JP6367545B2 - ルキソリチニブの重水素化誘導体 - Google Patents
ルキソリチニブの重水素化誘導体 Download PDFInfo
- Publication number
- JP6367545B2 JP6367545B2 JP2013259713A JP2013259713A JP6367545B2 JP 6367545 B2 JP6367545 B2 JP 6367545B2 JP 2013259713 A JP2013259713 A JP 2013259713A JP 2013259713 A JP2013259713 A JP 2013259713A JP 6367545 B2 JP6367545 B2 JP 6367545B2
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- deuterium
- hydrogen
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- 0 CC1(*)C(*)([C@@](*)(C(*)(*)C#N)[n]2nc(*)c(-c3nc(*)nc4c3c(*)c(*)[n]4)c2*)C(*)(*)C(*)(*)C1(*)* Chemical compound CC1(*)C(*)([C@@](*)(C(*)(*)C#N)[n]2nc(*)c(-c3nc(*)nc4c3c(*)c(*)[n]4)c2*)C(*)(*)C(*)(*)C1(*)* 0.000 description 1
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- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2013259713A JP6367545B2 (ja) | 2013-12-17 | 2013-12-17 | ルキソリチニブの重水素化誘導体 |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2013259713A JP6367545B2 (ja) | 2013-12-17 | 2013-12-17 | ルキソリチニブの重水素化誘導体 |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2018128417A Division JP6830460B2 (ja) | 2018-07-05 | 2018-07-05 | ルキソリチニブの重水素化誘導体 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2015117185A JP2015117185A (ja) | 2015-06-25 |
| JP2015117185A5 JP2015117185A5 (enExample) | 2017-02-09 |
| JP6367545B2 true JP6367545B2 (ja) | 2018-08-01 |
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2013259713A Active JP6367545B2 (ja) | 2013-12-17 | 2013-12-17 | ルキソリチニブの重水素化誘導体 |
Country Status (1)
| Country | Link |
|---|---|
| JP (1) | JP6367545B2 (enExample) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2018172421A (ja) * | 2018-07-05 | 2018-11-08 | コンサート ファーマシューティカルズ インコーポレイテッド | ルキソリチニブの重水素化誘導体 |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IL310969A (en) * | 2015-06-30 | 2024-04-01 | Eiger Group Int Inc | Use of chloroquine and clemizole compounds for treatment of inflammatory and cancerous conditions |
| KR102053556B1 (ko) * | 2015-09-29 | 2020-01-08 | 강푸 바이오파마슈티칼즈 리미티드 | 약물 조성물 및 이의 응용 |
| HRP20241345T1 (hr) | 2016-05-04 | 2024-12-20 | Sun Pharmaceutical Industries, Inc. | Liječenje poremećaja gubitka kose deuteriranim inhibitorima jak |
| EP3476850B1 (en) * | 2016-07-25 | 2024-12-11 | Shenzhen TargetRx, Inc. | Substituted boric acid compound, pharmaceutical composition comprising same, and application thereof |
| GB201907871D0 (en) * | 2019-06-03 | 2019-07-17 | Small Pharma Ltd | Therapeutic compositions |
| AU2021206286A1 (en) * | 2020-01-10 | 2024-08-08 | Consynance Therapeutics, Inc. | Therapeutic combinations of drugs and methods of using them |
| EP3902541B1 (en) * | 2020-06-02 | 2022-09-14 | Small Pharma Ltd | Therapeutic compositions comprising deuterated or partially deuterated n,n-dimethyltryptamine compounds |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TWI630207B (zh) * | 2005-12-13 | 2018-07-21 | 英塞特控股公司 | 作為傑納斯激酶（ＪＡＮＵＳ ＫＩＮＡＳＥ）抑制劑之經雜芳基取代之吡咯并〔２，３-ｂ〕吡啶及吡咯并〔２，３-ｂ〕嘧啶 |
| EP3050882B1 (en) * | 2010-03-10 | 2018-01-31 | Incyte Holdings Corporation | Piperidin-4-yl azetidine derivatives as jak1 inhibitors |
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2013
- 2013-12-17 JP JP2013259713A patent/JP6367545B2/ja active Active
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2018172421A (ja) * | 2018-07-05 | 2018-11-08 | コンサート ファーマシューティカルズ インコーポレイテッド | ルキソリチニブの重水素化誘導体 |
Also Published As
| Publication number | Publication date |
|---|---|
| JP2015117185A (ja) | 2015-06-25 |
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