JP6367545B2 - ルキソリチニブの重水素化誘導体 - Google Patents
ルキソリチニブの重水素化誘導体 Download PDFInfo
- Publication number
- JP6367545B2 JP6367545B2 JP2013259713A JP2013259713A JP6367545B2 JP 6367545 B2 JP6367545 B2 JP 6367545B2 JP 2013259713 A JP2013259713 A JP 2013259713A JP 2013259713 A JP2013259713 A JP 2013259713A JP 6367545 B2 JP6367545 B2 JP 6367545B2
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- deuterium
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- 0 CC1(*)C(*)([C@@](*)(C(*)(*)C#N)[n]2nc(*)c(-c3nc(*)nc4c3c(*)c(*)[n]4)c2*)C(*)(*)C(*)(*)C1(*)* Chemical compound CC1(*)C(*)([C@@](*)(C(*)(*)C#N)[n]2nc(*)c(-c3nc(*)nc4c3c(*)c(*)[n]4)c2*)C(*)(*)C(*)(*)C1(*)* 0.000 description 1
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Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2013259713A JP6367545B2 (ja) | 2013-12-17 | 2013-12-17 | ルキソリチニブの重水素化誘導体 |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2013259713A JP6367545B2 (ja) | 2013-12-17 | 2013-12-17 | ルキソリチニブの重水素化誘導体 |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2018128417A Division JP6830460B2 (ja) | 2018-07-05 | 2018-07-05 | ルキソリチニブの重水素化誘導体 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2015117185A JP2015117185A (ja) | 2015-06-25 |
| JP2015117185A5 JP2015117185A5 (enExample) | 2017-02-09 |
| JP6367545B2 true JP6367545B2 (ja) | 2018-08-01 |
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2013259713A Active JP6367545B2 (ja) | 2013-12-17 | 2013-12-17 | ルキソリチニブの重水素化誘導体 |
Country Status (1)
| Country | Link |
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| JP (1) | JP6367545B2 (enExample) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2018172421A (ja) * | 2018-07-05 | 2018-11-08 | コンサート ファーマシューティカルズ インコーポレイテッド | ルキソリチニブの重水素化誘導体 |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MX394605B (es) | 2015-06-30 | 2025-03-24 | Eiger Group Int Inc | Uso de compuestos de cloroquina y clemizol para el tratamiento de afecciones inflamatorias y cancerosas. |
| WO2017054739A1 (zh) * | 2015-09-29 | 2017-04-06 | 康朴生物医药技术（上海）有限公司 | 一种药物组合物及其应用 |
| KR20250070139A (ko) * | 2016-05-04 | 2025-05-20 | 썬 파마슈티칼 인더스트리즈 인코포레이티드 | 중수소화된 jak 저해제를 이용한 탈모 장애의 치료 |
| EP3476850B1 (en) | 2016-07-25 | 2024-12-11 | Shenzhen TargetRx, Inc. | Substituted boric acid compound, pharmaceutical composition comprising same, and application thereof |
| GB201907871D0 (en) * | 2019-06-03 | 2019-07-17 | Small Pharma Ltd | Therapeutic compositions |
| WO2021142395A1 (en) * | 2020-01-10 | 2021-07-15 | Consynance Therapeutics, Inc. | Therapeutic combinations of drugs and methods of using them |
| EP3902541B1 (en) * | 2020-06-02 | 2022-09-14 | Small Pharma Ltd | Therapeutic compositions comprising deuterated or partially deuterated n,n-dimethyltryptamine compounds |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PT1966202E (pt) * | 2005-12-13 | 2012-01-03 | Incyte Corp | Pirrolo[2,3-b] pirimidinas e pirrolo[2,3-b]piridinas substituídas com heteroarilo como inibidores de janus quinase |
| MX354212B (es) * | 2010-03-10 | 2018-02-19 | Incyte Corp | Derivados de piperidin-4-il azetidina como inhibidores de janus cinasa 1 (jak1). |
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2013
- 2013-12-17 JP JP2013259713A patent/JP6367545B2/ja active Active
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2018172421A (ja) * | 2018-07-05 | 2018-11-08 | コンサート ファーマシューティカルズ インコーポレイテッド | ルキソリチニブの重水素化誘導体 |
Also Published As
| Publication number | Publication date |
|---|---|
| JP2015117185A (ja) | 2015-06-25 |
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