAHEDRON: ASYMMETRY, vol. 15, JPN6024036766, 2004, pages 3045 - 3058, ISSN: 0005417484 *

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