JPWO2022255195A1 - - Google Patents
Info
- Publication number
- JPWO2022255195A1 JPWO2022255195A1 JP2022565830A JP2022565830A JPWO2022255195A1 JP WO2022255195 A1 JPWO2022255195 A1 JP WO2022255195A1 JP 2022565830 A JP2022565830 A JP 2022565830A JP 2022565830 A JP2022565830 A JP 2022565830A JP WO2022255195 A1 JPWO2022255195 A1 JP WO2022255195A1
- Authority
- JP
- Japan
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06008—Dipeptides with the first amino acid being neutral
- C07K5/06078—Dipeptides with the first amino acid being neutral and aromatic or cycloaliphatic
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
- C07K1/02—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length in solution
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
- C07K1/06—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents
- C07K1/08—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents using activating agents
- C07K1/088—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents using activating agents containing other elements, e.g. B, Si, As
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/08—Tripeptides
- C07K5/0802—Tripeptides with the first amino acid being neutral
- C07K5/0804—Tripeptides with the first amino acid being neutral and aliphatic
- C07K5/0806—Tripeptides with the first amino acid being neutral and aliphatic the side chain containing 0 or 1 carbon atoms, i.e. Gly, Ala
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- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Genetics & Genomics (AREA)
- Biochemistry (AREA)
- Biophysics (AREA)
- General Health & Medical Sciences (AREA)
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Molecular Biology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Life Sciences & Earth Sciences (AREA)
- Analytical Chemistry (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2021091438 | 2021-05-31 | ||
JP2021091438 | 2021-05-31 | ||
PCT/JP2022/021434 WO2022255195A1 (ja) | 2021-05-31 | 2022-05-25 | ペプチド化合物の製造方法及びアミド化反応剤 |
Publications (3)
Publication Number | Publication Date |
---|---|
JPWO2022255195A1 true JPWO2022255195A1 (ja) | 2022-12-08 |
JPWO2022255195A5 JPWO2022255195A5 (ja) | 2023-05-15 |
JP7327858B2 JP7327858B2 (ja) | 2023-08-16 |
Family
ID=84323169
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP2022565830A Active JP7327858B2 (ja) | 2021-05-31 | 2022-05-25 | ペプチド化合物の製造方法及びアミド化反応剤 |
Country Status (3)
Country | Link |
---|---|
EP (1) | EP4349848A1 (ja) |
JP (1) | JP7327858B2 (ja) |
WO (1) | WO2022255195A1 (ja) |
Citations (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP2009507906A (ja) * | 2005-09-13 | 2009-02-26 | ユニヴァーシティー オブ リーディング | ペプチドの不斉合成 |
WO2009060843A1 (ja) * | 2007-11-09 | 2009-05-14 | Gifu University | アミド化触媒、カルボン酸アミドの製造方法、及びペプチドの製造方法 |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP3466922A4 (en) | 2016-05-23 | 2020-01-08 | Chubu University Educational Foundation | ESTER CONVERSION CATALYST HAVING HYDROXYL GROUP AS AMIDE ALIGNMENT GROUP |
EP3617185A4 (en) | 2017-04-25 | 2021-01-20 | Chubu University Educational Foundation | METHOD FOR PREPARING AN AMIDE COMPOUND |
JPWO2018199146A1 (ja) | 2017-04-25 | 2020-02-27 | 学校法人中部大学 | オキシム・ヒドロキシアミンを基質とするエステルからアミドへの変換触媒 |
JP7122019B2 (ja) | 2018-04-25 | 2022-08-19 | 学校法人中部大学 | アミド化合物の製造方法 |
JP7244134B2 (ja) | 2019-10-30 | 2023-03-22 | 学校法人中部大学 | アミド反応用反応剤及びそれを用いたアミド化合物の製造方法 |
WO2021085635A1 (ja) | 2019-10-30 | 2021-05-06 | 学校法人中部大学 | アミド反応用反応剤及びそれを用いたアミド化合物の製造方法 |
US20230121469A1 (en) | 2020-01-22 | 2023-04-20 | Chubu University Educational Foundation | Catalyst for manufacturing amide compound, and method for manufacturing amide compound |
-
2022
- 2022-05-25 WO PCT/JP2022/021434 patent/WO2022255195A1/ja active Application Filing
- 2022-05-25 JP JP2022565830A patent/JP7327858B2/ja active Active
- 2022-05-25 EP EP22815945.5A patent/EP4349848A1/en active Pending
Patent Citations (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP2009507906A (ja) * | 2005-09-13 | 2009-02-26 | ユニヴァーシティー オブ リーディング | ペプチドの不斉合成 |
WO2009060843A1 (ja) * | 2007-11-09 | 2009-05-14 | Gifu University | アミド化触媒、カルボン酸アミドの製造方法、及びペプチドの製造方法 |
Non-Patent Citations (6)
Title |
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CHUNG, S. W. ET AL.: "Trimethylaluminium-Facilitated Direct Amidation of Carboxylic Acids", SYNLETT, JPN7022003898, 2011, pages 2072 - 2074, XP055132481, ISSN: 0004972143 * |
DUBOIS, N. ET AL.: "On DABAL-Me3 promoted formation of amides", TETRAHEDRON, vol. 69, JPN6022033694, 2013, pages 9890 - 9897, ISSN: 0004972145 * |
LI, J. ET AL.: "AlMe3-Promoted Formation of Amides from Acids and Amines", ORG. LETT., vol. 14, no. 1, JPN7022003899, 2012, pages 214 - 217, XP093009377, ISSN: 0004972144, DOI: 10.1021/ol203007s * |
MARTIN, S. F. ET AL.: "APPLICATION OF AIMe3-MEDIATED AMIDATION REACTIONS TO SOLUTION PHASE PEPTIDE SYNTHESIS", TETRAHEDRON LETTERS, vol. 39, JPN7022003895, 1998, pages 1517 - 1520, XP004108088, ISSN: 0004972140, DOI: 10.1016/S0040-4039(98)00071-9 * |
MURAMATSU, W. ET AL.: "Game Change from Reagent- to Substrate-Controlled Peptide Synthesis", BULL. CHEM. SOC. JPN., vol. 93, JPN7022003897, 2020, pages 759 - 767, XP055930673, ISSN: 0004972142, DOI: 10.1246/bcsj.20200057 * |
MURAMATSU, W. ET AL.: "Substrate-Directed Lewis-Acid Catalysis for Peptide Synthesis", J. AM. CHEM. SOC., vol. 141, JPN7022003896, 2019, pages 12288 - 12295, XP055930667, ISSN: 0004972141, DOI: 10.1021/jacs.9b03850 * |
Also Published As
Publication number | Publication date |
---|---|
WO2022255195A1 (ja) | 2022-12-08 |
EP4349848A1 (en) | 2024-04-10 |
JP7327858B2 (ja) | 2023-08-16 |
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