JPS5939429B2 - ベンジルピリミジンの製造方法 - Google Patents

ベンジルピリミジンの製造方法

Info

Publication number
JPS5939429B2
JPS5939429B2 JP49020031A JP2003174A JPS5939429B2 JP S5939429 B2 JPS5939429 B2 JP S5939429B2 JP 49020031 A JP49020031 A JP 49020031A JP 2003174 A JP2003174 A JP 2003174A JP S5939429 B2 JPS5939429 B2 JP S5939429B2
Authority
JP
Japan
Prior art keywords
formula
diamino
solution
mixture
pyrimidine
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
JP49020031A
Other languages
English (en)
Japanese (ja)
Other versions
JPS49117478A (nl
Inventor
ロ−ゼン ペリ−
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
F Hoffmann La Roche AG
Original Assignee
F Hoffmann La Roche AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by F Hoffmann La Roche AG filed Critical F Hoffmann La Roche AG
Publication of JPS49117478A publication Critical patent/JPS49117478A/ja
Publication of JPS5939429B2 publication Critical patent/JPS5939429B2/ja
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48—Two nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48—Two nitrogen atoms
    • C07D239/49—Two nitrogen atoms with an aralkyl radical, or substituted aralkyl radical, attached in position 5, e.g. trimethoprim

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Liquid Crystal Substances (AREA)
JP49020031A 1973-02-26 1974-02-21 ベンジルピリミジンの製造方法 Expired JPS5939429B2 (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US33609473A 1973-02-26 1973-02-26
US336094 1973-02-26

Publications (2)

Publication Number Publication Date
JPS49117478A JPS49117478A (nl) 1974-11-09
JPS5939429B2 true JPS5939429B2 (ja) 1984-09-22

Family

ID=23314538

Family Applications (1)

Application Number Title Priority Date Filing Date
JP49020031A Expired JPS5939429B2 (ja) 1973-02-26 1974-02-21 ベンジルピリミジンの製造方法

Country Status (8)

Country Link
JP (1) JPS5939429B2 (nl)
AT (1) AT338272B (nl)
BE (1) BE811504A (nl)
CH (1) CH592066A5 (nl)
DE (1) DE2405683A1 (nl)
FR (1) FR2219162B1 (nl)
GB (1) GB1409034A (nl)
NL (1) NL180104C (nl)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH039130Y2 (nl) * 1984-07-31 1991-03-07

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5888368A (ja) * 1981-11-09 1983-05-26 ザ・ウエルカム・フアウンデ−シヨン・リミテツド ベンジルピリミジン誘導体の製造法
EP0111440A1 (en) * 1982-10-15 1984-06-20 Ciba-Geigy Ag 2-Aminopyrimidines, their production and use

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
YU35002B (en) * 1970-10-22 1980-06-30 Wellcome Found Process for preparing 2,4-diamino-5-benzyl-pyrimidine
BE789904A (fr) * 1971-10-12 1973-04-10 Wellcome Found Procedes de synthese organique

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH039130Y2 (nl) * 1984-07-31 1991-03-07

Also Published As

Publication number Publication date
FR2219162B1 (nl) 1977-09-16
JPS49117478A (nl) 1974-11-09
NL180104C (nl) 1987-01-02
BE811504A (fr) 1974-08-26
CH592066A5 (nl) 1977-10-14
ATA151974A (de) 1976-12-15
NL7401764A (nl) 1974-08-28
DE2405683A1 (de) 1974-09-05
NL180104B (nl) 1986-08-01
GB1409034A (en) 1975-10-08
FR2219162A1 (nl) 1974-09-20
AT338272B (de) 1977-08-10

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