JPS60222497A - ５αリダクターゼの阻害剤としての１７β―Ｎ―モノ置換カルバモイル―４―アザ―５α―アンドロスタ―１―エン―３―オン類 - Google Patents

５αリダクターゼの阻害剤としての１７β―Ｎ―モノ置換カルバモイル―４―アザ―５α―アンドロスタ―１―エン―３―オン類

Info

Publication number
JPS60222497A
JPS60222497A JP60036714A JP3671485A JPS60222497A JP S60222497 A JPS60222497 A JP S60222497A JP 60036714 A JP60036714 A JP 60036714A JP 3671485 A JP3671485 A JP 3671485A JP S60222497 A JPS60222497 A JP S60222497A
Authority
JP
Japan
Prior art keywords
methyl
aza
hydrogen
compound
carbon atoms
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP60036714A
Other languages
English (en)
Japanese (ja)
Other versions
JPS6365080B2 (enExample
Inventor
ギヤレイ　エツチ．ラスムソン
グレン　エフ．レイノズル
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Merck and Co Inc
Original Assignee
Merck and Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck and Co Inc filed Critical Merck and Co Inc
Publication of JPS60222497A publication Critical patent/JPS60222497A/ja
Publication of JPS6365080B2 publication Critical patent/JPS6365080B2/ja
Granted legal-status Critical Current

Links

Landscapes

  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
JP60036714A 1984-02-27 1985-02-27 ５αリダクターゼの阻害剤としての１７β―Ｎ―モノ置換カルバモイル―４―アザ―５α―アンドロスタ―１―エン―３―オン類 Granted JPS60222497A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US58406184A 1984-02-27 1984-02-27
US584062 1984-02-27
US584061 1984-02-27

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP63135348A Division JPH0193600A (ja) 1984-02-27 1988-06-01 ５αリダクターゼの阻害剤としての１７β―アシル―４―アザ―５α―アンドロスタ―１―エン―３―オン類

Publications (2)

Publication Number Publication Date
JPS60222497A true JPS60222497A (ja) 1985-11-07
JPS6365080B2 JPS6365080B2 (enExample) 1988-12-14

Family

ID=24335771

Family Applications (1)

Application Number Title Priority Date Filing Date
JP60036714A Granted JPS60222497A (ja) 1984-02-27 1985-02-27 ５αリダクターゼの阻害剤としての１７β―Ｎ―モノ置換カルバモイル―４―アザ―５α―アンドロスタ―１―エン―３―オン類

Country Status (2)

Country Link
JP (1) JPS60222497A (enExample)
ZA (1) ZA851426B (enExample)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH05255381A (ja) * 1991-12-17 1993-10-05 Merck & Co Inc １７β−Ｎ−モノ置換カルバモイル−４−アザ−５α−アンドロスト−１−エン−３−オンによる前立腺癌予防剤
WO1997027875A1 (fr) * 1996-02-05 1997-08-07 Sankyo Company, Limited PREPARATION INHIBITRICE DE LA 5α-REDUCTASE ADMINISTRABLE PAR VOIE ORALE, PROCEDE DE PRODUCTION ET UTILISATION

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW382595B (en) 1993-10-15 2000-02-21 Merck & Co Inc Pharmaceutical composition for use in arresting and reversing androgenic alopecia

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS54145669A (en) * 1978-04-13 1979-11-14 Merck & Co Inc 44azaa177substitutedd5 alphaaandrostanee33one which is testosteronee5 alphaareductase repressor

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS54145669A (en) * 1978-04-13 1979-11-14 Merck & Co Inc 44azaa177substitutedd5 alphaaandrostanee33one which is testosteronee5 alphaareductase repressor

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH05255381A (ja) * 1991-12-17 1993-10-05 Merck & Co Inc １７β−Ｎ−モノ置換カルバモイル−４−アザ−５α−アンドロスト−１−エン−３−オンによる前立腺癌予防剤
WO1997027875A1 (fr) * 1996-02-05 1997-08-07 Sankyo Company, Limited PREPARATION INHIBITRICE DE LA 5α-REDUCTASE ADMINISTRABLE PAR VOIE ORALE, PROCEDE DE PRODUCTION ET UTILISATION

Also Published As

Publication number Publication date
ZA851426B (en) 1986-10-29
JPS6365080B2 (enExample) 1988-12-14

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