JPWO2005030722A1 - Ｎ−置換−ｎ−（４−ピペリジニル）アミド誘導体 - Google Patents

Ｎ−置換−ｎ−（４−ピペリジニル）アミド誘導体 Download PDF

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Publication number
JPWO2005030722A1
JPWO2005030722A1 JP2005514305A JP2005514305A JPWO2005030722A1 JP WO2005030722 A1 JPWO2005030722 A1 JP WO2005030722A1 JP 2005514305 A JP2005514305 A JP 2005514305A JP 2005514305 A JP2005514305 A JP 2005514305A JP WO2005030722 A1 JPWO2005030722 A1 JP WO2005030722A1
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JP
Japan
Prior art keywords
group
carbon atoms
alkyl
methyl
phenylpropionylamino
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2005514305A
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English (en)
Japanese (ja)
Inventor
高橋　俊弘
俊弘 高橋
遠藤　剛
剛 遠藤
佐久間　詔悟
詔悟 佐久間
望月　信孝
信孝 望月
山川　富雄
富雄 山川
喜一 四家
喜一 四家
透 川崎
透 川崎
利安 今井
利安 今井
謙二 平手
謙二 平手
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Nippon Chemiphar Co Ltd
Original Assignee
Nippon Chemiphar Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Nippon Chemiphar Co Ltd filed Critical Nippon Chemiphar Co Ltd
Publication of JPWO2005030722A1 publication Critical patent/JPWO2005030722A1/ja
Pending legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/60—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D211/62—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals attached in position 4
    • C07D211/66—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals attached in position 4 having a hetero atom as the second substituent in position 4
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pain & Pain Management (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
JP2005514305A 2003-09-29 2004-09-28 Ｎ−置換−ｎ−（４−ピペリジニル）アミド誘導体 Pending JPWO2005030722A1 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2003337480 2003-09-29
JP2003337480 2003-09-29
PCT/JP2004/014562 WO2005030722A1 (fr) 2003-09-29 2004-09-28 Derive d'amide de n-(4-piperidinyle) n-substitue

Publications (1)

Publication Number Publication Date
JPWO2005030722A1 true JPWO2005030722A1 (ja) 2006-12-07

Family

ID=34386125

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2005514305A Pending JPWO2005030722A1 (ja) 2003-09-29 2004-09-28 Ｎ−置換−ｎ−（４−ピペリジニル）アミド誘導体

Country Status (2)

Country Link
JP (1) JPWO2005030722A1 (fr)
WO (1) WO2005030722A1 (fr)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2006030931A1 (fr) * 2004-09-14 2006-03-23 Nippon Chemiphar Co., Ltd. Derive d’amide n-(4-piperidinyl) n-substitue
WO2016100940A1 (fr) 2014-12-19 2016-06-23 The Broad Institute, Inc. Ligands des récepteurs dopaminergiques d2
US10752588B2 (en) 2014-12-19 2020-08-25 The Broad Institute, Inc. Dopamine D2 receptor ligands
WO2017180659A1 (fr) * 2016-04-11 2017-10-19 Arizona Board Of Regents On Behalf Of University Of Arizona Modulateurs des récepteurs opioïdes

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA852315B (en) * 1984-04-09 1985-11-27 Boc Inc N-aryl-n-(4-piperindinyl)amides and pharmaceutical compositions and methods employing such compounds
US5019583A (en) * 1989-02-15 1991-05-28 Glaxo Inc. N-phenyl-N-(4-piperidinyl)amides useful as analgesics
JPWO2003082819A1 (ja) * 2002-04-01 2005-08-04 日本ケミファ株式会社 Ｎ−フェニル−ｎ−（４−ピペリジニル）アミド誘導体

Also Published As

Publication number Publication date
WO2005030722A1 (fr) 2005-04-07

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