JPS62198687A - ２β−置換チオメチルペニシリン誘導体 - Google Patents

２β−置換チオメチルペニシリン誘導体

Info

Publication number
JPS62198687A
JPS62198687A JP61043763A JP4376386A JPS62198687A JP S62198687 A JPS62198687 A JP S62198687A JP 61043763 A JP61043763 A JP 61043763A JP 4376386 A JP4376386 A JP 4376386A JP S62198687 A JPS62198687 A JP S62198687A
Authority
JP
Japan
Prior art keywords
acid
methyl
group
reaction
water
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP61043763A
Other languages
English (en)
Japanese (ja)
Other versions
JPH0523271B2 (cs
Inventor
Shigeru Torii
滋 鳥居
Hideo Tanaka
秀雄 田中
Motoaki Tanaka
基明 田中
Shozo Yamada
省三 山田
Akira Nakai
中井　章
Hisashi Obayashi
尚志 大林
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Taiho Pharmaceutical Co Ltd
Original Assignee
Taiho Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Taiho Pharmaceutical Co Ltd filed Critical Taiho Pharmaceutical Co Ltd
Priority to JP61043763A priority Critical patent/JPS62198687A/ja
Priority to US07/016,114 priority patent/US4861768A/en
Priority to AU69094/87A priority patent/AU573115B2/en
Priority to CA000530613A priority patent/CA1281319C/en
Priority to EP87301699A priority patent/EP0236074B1/en
Priority to ES198787301699T priority patent/ES2038656T3/es
Priority to DE8787301699T priority patent/DE3775794D1/de
Priority to KR1019870001744A priority patent/KR920005829B1/ko
Publication of JPS62198687A publication Critical patent/JPS62198687A/ja
Publication of JPH0523271B2 publication Critical patent/JPH0523271B2/ja
Granted legal-status Critical Current

Links

Classifications

    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
JP61043763A 1986-02-27 1986-02-27 ２β−置換チオメチルペニシリン誘導体 Granted JPS62198687A (ja)

Priority Applications (8)

Application Number Priority Date Filing Date Title
JP61043763A JPS62198687A (ja) 1986-02-27 1986-02-27 ２β−置換チオメチルペニシリン誘導体
US07/016,114 US4861768A (en) 1986-02-27 1987-02-18 2 β-substituted thiomethylpenicillin derivatives and their preparation and use
AU69094/87A AU573115B2 (en) 1986-02-27 1987-02-20 2b-substituted thiomethylpenicillin derivatives
CA000530613A CA1281319C (en) 1986-02-27 1987-02-25 2.beta.-SUBSTITUTED THIOMETHYLPENICILLIN DERIVATIVES AND THEIR PREPARATION AND USE
EP87301699A EP0236074B1 (en) 1986-02-27 1987-02-26 2beta-substituted thiomethylpenicillin derivatives and their preparation and use
ES198787301699T ES2038656T3 (es) 1986-02-27 1987-02-26 Derivados de la tiometilpenicilina substituidos en beta y su preparacion y uso.
DE8787301699T DE3775794D1 (de) 1986-02-27 1987-02-26 2-beta-substituierte thiomethyl-penizillinderivate und ihre herstellung und verwendung.
KR1019870001744A KR920005829B1 (ko) 1986-02-27 1987-02-27 2β-치환된 티오메틸페니실린 유도체 및 그의 염의 제조방법

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP61043763A JPS62198687A (ja) 1986-02-27 1986-02-27 ２β−置換チオメチルペニシリン誘導体

Publications (2)

Publication Number Publication Date
JPS62198687A true JPS62198687A (ja) 1987-09-02
JPH0523271B2 JPH0523271B2 (cs) 1993-04-02

Family

ID=12672794

Family Applications (1)

Application Number Title Priority Date Filing Date
JP61043763A Granted JPS62198687A (ja) 1986-02-27 1986-02-27 ２β−置換チオメチルペニシリン誘導体

Country Status (1)

Country Link
JP (1) JPS62198687A (cs)

Cited By (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6770759B2 (en) 1997-12-29 2004-08-03 Research Corporation Technologies, Inc. Penicillanic acid derivative compounds and methods of making
US6906054B2 (en) 1999-04-15 2005-06-14 Research Corporation Technologies, Inc. Compositions for inhibiting beta-lactamase
US6916801B2 (en) 2001-07-24 2005-07-12 Alamx, Llc 7-Alkylidene-3-substituted-3-cephem-4-carboxylates as β-lactamase inhibitors
US7022691B2 (en) 2002-04-04 2006-04-04 John D. Buynak Inhibitors of serine and metallo-β-lactamases
CN114423766A (zh) * 2019-09-11 2022-04-29 丹诺医药(苏州）有限公司 用于治疗细菌感染的青霉烷衍生物

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5657788A (en) * 1979-09-26 1981-05-20 Pfizer Acetoxymethylpenam compound as betaalactamase inhibitor
EP0170192A1 (en) * 1984-07-30 1986-02-05 Merck & Co. Inc. Penicillin derivatives as anti-inflammatory and antidegenerative agents

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5657788A (en) * 1979-09-26 1981-05-20 Pfizer Acetoxymethylpenam compound as betaalactamase inhibitor
EP0170192A1 (en) * 1984-07-30 1986-02-05 Merck & Co. Inc. Penicillin derivatives as anti-inflammatory and antidegenerative agents

Cited By (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6770759B2 (en) 1997-12-29 2004-08-03 Research Corporation Technologies, Inc. Penicillanic acid derivative compounds and methods of making
US7125986B2 (en) 1997-12-29 2006-10-24 Southern Methodist University Foundation For Research Penicillanic acid derivative compounds and methods of making
US6906054B2 (en) 1999-04-15 2005-06-14 Research Corporation Technologies, Inc. Compositions for inhibiting beta-lactamase
US6916801B2 (en) 2001-07-24 2005-07-12 Alamx, Llc 7-Alkylidene-3-substituted-3-cephem-4-carboxylates as β-lactamase inhibitors
US7488724B2 (en) 2001-07-24 2009-02-10 Southern Methodist University Foundation For Research 7-alkylidene-3-substituted-3-cephem-4-carboxylates as beta-lactamase inhibitors
US7022691B2 (en) 2002-04-04 2006-04-04 John D. Buynak Inhibitors of serine and metallo-β-lactamases
CN114423766A (zh) * 2019-09-11 2022-04-29 丹诺医药(苏州）有限公司 用于治疗细菌感染的青霉烷衍生物

Also Published As

Publication number Publication date
JPH0523271B2 (cs) 1993-04-02

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