JPWO2022251497A5 - - Google Patents

Download PDF

Info

Publication number
JPWO2022251497A5
JPWO2022251497A5 JP2023573154A JP2023573154A JPWO2022251497A5 JP WO2022251497 A5 JPWO2022251497 A5 JP WO2022251497A5 JP 2023573154 A JP2023573154 A JP 2023573154A JP 2023573154 A JP2023573154 A JP 2023573154A JP WO2022251497 A5 JPWO2022251497 A5 JP WO2022251497A5
Authority
JP
Japan
Prior art keywords
methyl
ethyl
amino
pyridazine
dione
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2023573154A
Other languages
English (en)
Japanese (ja)
Other versions
JP2024521818A (ja
JP2024521818A5 (https=
Publication date
Application filed filed Critical
Priority claimed from PCT/US2022/031133 external-priority patent/WO2022251497A1/en
Publication of JP2024521818A publication Critical patent/JP2024521818A/ja
Publication of JP2024521818A5 publication Critical patent/JP2024521818A5/ja
Publication of JPWO2022251497A5 publication Critical patent/JPWO2022251497A5/ja
Pending legal-status Critical Current

Links

JP2023573154A 2021-05-27 2022-05-26 ヘテロ環式化合物およびその使用方法 Pending JP2024521818A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US202163193831P 2021-05-27 2021-05-27
US63/193,831 2021-05-27
US202163226980P 2021-07-29 2021-07-29
US63/226,980 2021-07-29
PCT/US2022/031133 WO2022251497A1 (en) 2021-05-27 2022-05-26 Heterocyclic compounds and methods of use

Publications (3)

Publication Number Publication Date
JP2024521818A JP2024521818A (ja) 2024-06-04
JP2024521818A5 JP2024521818A5 (https=) 2025-06-03
JPWO2022251497A5 true JPWO2022251497A5 (https=) 2025-06-03

Family

ID=84229207

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023573154A Pending JP2024521818A (ja) 2021-05-27 2022-05-26 ヘテロ環式化合物およびその使用方法

Country Status (5)

Country Link
US (1) US20240279221A1 (https=)
EP (1) EP4346815A4 (https=)
JP (1) JP2024521818A (https=)
KR (1) KR20240013792A (https=)
WO (1) WO2022251497A1 (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW202334095A (zh) * 2021-12-23 2023-09-01 大陸商北京望實智慧科技有限公司 Sos1抑制劑
EP4463454A1 (en) 2022-01-14 2024-11-20 Jazz Pharmaceuticals Ireland Limited Novel amine-substituted phthalazines and derivatives as sos1 inhibitors
CR20240362A (es) * 2022-02-04 2024-10-03 Schroedinger Inc Compuestos heterocíclicos y métodos de uso

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EA200801996A1 (ru) * 2006-04-20 2009-04-28 Глаксо Груп Лимитед 2-замещенные производные 4-бензилфталазинонов в качестве гистаминовых h1- и h3-антагонистов
ATE459358T1 (de) * 2006-12-20 2010-03-15 Glaxo Group Ltd 4-benzyl-1(2h)-phthalazinone als h1-rezeptor- antagonisten
WO2014169843A1 (en) * 2013-04-18 2014-10-23 Shanghai Fochon Pharmaceutical Co Ltd Certain protein kinase inhibitors
EP3189049B1 (en) * 2014-09-05 2024-03-20 Genentech, Inc. Phthalazine derivatives of formula (i) as pcaf and gcn5 inhibitors for use in the treatment of cancer
RS64167B1 (sr) * 2017-12-21 2023-05-31 Boehringer Ingelheim Int Benzilamino supstituisani piridopirimidinoni i derivati kao sos1 inhibitori
TW202334095A (zh) * 2021-12-23 2023-09-01 大陸商北京望實智慧科技有限公司 Sos1抑制劑
CN118574830A (zh) * 2022-01-28 2024-08-30 中山优理生物医药有限公司 一种哒嗪并吡啶酮类化合物、其药物组合物及应用

Similar Documents

Publication Publication Date Title
JP2012528178A5 (https=)
RU2011152973A (ru) Индуцирующие апоптоз средства для лечения злокачественной опухоли и иммунных и аутоиммунных заболеваний
RU2473549C2 (ru) Пиримидиновые соединения, композиции и способы применения
JP2025535046A (ja) Kras g12c変異タンパク質の複素環阻害剤及びその使用
JP5808793B2 (ja) キナーゼ調節のための化合物および方法、ならびにそれらの適応症
HRP20240994T1 (hr) Spoj inhibitora jak i njegova uporaba
JP2019523233A5 (https=)
JP2010510319A5 (https=)
JP2017048219A5 (https=)
RU2014139601A (ru) Ингибиторы серин/треониновых киназ
JP2019038820A5 (https=)
JP2021506816A5 (https=)
JP5901634B2 (ja) キナゾリン化合物及びその使用方法
JP2018044008A5 (https=)
HRP20130106T1 (hr) Imidazotriazini i imidazopirimidini kao inhibitori kinaze
CA2984259A1 (en) Combinations of inhibitors of irak4 with inhibitors of btk
RU2012127760A (ru) Bcl-2-селективные апоптоз-индуцирующие средства для лечения рака и иммунных заболеваний
RU2012104493A (ru) Замещенные соединения пиразоло [1,5-a] пиримидина как ингибиторы киназы trk
CN113993866A (zh) 杂芳基衍生物、其制备方法、及含其作为有效成分的药物组合物
RU2019123319A (ru) Пиразолопиримидины и способы их применения
HRP20120457T1 (hr) 4-(4-cijano-2-tioaril)dihidropirimidinoni i njihova uporaba
JP2018512381A5 (https=)
JP2011511034A5 (https=)
JP2010523576A5 (https=)
JP2022500402A5 (https=)