JP5318757B2 - 神経因性疼痛の治療のための、組み合わされたセロトニンおよびノルエピネフリン再取り込み阻害を有する４−［２−（４−メチルフェニルスルファニル）−フェニル］ピペリジンの結晶形 - Google Patents

神経因性疼痛の治療のための、組み合わされたセロトニンおよびノルエピネフリン再取り込み阻害を有する４−［２−（４−メチルフェニルスルファニル）−フェニル］ピペリジンの結晶形 Download PDF

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JP5318757B2
JP5318757B2 JP2009514643A JP2009514643A JP5318757B2 JP 5318757 B2 JP5318757 B2 JP 5318757B2 JP 2009514643 A JP2009514643 A JP 2009514643A JP 2009514643 A JP2009514643 A JP 2009514643A JP 5318757 B2 JP5318757 B2 JP 5318757B2
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pain
compound
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addition salt
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JP2009539890A (ja
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バンク−アンデルセン・ベニー
ファルト・アンドレ
ステンスベル・ティネ・ブリュアン
ミラー・ジルケ
ロペス・デ・ディエゴ・ヘイディ
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ハー・ルンドベック・アクチエゼルスカベット
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    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
    • C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D211/20—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms
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JP2009514643A 2006-06-16 2007-06-15 神経因性疼痛の治療のための、組み合わされたセロトニンおよびノルエピネフリン再取り込み阻害を有する４−［２−（４−メチルフェニルスルファニル）−フェニル］ピペリジンの結晶形 Expired - Fee Related JP5318757B2 (ja)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US80500906P 2006-06-16 2006-06-16
US60/805,009 2006-06-16
DKPA200600816 2006-06-16
DKPA200600816 2006-06-16
DKPA200700423 2007-03-20
DKPA200700423 2007-03-20
PCT/DK2007/050076 WO2007144006A1 (en) 2006-06-16 2007-06-15 Crystalline forms of 4- [2- (4-methylphenylsulfanyl) -phenyl] piperidine with combined serotonin and norepinephrine reuptake inhibition for the treatment of neuropathic pain

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JP2013122095A Division JP5650280B2 (ja) 2006-06-16 2013-06-10 神経因性疼痛の治療のための、組み合わされたセロトニンおよびノルエピネフリン再取り込み阻害を有する４−［２−（４−メチルフェニルスルファニル）−フェニル］ピペリジンの結晶形

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JP2009539890A JP2009539890A (ja) 2009-11-19
JP2009539890A5 JP2009539890A5 (enExample) 2011-08-04
JP5318757B2 true JP5318757B2 (ja) 2013-10-16

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JP2009514643A Expired - Fee Related JP5318757B2 (ja) 2006-06-16 2007-06-15 神経因性疼痛の治療のための、組み合わされたセロトニンおよびノルエピネフリン再取り込み阻害を有する４−［２−（４−メチルフェニルスルファニル）−フェニル］ピペリジンの結晶形
JP2013122095A Expired - Fee Related JP5650280B2 (ja) 2006-06-16 2013-06-10 神経因性疼痛の治療のための、組み合わされたセロトニンおよびノルエピネフリン再取り込み阻害を有する４−［２−（４−メチルフェニルスルファニル）−フェニル］ピペリジンの結晶形

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US (4) US8299095B2 (enExample)
EP (1) EP2044020B1 (enExample)
JP (2) JP5318757B2 (enExample)
AU (1) AU2007260356B2 (enExample)
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MX2008016008A (es) * 2006-06-16 2009-01-16 Lundbeck & Co As H Formas cristalinas de 4-[2-(4-metilfenilsulfonil)-fenil] piperidina con inhibicion combinada de la recaptacion de serotonina y norepinefrina para el tratamiento del dolor neuropatico.
MY150647A (en) 2006-06-16 2014-02-14 Lundbeck & Co As H 1-[2-(2,4-dimethylphenylsulfanyl)-phenyl] piperazine as a compound with combined serotonin reuptake, 5-ht3 and 5-ht1a activity for the treatment of cognitive impairment
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IL195310A0 (en) 2009-08-03
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US20090264465A1 (en) 2009-10-22
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US8299095B2 (en) 2012-10-30
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US20150073018A1 (en) 2015-03-12
US20130190352A1 (en) 2013-07-25
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