JPH09188680A5 - - Google Patents

Info

Publication number
JPH09188680A5
JPH09188680A5 JP1996264860A JP26486096A JPH09188680A5 JP H09188680 A5 JPH09188680 A5 JP H09188680A5 JP 1996264860 A JP1996264860 A JP 1996264860A JP 26486096 A JP26486096 A JP 26486096A JP H09188680 A5 JPH09188680 A5 JP H09188680A5
Authority
JP
Japan
Prior art keywords
compound
formula
pharmaceutical composition
prophylactically
infection
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP1996264860A
Other languages
English (en)
Japanese (ja)
Other versions
JPH09188680A (ja
Filing date
Publication date
Application filed filed Critical
Publication of JPH09188680A publication Critical patent/JPH09188680A/ja
Publication of JPH09188680A5 publication Critical patent/JPH09188680A5/ja
Pending legal-status Critical Current

Links

JP8264860A 1995-10-06 1996-10-04 8−アリールアルキル−及び8−アリールヘテロアルキル−5,11−ジヒドロ−6H−ジピリド[3,2−b:2’,3’−e][1,4]ジアゼピン及びHIV 感染症の予防または治療におけるそれらの使用 Pending JPH09188680A (ja)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US480695P 1995-10-06 1995-10-06
US869595P 1995-12-15 1995-12-15
US60/004806 1995-12-15
US60/008695 1995-12-15

Publications (2)

Publication Number Publication Date
JPH09188680A JPH09188680A (ja) 1997-07-22
JPH09188680A5 true JPH09188680A5 (enExample) 2004-10-14

Family

ID=26673503

Family Applications (1)

Application Number Title Priority Date Filing Date
JP8264860A Pending JPH09188680A (ja) 1995-10-06 1996-10-04 8−アリールアルキル−及び8−アリールヘテロアルキル−5,11−ジヒドロ−6H−ジピリド[3,2−b:2’,3’−e][1,4]ジアゼピン及びHIV 感染症の予防または治療におけるそれらの使用

Country Status (8)

Country Link
US (1) US5705499A (enExample)
EP (1) EP0767172B1 (enExample)
JP (1) JPH09188680A (enExample)
AT (1) ATE235495T1 (enExample)
DE (1) DE69626915T2 (enExample)
DK (1) DK0767172T3 (enExample)
ES (1) ES2191075T3 (enExample)
PT (1) PT767172E (enExample)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5747488A (en) * 1996-01-30 1998-05-05 Boehringer Ingelheim Pharmaceuticals, Inc. 2-aryl-5,11-dihydro-6H-dipyrido 3,2-B:2',3'-E! 1, 4!diazepines and their use in the treatment of HIV infection
GB9715584D0 (en) * 1997-07-23 1997-10-01 Eisai Co Ltd Compounds
UA71971C2 (en) 1999-06-04 2005-01-17 Agoron Pharmaceuticals Inc Diaminothiazoles, composition based thereon, a method for modulation of protein kinases activity, a method for the treatment of diseases mediated by protein kinases
US6455554B1 (en) 1999-06-07 2002-09-24 Targacept, Inc. Oxopyridinyl pharmaceutical compositions and methods for use
US7141581B2 (en) * 1999-07-02 2006-11-28 Agouron Pharmaceuticals, Inc. Indazole compounds and pharmaceutical compositions for inhibiting protein kinases, and methods for their use
TWI262914B (en) 1999-07-02 2006-10-01 Agouron Pharma Compounds and pharmaceutical compositions for inhibiting protein kinases
HN2001000008A (es) * 2000-01-21 2003-12-11 Inc Agouron Pharmaceuticals Compuesto de amida y composiciones farmaceuticas para inhibir proteinquinasas, y su modo de empleo
WO2001079198A1 (en) 2000-04-18 2001-10-25 Agouron Pharmaceuticals, Inc. Pyrazoles for inhibiting protein kinase
SI1294720T1 (sl) * 2000-06-16 2006-08-31 Boehringer Ingelheim Ca Ltd Nenukleozidni inhibitorji reverzne transkriptaze
TWI270547B (en) * 2000-06-16 2007-01-11 Boehringer Ingelheim Ca Ltd Non-nucleoside reverse transcriptase inhibitors
US6716836B2 (en) * 2001-03-22 2004-04-06 Boehringer Ingelheim (Canada) Ltd. Non-nucleoside reverse transcriptase inhibitors
US6673791B2 (en) 2001-07-30 2004-01-06 Boehringer Ingelheim (Canada) Ltd. Non-nucleoside reverse transcriptase inhibitors
US6706706B2 (en) * 2002-03-27 2004-03-16 Boehringer Ingelheim International Gmbh Non-nucleoside reverse transcriptase inhibitors
US6806265B2 (en) * 2002-05-16 2004-10-19 Boehringer Ingelheim International Gmbh Non-nucleoside reverse transcriptase inhibitors
EP1554276B1 (en) * 2002-09-19 2006-06-28 Boehringer Ingelheim (Canada) Ltd. Non-nucleoside reverse transcriptase inhibitors
JP2006505532A (ja) * 2002-09-19 2006-02-16 ベーリンガー インゲルハイム (カナダ) リミテッド 非ヌクレオシド逆転写酵素インヒビター
WO2004043367A2 (en) 2002-11-06 2004-05-27 Bristol-Myers Squibb Company Fused heterocyclic compounds and use thereof
WO2004087140A1 (en) * 2003-03-27 2004-10-14 Boehringer Ingelheim International Gmbh Antiviral combination of a dipyridodiazepinone and a further antiretroviral compound
RU2006139933A (ru) * 2004-04-13 2008-05-20 Икаген, Инк. (Us) Полициклические пиридины как модуляторы калиевых ионных каналов
CA2573673A1 (en) 2004-07-16 2006-01-26 Proteosys Ag Muscarinic antagonists with parp and sir modulating activity as cytoprotective agents
EP2379080A1 (en) 2009-01-13 2011-10-26 ProteoSys AG Pirenzepine as otoprotective agent
CN107428747A (zh) 2014-11-25 2017-12-01 拜耳制药股份公司 取代的吡啶并苯并二氮杂*酮衍生物及其用途

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5366972A (en) * 1989-04-20 1994-11-22 Boehringer Ingelheim Pharmaceuticals, Inc. 5,11-dihydro-6H-dipyrido(3,2-B:2',3'-E)(1,4)diazepines and their use in the prevention or treatment of HIV infection
EP0745083B1 (en) * 1994-02-18 1998-05-20 Boehringer Ingelheim Pharmaceuticals Inc. 2-HETEROARYL-5,11-DIHYDRO-6H-DIPYRIDO [3,2-b:2',3'-e][1,4]DIAZEPINES AND THEIR USE IN THE PREVENTION OR TREATMENT OF HIV INFECTION

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