ES2191075T3 - 8-arilalquil- y 8-arilheteroalquil-5,11-dihidro-6h-dipirido-(3,2-b:2',3'-e)(1,4)diazepinas y su uso en la prevencion o tratamiento de infecciones por hiv. - Google Patents
8-arilalquil- y 8-arilheteroalquil-5,11-dihidro-6h-dipirido-(3,2-b:2',3'-e)(1,4)diazepinas y su uso en la prevencion o tratamiento de infecciones por hiv.Info
- Publication number
- ES2191075T3 ES2191075T3 ES96115901T ES96115901T ES2191075T3 ES 2191075 T3 ES2191075 T3 ES 2191075T3 ES 96115901 T ES96115901 T ES 96115901T ES 96115901 T ES96115901 T ES 96115901T ES 2191075 T3 ES2191075 T3 ES 2191075T3
- Authority
- ES
- Spain
- Prior art keywords
- prevention
- treatment
- hiv
- dipirido
- arilheteroalquil
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
- C07D471/14—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/04—Immunostimulants
-
- C—CHEMISTRY; METALLURGY
- C09—DYES; PAINTS; POLISHES; NATURAL RESINS; ADHESIVES; COMPOSITIONS NOT OTHERWISE PROVIDED FOR; APPLICATIONS OF MATERIALS NOT OTHERWISE PROVIDED FOR
- C09B—ORGANIC DYES OR CLOSELY-RELATED COMPOUNDS FOR PRODUCING DYES, e.g. PIGMENTS; MORDANTS; LAKES
- C09B57/00—Other synthetic dyes of known constitution
Abstract
LA INVENCION SE REFIERE A NUEVAS 8-ARILALQUIL-5,11-DIHIDRO-6HDIPIRIDO-[[]3,2-B:2'',3''-E[]][[]1,4[]]DIAZEPINAS DE FORMULA GENERAL 1 LAS CUALES SON UTILES EN LA PREVENCION O TRATAMIENTO DE INFECCION POR VIH.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US480695P | 1995-10-06 | 1995-10-06 | |
US869595P | 1995-12-15 | 1995-12-15 |
Publications (1)
Publication Number | Publication Date |
---|---|
ES2191075T3 true ES2191075T3 (es) | 2003-09-01 |
Family
ID=26673503
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES96115901T Expired - Lifetime ES2191075T3 (es) | 1995-10-06 | 1996-10-04 | 8-arilalquil- y 8-arilheteroalquil-5,11-dihidro-6h-dipirido-(3,2-b:2',3'-e)(1,4)diazepinas y su uso en la prevencion o tratamiento de infecciones por hiv. |
Country Status (8)
Country | Link |
---|---|
US (1) | US5705499A (es) |
EP (1) | EP0767172B1 (es) |
JP (1) | JPH09188680A (es) |
AT (1) | ATE235495T1 (es) |
DE (1) | DE69626915T2 (es) |
DK (1) | DK0767172T3 (es) |
ES (1) | ES2191075T3 (es) |
PT (1) | PT767172E (es) |
Families Citing this family (22)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5747488A (en) * | 1996-01-30 | 1998-05-05 | Boehringer Ingelheim Pharmaceuticals, Inc. | 2-aryl-5,11-dihydro-6H-dipyrido 3,2-B:2',3'-E! 1, 4!diazepines and their use in the treatment of HIV infection |
GB9715584D0 (en) * | 1997-07-23 | 1997-10-01 | Eisai Co Ltd | Compounds |
UA71971C2 (en) | 1999-06-04 | 2005-01-17 | Agoron Pharmaceuticals Inc | Diaminothiazoles, composition based thereon, a method for modulation of protein kinases activity, a method for the treatment of diseases mediated by protein kinases |
US6455554B1 (en) | 1999-06-07 | 2002-09-24 | Targacept, Inc. | Oxopyridinyl pharmaceutical compositions and methods for use |
US7141581B2 (en) * | 1999-07-02 | 2006-11-28 | Agouron Pharmaceuticals, Inc. | Indazole compounds and pharmaceutical compositions for inhibiting protein kinases, and methods for their use |
TWI262914B (en) * | 1999-07-02 | 2006-10-01 | Agouron Pharma | Compounds and pharmaceutical compositions for inhibiting protein kinases |
HN2001000008A (es) * | 2000-01-21 | 2003-12-11 | Inc Agouron Pharmaceuticals | Compuesto de amida y composiciones farmaceuticas para inhibir proteinquinasas, y su modo de empleo |
JP2004501083A (ja) | 2000-04-18 | 2004-01-15 | アゴーロン・ファーマシューティカルズ・インコーポレイテッド | プロテインキナーゼを阻害するためのピラゾール |
SI1294720T1 (sl) * | 2000-06-16 | 2006-08-31 | Boehringer Ingelheim Ca Ltd | Nenukleozidni inhibitorji reverzne transkriptaze |
TWI270547B (en) * | 2000-06-16 | 2007-01-11 | Boehringer Ingelheim Ca Ltd | Non-nucleoside reverse transcriptase inhibitors |
US6716836B2 (en) | 2001-03-22 | 2004-04-06 | Boehringer Ingelheim (Canada) Ltd. | Non-nucleoside reverse transcriptase inhibitors |
US6673791B2 (en) * | 2001-07-30 | 2004-01-06 | Boehringer Ingelheim (Canada) Ltd. | Non-nucleoside reverse transcriptase inhibitors |
US6706706B2 (en) * | 2002-03-27 | 2004-03-16 | Boehringer Ingelheim International Gmbh | Non-nucleoside reverse transcriptase inhibitors |
US6806265B2 (en) * | 2002-05-16 | 2004-10-19 | Boehringer Ingelheim International Gmbh | Non-nucleoside reverse transcriptase inhibitors |
AU2003269628A1 (en) * | 2002-09-19 | 2004-04-08 | Boehringer Ingelheim (Canada) Ltd. | Non-nucleoside reverse transcriptase inhibitors |
JP4391426B2 (ja) * | 2002-09-19 | 2009-12-24 | ベーリンガー インゲルハイム (カナダ) リミテッド | 非ヌクレオシド逆転写酵素インヒビター |
US7384937B2 (en) | 2002-11-06 | 2008-06-10 | Bristol-Myers Squibb Co. | Fused heterocyclic compounds and use thereof |
WO2004087140A1 (en) * | 2003-03-27 | 2004-10-14 | Boehringer Ingelheim International Gmbh | Antiviral combination of a dipyridodiazepinone and a further antiretroviral compound |
RU2006139933A (ru) * | 2004-04-13 | 2008-05-20 | Икаген, Инк. (Us) | Полициклические пиридины как модуляторы калиевых ионных каналов |
AU2005263578B2 (en) | 2004-07-16 | 2010-09-02 | Proteosys Ag | Muscarinic antagonists with PARP and SIR modulating activity as agents for inflammatory diseases |
EP2387405A2 (en) | 2009-01-13 | 2011-11-23 | ProteoSys AG | Pirenzepine as an agent in cancer treatment |
WO2016083276A1 (de) | 2014-11-25 | 2016-06-02 | Bayer Pharma Aktiengesellschaft | Substituierte pyridobenzodiazepinon-derivate und ihre verwendung |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5366972A (en) * | 1989-04-20 | 1994-11-22 | Boehringer Ingelheim Pharmaceuticals, Inc. | 5,11-dihydro-6H-dipyrido(3,2-B:2',3'-E)(1,4)diazepines and their use in the prevention or treatment of HIV infection |
TW327171B (en) * | 1994-02-18 | 1998-02-21 | Boehringer Ingelheim Pharma | 2-heteroaryl-5 for prevention or treatment of HIV infection |
-
1996
- 1996-09-25 US US08/710,996 patent/US5705499A/en not_active Expired - Lifetime
- 1996-10-04 DK DK96115901T patent/DK0767172T3/da active
- 1996-10-04 JP JP8264860A patent/JPH09188680A/ja active Pending
- 1996-10-04 DE DE69626915T patent/DE69626915T2/de not_active Expired - Fee Related
- 1996-10-04 EP EP96115901A patent/EP0767172B1/en not_active Expired - Lifetime
- 1996-10-04 PT PT96115901T patent/PT767172E/pt unknown
- 1996-10-04 AT AT96115901T patent/ATE235495T1/de not_active IP Right Cessation
- 1996-10-04 ES ES96115901T patent/ES2191075T3/es not_active Expired - Lifetime
Also Published As
Publication number | Publication date |
---|---|
PT767172E (pt) | 2003-08-29 |
EP0767172B1 (en) | 2003-03-26 |
DK0767172T3 (da) | 2003-07-21 |
ATE235495T1 (de) | 2003-04-15 |
DE69626915D1 (de) | 2003-04-30 |
DE69626915T2 (de) | 2003-11-13 |
US5705499A (en) | 1998-01-06 |
EP0767172A1 (en) | 1997-04-09 |
JPH09188680A (ja) | 1997-07-22 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
ES2191075T3 (es) | 8-arilalquil- y 8-arilheteroalquil-5,11-dihidro-6h-dipirido-(3,2-b:2',3'-e)(1,4)diazepinas y su uso en la prevencion o tratamiento de infecciones por hiv. | |
ID26043A (id) | Turunan-turunan 1,3,5-triazina tertrisubstitusi untuk pengobatan infeksi-infeksi hiv | |
ES2130114T3 (es) | 5,11-dihidro-6h-dipirido(3,2-b:2',3'-e)(1,4)diazepinas y su uso en la prevencion o tratamiento de infeccion por hiv. | |
FI933568A0 (fi) | 9-((substituerad glycyl)amido)-6-demetyl-6-deoxitetracykliner | |
DE69433784D1 (de) | 9-(Substituiertes Glycyl)amido-6-(substituiert)-5-hydroxy-6-deoxytetracycline | |
FI20000516A (fi) | Bis-indolyylimaleimidijohdannaiset ja niiden valmistus | |
DK1109817T3 (da) | Phosphohalogenhydriner, deres fremstilling og anvendelse | |
DK0604183T3 (da) | HIV-protease-inhibitorer anvendelige i behandlingen af AIDS | |
DE69825128D1 (de) | Verwendung von azithromycin zur topischen behandlung von augeninfektionen | |
EP0387802A3 (en) | 5-substituted-1,4-dihydro-4-oxonaphthyridine-3-carboxylate antibacterial agents | |
HUP0002836A2 (hu) | Makrociklusos bisz(3,3'-indolil)-maleinimid-származékok alkalmazása bőrrendellenességek kezelésére szolgáló gyógyszerkészítmények előállítására | |
TW327171B (en) | 2-heteroaryl-5 for prevention or treatment of HIV infection | |
ES2102772T3 (es) | Compuesto citotoxico y antiviral. | |
MA25501A1 (fr) | Traitement de l'endometriosis ou de la sterilite ou amelioration de la fertilite. | |
DK291390D0 (da) | Terapeutiske anvendelser af 2',5'-oligoadenylatderivater | |
EE03514B1 (et) | Ühendite kombinatsioon HIV infektsiooni või AIDS-i raviks, selle kasutamine ja farmatseutiline kompositsioon | |
BG102404A (en) | The application of flupirtin for the prevention and treatment of diseases related to impairement of the haematopoeic cellular system | |
AU2979899A (en) | Treatment of viral disease in swine | |
GR3015469T3 (en) | 5,11-dihydro-6H-pyrido[2,3,-b][1,4]benzodiazepin-6-ones and -thiones and their use in the prevention or treatment of AIDS. | |
PT889044E (pt) | Derivados do 5-(heteroaril)alquil-3-oxo-pirido-(1,2-a)benzimidazole-4-carboxamida (pbi) uteis no tratamento de perturbacoes do sistema nervoso central | |
DK0544168T3 (da) | Anvendelse af aminoalkyl-substituerede 5,6-dihydro-dibenz(b,e) azepin-6,11-dion-11-oximer som antivirale midler | |
ES2078380T3 (es) | Oligofosfatos de accion antiviral. | |
NO960551D0 (no) | Antistoff basert behandling av HIV infeksjon | |
DK0412941T3 (da) | Phospholipider til behandling af dissemineret sklerose | |
MX9604346A (es) | 8-arilalquil- y 8-arilheteroalquil-5,11-dihidro-6h-dipirido [3,2-b :2',3'-e] [1,4]diazepinas y su uso en la prevencion o tratamiento de infeccion por hiv. |