JP7700229B2 - ベンゾイミダゾール化合物又はその塩類及び該化合物を含有する犬糸状虫症防除剤並びにその使用方法 - Google Patents
ベンゾイミダゾール化合物又はその塩類及び該化合物を含有する犬糸状虫症防除剤並びにその使用方法 Download PDFInfo
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- JP7700229B2 JP7700229B2 JP2023525915A JP2023525915A JP7700229B2 JP 7700229 B2 JP7700229 B2 JP 7700229B2 JP 2023525915 A JP2023525915 A JP 2023525915A JP 2023525915 A JP2023525915 A JP 2023525915A JP 7700229 B2 JP7700229 B2 JP 7700229B2
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- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
- A01N43/50—1,3-Diazoles; Hydrogenated 1,3-diazoles
- A01N43/52—1,3-Diazoles; Hydrogenated 1,3-diazoles condensed with carbocyclic rings, e.g. benzimidazoles
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01P—BIOCIDAL, PEST REPELLANT, PEST ATTRACTANT OR PLANT GROWTH REGULATORY ACTIVITY OF CHEMICAL COMPOUNDS OR PREPARATIONS
- A01P7/00—Arthropodicides
- A01P7/04—Insecticides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/141—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
- A61K9/143—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with inorganic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/141—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
- A61K9/145—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1617—Organic compounds, e.g. phospholipids, fats
- A61K9/1623—Sugars or sugar alcohols, e.g. lactose; Derivatives thereof; Homeopathic globules
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/14—Ectoparasiticides, e.g. scabicides
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Epidemiology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Tropical Medicine & Parasitology (AREA)
- Pest Control & Pesticides (AREA)
- Plant Pathology (AREA)
- Environmental Sciences (AREA)
- Zoology (AREA)
- Wood Science & Technology (AREA)
- Biophysics (AREA)
- Inorganic Chemistry (AREA)
- Molecular Biology (AREA)
- Insects & Arthropods (AREA)
- Agronomy & Crop Science (AREA)
- Dentistry (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2021092795 | 2021-06-02 | ||
| JP2021092795 | 2021-06-02 | ||
| JP2022021145 | 2022-02-15 | ||
| JP2022021145 | 2022-02-15 | ||
| PCT/JP2022/022536 WO2022255460A1 (ja) | 2021-06-02 | 2022-06-02 | ベンゾイミダゾール化合物又はその塩類及び該化合物を含有する犬糸状虫症防除剤並びにその使用方法 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JPWO2022255460A1 JPWO2022255460A1 (https=) | 2022-12-08 |
| JPWO2022255460A5 JPWO2022255460A5 (https=) | 2024-03-11 |
| JP7700229B2 true JP7700229B2 (ja) | 2025-06-30 |
Family
ID=84324302
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2023525915A Active JP7700229B2 (ja) | 2021-06-02 | 2022-06-02 | ベンゾイミダゾール化合物又はその塩類及び該化合物を含有する犬糸状虫症防除剤並びにその使用方法 |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US20240270712A1 (https=) |
| EP (1) | EP4349824A4 (https=) |
| JP (1) | JP7700229B2 (https=) |
| KR (1) | KR20240012540A (https=) |
| AU (1) | AU2022286144A1 (https=) |
| BR (1) | BR112023024371A2 (https=) |
| CA (1) | CA3222199A1 (https=) |
| CL (1) | CL2023003509A1 (https=) |
| CO (1) | CO2023017613A2 (https=) |
| MX (1) | MX2023014032A (https=) |
| PH (1) | PH12023553295A1 (https=) |
| UA (1) | UA130072C2 (https=) |
| WO (1) | WO2022255460A1 (https=) |
| ZA (1) | ZA202311796B (https=) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MX2022016546A (es) * | 2020-07-03 | 2023-02-01 | Nihon Nohyaku Co Ltd | Agente anticoccidio y metodo para su uso. |
Citations (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2010524892A (ja) | 2007-04-19 | 2010-07-22 | ノバルティス アーゲー | 代謝型グルタミン酸受容体−5の修飾因子としてのニコチン酸誘導体 |
| WO2012020725A1 (ja) | 2010-08-10 | 2012-02-16 | 塩野義製薬株式会社 | Npy y5受容体拮抗作用を有するヘテロ環誘導体 |
| JP2013522365A (ja) | 2010-03-23 | 2013-06-13 | シーメンス メディカル ソリューションズ ユーエスエー インコーポレイテッド | 神経性疾患の検出のためのイメージング剤 |
| CN108440396A (zh) | 2018-03-23 | 2018-08-24 | 吉林奥来德光电材料股份有限公司 | 一种有机发光材料及其制备方法和应用 |
| WO2019049061A1 (en) | 2017-09-07 | 2019-03-14 | Glaxosmithkline Intellectual Property Development Limited | 5- (1H-BENZO [D] IMIDAZO-2-YL) -PYRIDIN-2-AMINE AND 5- (3H-IMIDAZO [4,5-B] PYRIDIN-6-YL) -PYRIDIN-2- DERIVATIVES AMINE AS HISTONE ACETYLTRANSFERASE INHIBITORS OF C-MYC AND P300 / CBP FOR THE TREATMENT OF CANCER |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TWI652014B (zh) * | 2013-09-13 | 2019-03-01 | 美商艾佛艾姆希公司 | 雜環取代之雙環唑殺蟲劑 |
| EP3798212A4 (en) * | 2018-05-22 | 2022-03-23 | Nihon Nohyaku Co., Ltd. | BENZIMIDAZOLE COMPOUND OR SALT THEREOF, INSECTICIDE AND ACARICIDE FOR AGRICULTURE AND HORTICULTURE WITH THIS COMPOUND AND METHODS OF USE |
| MX2022016546A (es) * | 2020-07-03 | 2023-02-01 | Nihon Nohyaku Co Ltd | Agente anticoccidio y metodo para su uso. |
-
2022
- 2022-06-02 WO PCT/JP2022/022536 patent/WO2022255460A1/ja not_active Ceased
- 2022-06-02 UA UAA202306097A patent/UA130072C2/uk unknown
- 2022-06-02 JP JP2023525915A patent/JP7700229B2/ja active Active
- 2022-06-02 PH PH1/2023/553295A patent/PH12023553295A1/en unknown
- 2022-06-02 MX MX2023014032A patent/MX2023014032A/es unknown
- 2022-06-02 CA CA3222199A patent/CA3222199A1/en active Pending
- 2022-06-02 BR BR112023024371A patent/BR112023024371A2/pt unknown
- 2022-06-02 AU AU2022286144A patent/AU2022286144A1/en active Pending
- 2022-06-02 US US18/566,534 patent/US20240270712A1/en active Pending
- 2022-06-02 EP EP22816205.3A patent/EP4349824A4/en not_active Withdrawn
- 2022-06-02 KR KR1020237044492A patent/KR20240012540A/ko not_active Ceased
-
2023
- 2023-11-24 CL CL2023003509A patent/CL2023003509A1/es unknown
- 2023-12-15 CO CONC2023/0017613A patent/CO2023017613A2/es unknown
- 2023-12-21 ZA ZA2023/11796A patent/ZA202311796B/en unknown
Patent Citations (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2010524892A (ja) | 2007-04-19 | 2010-07-22 | ノバルティス アーゲー | 代謝型グルタミン酸受容体−5の修飾因子としてのニコチン酸誘導体 |
| JP2013522365A (ja) | 2010-03-23 | 2013-06-13 | シーメンス メディカル ソリューションズ ユーエスエー インコーポレイテッド | 神経性疾患の検出のためのイメージング剤 |
| WO2012020725A1 (ja) | 2010-08-10 | 2012-02-16 | 塩野義製薬株式会社 | Npy y5受容体拮抗作用を有するヘテロ環誘導体 |
| WO2019049061A1 (en) | 2017-09-07 | 2019-03-14 | Glaxosmithkline Intellectual Property Development Limited | 5- (1H-BENZO [D] IMIDAZO-2-YL) -PYRIDIN-2-AMINE AND 5- (3H-IMIDAZO [4,5-B] PYRIDIN-6-YL) -PYRIDIN-2- DERIVATIVES AMINE AS HISTONE ACETYLTRANSFERASE INHIBITORS OF C-MYC AND P300 / CBP FOR THE TREATMENT OF CANCER |
| CN108440396A (zh) | 2018-03-23 | 2018-08-24 | 吉林奥来德光电材料股份有限公司 | 一种有机发光材料及其制备方法和应用 |
Non-Patent Citations (3)
| Title |
|---|
| Journal of Medicinal Chemistry,2017年,Vol. 60,p. 3594-3605 |
| REGISTRY(STN)[online],2021年03月15日,[検索日] 2024.11.13 ,CAS登録番号2610844-42-1他 |
| Tetrahedron Letters,2008年,Vol. 49, No. 47,p. 6667-6669 |
Also Published As
| Publication number | Publication date |
|---|---|
| CO2023017613A2 (es) | 2024-01-15 |
| JPWO2022255460A1 (https=) | 2022-12-08 |
| WO2022255460A1 (ja) | 2022-12-08 |
| UA130072C2 (uk) | 2025-10-29 |
| KR20240012540A (ko) | 2024-01-29 |
| CA3222199A1 (en) | 2022-12-08 |
| MX2023014032A (es) | 2023-12-15 |
| BR112023024371A2 (pt) | 2024-02-15 |
| AU2022286144A1 (en) | 2024-01-18 |
| ZA202311796B (en) | 2025-04-30 |
| EP4349824A1 (en) | 2024-04-10 |
| CL2023003509A1 (es) | 2024-05-17 |
| US20240270712A1 (en) | 2024-08-15 |
| PH12023553295A1 (en) | 2024-03-18 |
| EP4349824A4 (en) | 2024-10-16 |
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