JPWO2024009977A1 - - Google Patents

Info

Publication number
JPWO2024009977A1
JPWO2024009977A1 JP2024532139A JP2024532139A JPWO2024009977A1 JP WO2024009977 A1 JPWO2024009977 A1 JP WO2024009977A1 JP 2024532139 A JP2024532139 A JP 2024532139A JP 2024532139 A JP2024532139 A JP 2024532139A JP WO2024009977 A1 JPWO2024009977 A1 JP WO2024009977A1
Authority
JP
Japan
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2024532139A
Other languages
Japanese (ja)
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of JPWO2024009977A1 publication Critical patent/JPWO2024009977A1/ja
Pending legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
JP2024532139A 2022-07-05 2023-07-04 Pending JPWO2024009977A1 (enExample)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2022108654 2022-07-05
PCT/JP2023/024703 WO2024009977A1 (ja) 2022-07-05 2023-07-04 5H-ピロロ[2,3-d]ピリミジン-6(7H)-オン及びその塩体の結晶

Publications (1)

Publication Number Publication Date
JPWO2024009977A1 true JPWO2024009977A1 (enExample) 2024-01-11

Family

ID=89453401

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024532139A Pending JPWO2024009977A1 (enExample) 2022-07-05 2023-07-04

Country Status (7)

Country Link
US (1) US20260001883A1 (enExample)
EP (1) EP4553078A1 (enExample)
JP (1) JPWO2024009977A1 (enExample)
CN (1) CN119403807A (enExample)
MA (1) MA71401A (enExample)
TW (1) TW202421127A (enExample)
WO (1) WO2024009977A1 (enExample)

Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2007534687A (ja) * 2004-04-23 2007-11-29 エグゼリクシス, インコーポレイテッド キナーゼ調節因子および使用方法
JP2012508274A (ja) * 2008-11-11 2012-04-05 イーライ リリー アンド カンパニー Aktおよびp70s6キナーゼ阻害剤
WO2017200087A1 (ja) * 2016-05-20 2017-11-23 大鵬薬品工業株式会社 新規5H-ピロロ[2,3-d]ピリミジン-6(7H)-オン誘導体

Patent Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2007534687A (ja) * 2004-04-23 2007-11-29 エグゼリクシス, インコーポレイテッド キナーゼ調節因子および使用方法
JP2012508274A (ja) * 2008-11-11 2012-04-05 イーライ リリー アンド カンパニー Aktおよびp70s6キナーゼ阻害剤
WO2017200087A1 (ja) * 2016-05-20 2017-11-23 大鵬薬品工業株式会社 新規5H-ピロロ[2,3-d]ピリミジン-6(7H)-オン誘導体

Non-Patent Citations (2)

* Cited by examiner, † Cited by third party
Title
平山 令明, 有機化合物結晶作製ハンドブック, JPN6014035600, 2008, pages 17 - 23, ISSN: 0005610294 *
芦澤 一英: "塩・結晶形の最適化と結晶化技術", PHARM TECH JAPAN, vol. 18, no. 10, JPN6013060608, 2002, pages 81 - 96, ISSN: 0005610295 *

Also Published As

Publication number Publication date
WO2024009977A1 (ja) 2024-01-11
TW202421127A (zh) 2024-06-01
EP4553078A1 (en) 2025-05-14
MA71401A (fr) 2025-04-30
CN119403807A (zh) 2025-02-07
US20260001883A1 (en) 2026-01-01

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